NCT01448707

Brief Summary

The purpose of this study is to compare the efficacy, safety and tolerability of darunavir/ritonavir 800/100 mg monotherapy with a triple combination therapy containing darunavir/ritonavir 800/100 mg and 2 nucleoside/nucleotide reverse transcriptase inhibitors (N\[t\]RTIs) in approximately 260 Human Immunodeficiency Virus-1 (HIV-1) infected patients who have been on Highly Active AntiRetroviral Therapy (HAART) medication and have a plasma Viral Load below 50 copies/mL for at least 48 weeks. Also the changes in neurocognitive function will be compared throughout the study.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
274

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Mar 2012

Typical duration for phase_3

Geographic Reach
13 countries

34 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 2, 2011

Completed
4 months until next milestone

First Posted

Study publicly available on registry

October 7, 2011

Completed
5 months until next milestone

Study Start

First participant enrolled

March 15, 2012

Completed
2.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 11, 2014

Completed
9 months until next milestone

Study Completion

Last participant's last visit for all outcomes

March 18, 2015

Completed
9 months until next milestone

Results Posted

Study results publicly available

December 3, 2015

Completed
Last Updated

November 27, 2017

Status Verified

October 1, 2017

Enrollment Period

2.2 years

First QC Date

June 2, 2011

Results QC Date

October 30, 2015

Last Update Submit

October 23, 2017

Conditions

Keywords

Darunavir (DRV)TMC114PrezistaHIVvirologic responseneurocognitive function

Outcome Measures

Primary Outcomes (1)

  • Virologic Response (Food Drug and Administration [FDA] Snapshot, Switch = Failure)

    The percentage of participants who have plasma human immunodeficiency virus type-1 (HIV-1) ribonucleic acid (RNA) levels \<50 copies/milliliters \[mL\] after 48 weeks of follow-up. Switch = Failure is defined as switch in background nucleoside/nucleotide reverse transcriptase inhibitors (N\[t\]RTIs) not permitted by the trial protocol or plasma HIV-1 RNA assessment closest to target date of the analysis time point window (44-52 weeks) and next/confirmation of Plasma HIV-1 RNA in the analysis time point window above the threshold or discontinuation for any other reason.

    Week 48

Secondary Outcomes (6)

  • Virologic Response (Food Drug and Administration [FDA] Snapshot, Switch = Failure)

    Week 96

  • Virologic Response (FDA Snapshot, Switch Included)

    Week 48 and 96

  • Change From Baseline in Global Neurocognitive Performance z-Score

    Baseline, Week 48 and 96

  • Time to Loss of Virologic Response

    Baseline up to Week 96 or early withdrawal

  • Number of Participants Reporting Treatment-Emergent Phenotypic Drug Resistance

    At Weeks 48 and 96

  • +1 more secondary outcomes

Study Arms (2)

Darunavir monotherapy

EXPERIMENTAL

Darunavir (DRV) + ritonavir (rtv): 2 tablets DRV 400 mg should be taken together with 1 tablet rtv 100 mg within 30 minutes after a meal. Following the primary efficacy analysis after Week 48, patients who entered the study with a nadir CD4+ count of \<200 cells/μL will also receive 2 N\[t\]RTIs (ie, triple therapy) as soon as possible

Drug: DarunavirDrug: Ritonavir

Triple therapy containing darunavir

ACTIVE COMPARATOR

Darunavir (DRV) + ritonavir (rtv) + 2 N\[t\]RTIs: 2 tablets DRV 400 mg should be taken together with 1 tablet rtv 100 mg within 30 minutes after a meal in combination with 2 N\[t\]RTIs (an investigator-selected dual combination of either abacavir (ABC), lamivudine (3TC), zidovudine (AZT), tenofovir disoproxil fumarate (TDF) or emtricitabine (FTC)

Drug: DarunavirDrug: Ritonavir

Interventions

Darunavir (DRV): type = exact number, unit = mg, number = 800, form = tablet, route = oral use

Darunavir monotherapyTriple therapy containing darunavir

ritonavir (rtv): type = exact number, unit = mg, number = 100, form = tablet, route = oral use

Darunavir monotherapyTriple therapy containing darunavir

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • HIV-1 infection
  • receiving HAART for at least 48 weeks
  • Have at least 2 documented plasma HIV-1 RNA \<50 copies/mL, and no HIV-1 RNA \>=50 copies/mL in the 48 weeks prior to the screening
  • Be taking the same antiretroviral (ARV) combination for at least 8 weeks before screening
  • Have the preference, together with the physician, to change the current HAART regimen for reasons of simplification and/or toxicity

You may not qualify if:

  • Has a history of virologic failure defined as 2 consecutive plasma HIV-1 RNA \>500 copies/mL while on previous or current antiretroviral therapy
  • Has a history of any primary PI mutations
  • Has clinical or laboratory evidence of significantly decreased hepatic function or decompensation, irrespective of liver enzyme levels (liver insufficiency)
  • Is diagnosed with acute viral hepatitis at screening or before Baseline 1
  • Is co-infected with hepatitis B

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (34)

Unknown Facility

Graz, Austria

Location

Unknown Facility

Vienna, Austria

Location

Unknown Facility

Antwerp, Belgium

Location

Unknown Facility

Brussels, Belgium

Location

Unknown Facility

Ghent, Belgium

Location

Unknown Facility

Copenhagen, Denmark

Location

Unknown Facility

Hvidovre, Denmark

Location

Unknown Facility

Bobigny, France

Location

Unknown Facility

Bondy, France

Location

Unknown Facility

Dijon, France

Location

Unknown Facility

Paris, France

Location

Unknown Facility

Berlin, Germany

Location

Unknown Facility

Bonn, Germany

Location

Unknown Facility

Cologne, Germany

Location

Unknown Facility

Frankfurt, Germany

Location

Unknown Facility

Hanover, Germany

Location

Unknown Facility

Budapest, Hungary

Location

Unknown Facility

Dublin, Ireland

Location

Unknown Facility

Galway, Ireland

Location

Unknown Facility

Beersheba, Israel

Location

Unknown Facility

Ramat Gan, Israel

Location

Unknown Facility

Tel Aviv, Israel

Location

Unknown Facility

Warsaw, Poland

Location

Unknown Facility

Badalona, Spain

Location

Unknown Facility

Barcelona, Spain

Location

Unknown Facility

Córdoba, Spain

Location

Unknown Facility

Granada, Spain

Location

Unknown Facility

Madrid, Spain

Location

Unknown Facility

Stockholm, Sweden

Location

Unknown Facility

Sankt Gallen, Switzerland

Location

Unknown Facility

Zurich, Switzerland

Location

Unknown Facility

Brighton, United Kingdom

Location

Unknown Facility

London, United Kingdom

Location

Unknown Facility

Manchester, United Kingdom

Location

Related Publications (1)

  • Girard PM, Antinori A, Arribas JR, Ripamonti D, Bicer C, Netzle-Sveine B, Hadacek B, Moecklinghoff C. Week 96 efficacy and safety of darunavir/ritonavir monotherapy vs. darunavir/ritonavir with two nucleoside reverse transcriptase inhibitors in the PROTEA trial. HIV Med. 2017 Jan;18(1):5-12. doi: 10.1111/hiv.12386. Epub 2016 Jun 9.

MeSH Terms

Conditions

Acquired Immunodeficiency SyndromeInfectionsVirus Diseases

Interventions

DarunavirRitonavir

Condition Hierarchy (Ancestors)

HIV InfectionsBlood-Borne InfectionsCommunicable DiseasesSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsSlow Virus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

SulfonamidesAmidesOrganic ChemicalsCarbamatesAcids, AcyclicCarboxylic AcidsSulfonesSulfur CompoundsFuransHeterocyclic Compounds, 1-RingHeterocyclic CompoundsThiazolesAzoles

Results Point of Contact

Title
EMEA Medical Affairs Program Lead
Organization
Janssen Research & Development, LLC

Study Officials

  • Janssen-Cilag International NV Clinical Trial

    Janssen-Cilag International NV

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 2, 2011

First Posted

October 7, 2011

Study Start

March 15, 2012

Primary Completion

June 11, 2014

Study Completion

March 18, 2015

Last Updated

November 27, 2017

Results First Posted

December 3, 2015

Record last verified: 2017-10

Locations