NCT01434498

Brief Summary

This is a Phase 2 Randomized, Double-Blind, Placebo-Controlled Study of GS-5885, GS-9451, Tegobuvir and Ribavirin; GS-5885, GS-9451 and Tegobuvir; GS-5885, GS-9451 and Ribavirin in Interferon Ineligible or Intolerant Subjects with Chronic Genotype 1a or 1b HCV Infection.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
163

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Sep 2011

Shorter than P25 for phase_2

Geographic Reach
3 countries

50 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2011

Completed
8 days until next milestone

First Submitted

Initial submission to the registry

September 9, 2011

Completed
6 days until next milestone

First Posted

Study publicly available on registry

September 15, 2011

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2013

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2013

Completed
Last Updated

December 20, 2013

Status Verified

November 1, 2013

Enrollment Period

1.3 years

First QC Date

September 9, 2011

Last Update Submit

November 26, 2013

Conditions

Keywords

Hepatitis CHCVRapid Virologic ResponseSustained Virologic ResponseDirect Acting AntiviralCombination TherapyTegobuvirTreatment naĂ¯veHCV RNAPolymerase inhibitorProtease inhibitorInterferon intolerantInterferon ineligibleGS-9190GS-9451GS-5885

Outcome Measures

Primary Outcomes (2)

  • Safety and Tolerability

    To evaluate safety and tolerability of combination therapy with GS-5885, GS-9451, tegobuvir and ribavirin or GS-5885, GS-9451 and tegobuvir or GS-5885, GS-9451 and ribavirin. Safety will be assessed during the study through the reporting of adverse events, clinical laboratory tests, physical examinations, vital signs and 12-lead ECGs at various time points during the study.

    Through 24 weeks of off-treatment follow-up

  • Antiviral Activity

    To evaluate antiviral efficacy as measured by sustained virologic response (defined as HCV RNA \< lower limit of quantitation 24-weeks post-treatment) of combination therapy with GS-5885, GS-9451, tegobuvir and ribavirin or GS-5885, GS-9451 and tegobuvir or GS-5885, GS-9451 and ribavirin.

    Through 24 weeks of off-treatment follow-up

Secondary Outcomes (2)

  • Viral Dynamics

    Through 10 days of therapy

  • Composite (or Profile) of Pharmacokinetics

    predose, 1, 2, 3, 4, 6, 8, 10, 12 and 24 hours post-dose

Study Arms (3)

Arm 1

ACTIVE COMPARATOR

GS-5885, GS-9451, tegobuvir (GS-9190), and Copegus® for 24 weeks

Drug: GS-5885 tabletDrug: GS-9451 tabletDrug: tegobuvir capsuleDrug: ribavirin tablet

Arm 2

ACTIVE COMPARATOR

GS-5885, GS-9451, tegobuvir (GS-9190), and a placebo matching ribavirin for 24 weeks

Drug: GS-5885 tabletDrug: GS-9451 tabletDrug: tegobuvir capsuleDrug: placebo matching ribavirin tablet

Arm 3

ACTIVE COMPARATOR

GS-5885, GS-9451, a placebo matching tegobuvir, and Copegus® for 24 weeks

Drug: GS-5885 tabletDrug: GS-9451 tabletDrug: ribavirin tabletDevice: placebo matching tegobuvir capsule

Interventions

GS-5885 tablet, 90 mg, QD

Arm 1Arm 2Arm 3

GS-9451 tablet, 200 mg QD

Arm 1Arm 2Arm 3

tegobuvir capsule, 30 mg BID

Arm 1Arm 2

ribavirin tablet (weight based: 1000 mg/day \<75 kg; 1200 mg/day ≥ 75 kg) divided twice daily (BID)

Arm 1Arm 3

placebo matching ribavirin tablet, BID

Arm 2

placebo matching tegobuvir capsule, BID

Arm 3

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Adult subjects 18 and older with chronic HCV infection
  • Liver biopsy results (performed no more than 3 years prior to Screening) indicating the absence of cirrhosis
  • Monoinfection with HCV genotype 1a or 1b
  • Interferon ineligible or intolerant
  • Body mass index (BMI) between 18 and 40 kg/m2
  • Use of highly effective contraception methods if female of childbearing potential or sexually active male
  • Screening laboratory values within defined thresholds
  • Has not been exposed to any investigational drug or device within 30 days of the Screening visit
  • Able to comply with the dosing instructions for study drug administration and able to complete the study schedule of assessments

You may not qualify if:

  • Prior treatment of HCV with any direct-acting antiviral (whether approved or experimental)
  • Decompensated liver disease or cirrhosis
  • Co-infection with human immunodeficiency virus (HIV), hepatitis B virus (HBV), or another HCV genotype
  • History of difficulty with blood collection and/or poor venous access
  • Pregnant or nursing female or male with pregnant female partner
  • Chronic liver disease of a non-HCV etiology
  • Suspicion of hepatocellular carcinoma
  • Clinically-relevant drug abuse

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (50)

California Liver Institute

Beverly Hills, California, 90211, United States

Location

SCTI Research Foundation Liver Center

Coronado, California, 92118, United States

Location

Scripps Clinic

La Jolla, California, 92037, United States

Location

University of California, San Diego

La Jolla, California, 92161, United States

Location

Kaiser Permanente Medical Center

Los Angeles, California, 90027, United States

Location

Lightsource Medical

Los Angeles, California, 90036, United States

Location

Medical Associates Research Group, Inc.

San Diego, California, 92123, United States

Location

Kaiser Permanente

San Diego, California, 92154, United States

Location

California Pacific Medical Center

San Francisco, California, 94115, United States

Location

University of Colorado

Aurora, Colorado, 80045, United States

Location

University of Miami, Center for Liver Diseases

Miami, Florida, 33136, United States

Location

Orlando Immunology Center (ACH)

Orlando, Florida, 32803-1851, United States

Location

Gastrointestinal Specialists of Georgia, PC

Marietta, Georgia, 30060, United States

Location

Indianapolis Gastroenterology Research Foundation

Indianapolis, Indiana, 46237, United States

Location

University of Kansas Medical Center

Kansas City, Kansas, 66160, United States

Location

Johns Hopkins University

Lutherville, Maryland, 21093, United States

Location

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

Location

Beth Israel Deconess Medical Center

Boston, Massachusetts, 02215, United States

Location

The Research Institute

Springfield, Massachusetts, 01105, United States

Location

Henry Ford Health System

Novi, Michigan, 48377, United States

Location

Saint Michael's Medical Center

Newark, New Jersey, 07102, United States

Location

Weill Cornell Medical College

New York, New York, 10021, United States

Location

Asheville Gastroenterology Associates, P.A.

Asheville, North Carolina, 28801, United States

Location

University of North Carolina at Chapel Hill

Chapel Hill, North Carolina, 27599, United States

Location

University of Pennsylvania

Philadelphia, Pennsylvania, 19104, United States

Location

Thomas Jefferson University Hospital

Philadelphia, Pennsylvania, 19107, United States

Location

University Gastroenterology

Providence, Rhode Island, 02905, United States

Location

Gastro One

Germantown, Tennessee, 38138, United States

Location

The North Texas Research Institute

Arlington, Texas, 76012, United States

Location

The University of Texas Medical Branch

Galveston, Texas, 77555, United States

Location

The University of Texas Health Sciences Center at Houston

Houston, Texas, 77030, United States

Location

Alamo Medical Research

San Antonio, Texas, 78215, United States

Location

Inova Fairfax Hospital Center for Liver Diseases

Falls Church, Virginia, 22042, United States

Location

Bon Secours St. Mary's Hospital of Richmond, Inc.

Newport News, Virginia, 23602, United States

Location

Digestive and Liver Disease Specialists

Norfolk, Virginia, 23502, United States

Location

Virginia Mason Medical Center

Seattle, Washington, 98101, United States

Location

University of Calgary

Calgary, Alberta, T2N 4Z6, Canada

Location

University Of Alberta Hospital

Edmonton, Alberta, T6G 2C8, Canada

Location

University of Alberta

Edmonton, Alberta, T6G 2X8, Canada

Location

Gordon & Leslie Diamond Health Care Centre

Vancouver, British Columbia, V5Z 1M9, Canada

Location

University of British Columbia

Vancouver, British Columbia, V6Z 2C9, Canada

Location

GIRI GI Research Institute

Vancouver, British Columbia, V6Z 2K5, Canada

Location

University of Manitoba

Winnipeg, Manitoba, R3E 3P4, Canada

Location

London Health Sciences Centre

London, Ontario, N6A 5A5, Canada

Location

The Ottawa Hospital

Ottawa, Ontario, K1H 8L6, Canada

Location

Toronto General Hospital, University Health Network

Toronto, Ontario, M5G 2C4, Canada

Location

Toronto General Hospital, University Health Network

Toronto, Ontario, M5G 2N2, Canada

Location

Toronto Western Hospital

Toronto, Ontario, M5T2S8, Canada

Location

Hospital Saint-Luc DU CHUM

Montreal, Quebec, H2X3J4, Canada

Location

Clinical Research Puerto Rico Inc

San Juan, 00909-1711, Puerto Rico

Location

MeSH Terms

Conditions

Hepatitis C

Interventions

ledipasvirGS-9451tegobuvirRibavirin

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsHepatitis, Viral, HumanVirus DiseasesFlaviviridae InfectionsRNA Virus InfectionsHepatitisLiver DiseasesDigestive System Diseases

Intervention Hierarchy (Ancestors)

RibonucleosidesNucleosidesNucleic Acids, Nucleotides, and Nucleosides

Study Officials

  • John McNally, PhD

    Gilead Sciences

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 9, 2011

First Posted

September 15, 2011

Study Start

September 1, 2011

Primary Completion

January 1, 2013

Study Completion

January 1, 2013

Last Updated

December 20, 2013

Record last verified: 2013-11

Locations