NCT01401985

Brief Summary

A Single-Blind, Pilot Study to Determine the Tolerability and Safety of TD-1211 in Subjects with Opioid-Induced Constipation

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
95

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Oct 2011

Shorter than P25 for phase_2

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

July 19, 2011

Completed
7 days until next milestone

First Posted

Study publicly available on registry

July 26, 2011

Completed
2 months until next milestone

Study Start

First participant enrolled

October 1, 2011

Completed
7 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2012

Completed
3 months until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2012

Completed
Last Updated

May 25, 2021

Status Verified

May 1, 2021

Enrollment Period

7 months

First QC Date

July 19, 2011

Last Update Submit

May 20, 2021

Conditions

Keywords

Opioid induced constipationOICConstipationOpioid side effectsmorphine induced constipation

Outcome Measures

Primary Outcomes (1)

  • Safety and tolerability of TD-1211

    14 days

Secondary Outcomes (1)

  • Complete spontaneous bowel movements (CSBM); Spontaneous bowel movements (SBM)

    Weekly assessments throughout Treatment Period

Study Arms (6)

Cohort 1

EXPERIMENTAL

5 mg TD-1211 once daily for 4 days followed by 10 mg for 14 days

Drug: TD-1211

Cohort 2

EXPERIMENTAL

5 mg TD-1211 once daily for 4 days followed by 15 mg for 14 days

Drug: TD-1211

Cohort 3

EXPERIMENTAL

5 mg TD-1211 once daily for 2 days followed by 10 mg for 14 days

Drug: TD-1211

Cohort 4

EXPERIMENTAL

5 mg TD-1211 once daily for 2 days followed by 15 mg for 14 days

Drug: TD-1211

Cohort 5

EXPERIMENTAL

2 mg TD-1211 once daily for 14 days

Drug: TD-1211Drug: Placebo

Cohort 6

EXPERIMENTAL

2.5 mg TD-1211 every 6 hours for 14 days

Drug: TD-1211Drug: Placebo

Interventions

Capsules

Cohort 1Cohort 2Cohort 3Cohort 4Cohort 5Cohort 6

Capsules

Cohort 5Cohort 6

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • stable dose of opioids for at least 12 weeks before screening visit
  • less than or equal to 5 spontaneous bowel movements for a 2 week period and experiencing at least one other symptom of constipation
  • willing to stop laxatives and other bowel treatments; rescue laxative allowed

You may not qualify if:

  • Clinically significant condition or illness (other than the condition for which the pain medication was prescribed)
  • Have participated in another clinical trial of an investigational drug 30 days prior to screening
  • History of cancer treatment except adequately treated localized skin cancer within 5 years of screening
  • History of chronic constipation prior to opioid therapy
  • Females who are pregnant or breast feeding
  • Have any condition that may affect drug absorption (e.g. previous GI surgery)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Theravance Biopharma Investigational Site

Pasadena, California, 91105, United States

Location

MeSH Terms

Conditions

Opioid-Induced ConstipationConstipation

Interventions

3-(8-(2-(cyclohexylmethyl(2,3-dihydroxypropionyl)amino)ethyl)-8-azabicyclo(3.2.1)oct-3-yl)benzamide

Condition Hierarchy (Ancestors)

Signs and Symptoms, DigestiveSigns and SymptomsPathological Conditions, Signs and SymptomsNarcotic-Related DisordersSubstance-Related DisordersChemically-Induced DisordersMental Disorders

Study Officials

  • Medical Monitor

    Theravance Biopharma

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NON RANDOMIZED
Masking
SINGLE
Who Masked
PARTICIPANT
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

July 19, 2011

First Posted

July 26, 2011

Study Start

October 1, 2011

Primary Completion

May 1, 2012

Study Completion

August 1, 2012

Last Updated

May 25, 2021

Record last verified: 2021-05

Data Sharing

IPD Sharing
Will not share

Theravance Biopharma, Inc. will not be sharing individual de-identified participant data or other relevant study documents.

Locations