NCT01319019

Brief Summary

This study is primarily designed to assess the dose response, dose interval, efficacy and safety of three once daily (QD) doses (100mcg, 400mcg and 800mcg) and three twice daily (BID) doses (100mcg, 200mcg and 400mcg,) of GSK961081 administered via DISKUS™ for 28 days in subjects with moderate/severe COPD versus placebo. Salmeterol 50mcg BID is included in the study as an active comparator.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
437

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Dec 2010

Shorter than P25 for phase_2

Geographic Reach
9 countries

49 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

December 1, 2010

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

March 3, 2011

Completed
18 days until next milestone

First Posted

Study publicly available on registry

March 21, 2011

Completed
5 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2011

Completed
Last Updated

December 1, 2016

Status Verified

November 1, 2016

Enrollment Period

9 months

First QC Date

March 3, 2011

Last Update Submit

November 30, 2016

Conditions

Keywords

lung functionbronchodilatorCOPD, dose response, dosing interval, efficacy, safety, PD, PK

Outcome Measures

Primary Outcomes (1)

  • Change in FEV1 from baseline in pre-dose AM trough.

    Pre-dose change in AM FEV1 on day 29 vs baseline . (defined as the mean values recorded 11 and 12 hours after the PM dose on day 28)

    28 Day

Secondary Outcomes (1)

  • Weighted Mean and Serial FEV1 at multiple timepoints

    28 Days

Study Arms (8)

GSK961081 100 mcg QD

EXPERIMENTAL
Drug: GSK961081

GSK961081 100mcg BD

EXPERIMENTAL
Drug: GSK961081

GSK961081 200mcg QD

EXPERIMENTAL
Drug: GSK961081

GSK961081 400mcg QD

EXPERIMENTAL
Drug: GSK961081

GSK961081 400mcg BD

EXPERIMENTAL
Drug: GSK961081

GSK961081 800mcg QD

EXPERIMENTAL
Drug: GSK961081

Salmeterol 50mcg BD

ACTIVE COMPARATOR
Drug: Salmeterol

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

Comparison of different doses and dosing regimens of the drug

GSK961081 100 mcg QDGSK961081 100mcg BDGSK961081 200mcg QDGSK961081 400mcg BDGSK961081 400mcg QDGSK961081 800mcg QD

Positive control

Salmeterol 50mcg BD

Placebo arm

Placebo

Eligibility Criteria

Age40 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Outpatient Subjects
  • Subjects who give their signed and dated informed consent to participate
  • or more years of age, inclusive, at Visit 1
  • Male or females
  • Subjects with an established clinical history of COPD
  • Current or previous cigarette smokers with a history of ≥ 10 pack-years of cigarette smoking
  • Subjects with the following liver function test values:
  • Subjects with a measured post-salbutamol FEV1/FVC ratio of \< 0.70 at Visit 1 (Screening).
  • Subjects with a measured post-salbutamol FEV1 30-70% of predicted normal values

You may not qualify if:

  • Women who are pregnant or lactating or are planning to become pregnant during the study.
  • Current diagnosis of asthma
  • Other significant respiratory disorders besides COPD, including alpha-1 deficiency
  • Previous lung resection surgery
  • Significant abnormalities in chest x-ray presentation
  • Hospitalization for a COPD exacerbation within 12 weeks prior screening
  • Use of oral corticosteroids or antibiotics for COPD or antibiotics for a lower respiratory tract infection within 6 weeks
  • Any significant disease that would put subject at risk through study participation
  • BMI greater than 35
  • Pacemaker
  • Significantly abnormal ECG, clinical lab finding (including Hepatitis B or C)
  • Cancer
  • Allergy or hypersensitivity to beta adrenergic receptor-agonist, sympathomimetic, anticholinergic/anti-muscarinic receptor antagonist, or inhaler excipients
  • Diseases that would contra-indicate the use of anticholinergics
  • Use of sysemic corticosteroids within 6 weeks of screening
  • +12 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (49)

GSK Investigational Site

Tallinn, 10138, Estonia

Location

GSK Investigational Site

Tallinn, 13419, Estonia

Location

GSK Investigational Site

Tallinn, 13619, Estonia

Location

GSK Investigational Site

Tartu, 51014, Estonia

Location

GSK Investigational Site

Frankfurt am Main, Hesse, 60596, Germany

Location

GSK Investigational Site

Gelnhausen, Hesse, 63571, Germany

Location

GSK Investigational Site

Dresden, Saxony, 01307, Germany

Location

GSK Investigational Site

Lübeck, Schleswig-Holstein, 23552, Germany

Location

GSK Investigational Site

Berlin, State of Berlin, 10367, Germany

Location

GSK Investigational Site

Berlin, State of Berlin, 10717, Germany

Location

GSK Investigational Site

Berlin, State of Berlin, 10787, Germany

Location

GSK Investigational Site

Almelo, 7609 PP, Netherlands

Location

GSK Investigational Site

Breda, 4819 EV, Netherlands

Location

GSK Investigational Site

Eindhoven, 5623 EJ, Netherlands

Location

GSK Investigational Site

Hoorn, 1624 NP, Netherlands

Location

GSK Investigational Site

Veldhoven, 5504 DB, Netherlands

Location

GSK Investigational Site

Zutphen, 7207 AE, Netherlands

Location

GSK Investigational Site

Bucharest, 020125, Romania

Location

GSK Investigational Site

Bucharest, 050159, Romania

Location

GSK Investigational Site

Iași, 700115, Romania

Location

GSK Investigational Site

Timișoara, 300310, Romania

Location

GSK Investigational Site

Moscow, 105 077, Russia

Location

GSK Investigational Site

Moscow, 115446, Russia

Location

GSK Investigational Site

Saint Petersburg, 197022, Russia

Location

GSK Investigational Site

Tomsk, 634001, Russia

Location

GSK Investigational Site

Yekaterinburg, 620109, Russia

Location

GSK Investigational Site

Bratislava, 826 06, Slovakia

Location

GSK Investigational Site

Košice, 040 01, Slovakia

Location

GSK Investigational Site

Nitra, 949 01, Slovakia

Location

GSK Investigational Site

Nové Zámky, 940 01, Slovakia

Location

GSK Investigational Site

Zvolen, 960 01, Slovakia

Location

GSK Investigational Site

Bellville, 7530, South Africa

Location

GSK Investigational Site

Durban, 4001, South Africa

Location

GSK Investigational Site

Gatesville, 7764, South Africa

Location

GSK Investigational Site

Mowbray, 7700, South Africa

Location

GSK Investigational Site

Panorama, 7500, South Africa

Location

GSK Investigational Site

Tygerberg, 7505, South Africa

Location

GSK Investigational Site

Boden, SE-961 64, Sweden

Location

GSK Investigational Site

Gothenburg, SE-413 45, Sweden

Location

GSK Investigational Site

Lund, SE-221 85, Sweden

Location

GSK Investigational Site

Stockholm, SE-171 76, Sweden

Location

GSK Investigational Site

Dnipropetrovsk, 49074, Ukraine

Location

GSK Investigational Site

Ivano-Frankivsk, 76018, Ukraine

Location

GSK Investigational Site

Kharkiv, 61124, Ukraine

Location

GSK Investigational Site

Kiev, 03680, Ukraine

Location

GSK Investigational Site

Kyiv, 03115, Ukraine

Location

GSK Investigational Site

Kyiv, 03680, Ukraine

Location

GSK Investigational Site

Simferopol, 95043, Ukraine

Location

GSK Investigational Site

Vinnytsia, 21029, Ukraine

Location

Related Publications (1)

  • Wielders PL, Ludwig-Sengpiel A, Locantore N, Baggen S, Chan R, Riley JH. A new class of bronchodilator improves lung function in COPD: a trial with GSK961081. Eur Respir J. 2013 Oct;42(4):972-81. doi: 10.1183/09031936.00165712. Epub 2013 Feb 21.

    PMID: 23429913BACKGROUND

Related Links

MeSH Terms

Conditions

Pulmonary Disease, Chronic Obstructive

Interventions

batefenterolSalmeterol Xinafoate

Condition Hierarchy (Ancestors)

Lung Diseases, ObstructiveLung DiseasesRespiratory Tract DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

AlbuterolEthanolaminesAmino AlcoholsAlcoholsOrganic ChemicalsAminesPhenethylaminesEthylamines

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 3, 2011

First Posted

March 21, 2011

Study Start

December 1, 2010

Primary Completion

September 1, 2011

Study Completion

September 1, 2011

Last Updated

December 1, 2016

Record last verified: 2016-11

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Individual Participant Data Set (115032)Access
Annotated Case Report Form (115032)Access
Dataset Specification (115032)Access
Clinical Study Report (115032)Access
Informed Consent Form (115032)Access
Study Protocol (115032)Access
Statistical Analysis Plan (115032)Access

Locations