NCT01314898

Brief Summary

24-hr urinary sodium/potassium ratio will be a sensitive biomarker of antimineralocorticoid activity. The dose-response relationship of the antimineralocorticoid activity of PF-03882845 can be established following single oral doses.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
12

participants targeted

Target at below P25 for phase_1 healthy-volunteers

Timeline
Completed

Started Mar 2011

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2011

Completed
2 days until next milestone

First Submitted

Initial submission to the registry

March 3, 2011

Completed
12 days until next milestone

First Posted

Study publicly available on registry

March 15, 2011

Completed
3 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2011

Completed
Last Updated

July 6, 2011

Status Verified

July 1, 2011

Enrollment Period

3 months

First QC Date

March 3, 2011

Last Update Submit

July 5, 2011

Conditions

Keywords

Single dosecross-overactive-controlplacebo controlantimineralocorticoid activity

Outcome Measures

Primary Outcomes (1)

  • Twenty-four hour urinary Na/K ratio (AUC(0-24)).

    0-24hr postdose per period

Secondary Outcomes (4)

  • Area Under the Curve(AUClast) from the time of dosing to the last data point of PF-03882845.

    0-24 hr post dose per period

  • Time of Maximum concentration(Tmax) of PF-03882845.

    0-24 hr post dose per period

  • Maximum concentration (Cmax) of PF-03882845.

    0-24 hr post dose per period

  • Safety and tolerability: Physical examinations, adverse event monitoring, clinical safety laboratory assessments, vital sign measurements and 12-lead ECGs.

    2 months

Study Arms (1)

Treatment

EXPERIMENTAL
Drug: 3 mg PF-03882845Drug: 10 mg PF-03882845Drug: 30 mg PF-03882845Drug: 100 mg PF-03882845Drug: Spironolactone

Interventions

3 mg PF-03882845, single oral dose

Treatment

10 mg PF-03882845, single oral dose

Treatment

30 mg PF-03882845, single oral dose

Treatment

100 mg PF-03882845, single oral dose

Treatment

100 mg spironolactone, single oral dose

Treatment

Eligibility Criteria

Age18 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Male and/or female healthy volunteers, age 18 to 55 years. Females must be of non-childbearing potential.
  • Body Mass Index (BMI) of 17.5 to 30.5 kg/m2; and a total body weight \>50 kg (110 lbs).
  • Subjects who are willing and able to comply with scheduled visits, treatment plan, laboratory tests, diet restrictions and other trial procedures.

You may not qualify if:

  • Subjects with a supine BP \>140 mm Hg systolic or \>90 mm Hg diastolic or \<100 mm Hg systolic or \<60 mm Hg diastolic based on the average of the triplicate
  • Serum potassium \>=5.1 mmol/L or \<3.5 mmol/L at screening, confirmed by a single repeat if deemed necessary.
  • Estimated GFR \<60 mL/min/1.73 m2 using the Cockcroft-Gault formula measurement of the individual parameters following at least 5 minutes of rest at Screening.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Pfizer Investigational Site

New Haven, Connecticut, 06511, United States

Location

Related Links

MeSH Terms

Interventions

(3S,3aR)-2-(3-chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo(g)indazole-7-carboxylic acidSpironolactone

Intervention Hierarchy (Ancestors)

LactonesOrganic ChemicalsPregnenesPregnanesSteroidsFused-Ring CompoundsPolycyclic Compounds

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

March 3, 2011

First Posted

March 15, 2011

Study Start

March 1, 2011

Primary Completion

June 1, 2011

Study Completion

June 1, 2011

Last Updated

July 6, 2011

Record last verified: 2011-07

Locations