NCT01200394

Brief Summary

PF-00489791 is an inhibitor of phosphodiesterase type 5. Our hypothesis is that PF-00489791 will enhance the relaxation of blood vessels within the kidney and so reduce blood pressure, improving renal function.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
256

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Dec 2010

Geographic Reach
14 countries

154 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 10, 2010

Completed
3 days until next milestone

First Posted

Study publicly available on registry

September 13, 2010

Completed
3 months until next milestone

Study Start

First participant enrolled

December 1, 2010

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2013

Completed
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2013

Completed
5.6 years until next milestone

Results Posted

Study results publicly available

March 12, 2019

Completed
Last Updated

March 12, 2019

Status Verified

February 1, 2019

Enrollment Period

2.6 years

First QC Date

September 10, 2010

Results QC Date

January 3, 2019

Last Update Submit

February 18, 2019

Conditions

Keywords

Diabetic nephropathychronic kidney diseasePF-00489791phosphodiesterasePDE5

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Urinary Albumin Creatinine Ratio (UACR) at Week 12

    UACR was ratio of albumin measured in urine (milligram) to creatinine measured in urine (millimole), reported in units milligram per millimole (mg/mmol). A decrease in UACR may be associated with improved renal and cardiovascular function. The mean values of the 3 consecutive first morning void urine samples (obtained 2 days prior to \[Day 5, 6 of Week 12\], and with last sample collected on the morning of scheduled clinic visit \[Day 7 of Week 12\]) were used to determine UACR at the scheduled clinic visit. The mean values of the 3 consecutive first morning void urine samples obtained at screening were used to determine baseline UACR.

    Baseline, Week 12 (Day 5, 6, 7)

Secondary Outcomes (9)

  • Change From Baseline in Urinary Albumin Creatinine Ratio (UACR) at Week 3, 6 and 16

    Baseline, Week 3 (Day 5, 6, 7), Week 6 (Day 5, 6, 7), Week 16 (Day 5, 6, 7)

  • Change From Baseline in Urinary Protein Creatinine Ratio (UPCR) at Week 3, 6, 12, and 16

    Baseline, Week 3 (Day 5, 6, 7), Week 6 (Day 5, 6, 7), Week 12 (Day 5, 6, 7), Week 16 (Day 5, 6, 7)

  • Change From Baseline in Estimated Glomerular Filtration Rate (eGFR) at Week 3, 6, 12, and 16

    Baseline, Week 3, 6, 12, 16 (follow-up)

  • Systolic, Diastolic and Mean Blood Pressure at Week 0, 3, 6, 12, and 16

    Week 0, 3, 6, 12, 16 (follow-up)

  • Change From Baseline in Serum Creatinine Concentration at Week 3, 6, 12, and 16

    Baseline, Week 3, 6, 12, 16 (follow-up)

  • +4 more secondary outcomes

Other Outcomes (6)

  • Change From Baseline in Plasma Glycosylated Hemoglobin (HbA1c) Level at Week 12 and 16

    Baseline, Week 12, 16 (follow-up)

  • Number of Participants With Vital Signs Abnormalities

    Baseline up to Week 16 (follow-up)

  • Number of Participants With Edema and Fluid Overload

    Week 0, 3, 6, 12, 16 (follow-up)

  • +3 more other outcomes

Study Arms (2)

PF-00489791

EXPERIMENTAL
Drug: PF-00489791

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

Tablet, 20 mg once daily for 12 weeks

PF-00489791

Tablet, placebo once daily for 12 weeks

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male or female subjects greater than or equal to 18 years. Female subjects must be of non-child bearing potential.
  • Clinical diagnosis of type 2 diabetes together with stages 3a, 3b or 4 CKD, based on an eGFR of 25-59 mL/min/1.73m2.
  • Evidence of persistent, overt albuminuria; defined as a UACR greater than or equal to 300 mg/g (greater than or equal to 33.9 mg/mmol) for greater than 3 months.

You may not qualify if:

  • Subjects with CKD resulting from type 1 diabetes or non-diabetic CKD.
  • Subjects with poorly controlled diabetes mellitus, defined as HbA1C \>9%.
  • Subjects on combination ACE inhibitor/ARB therapy.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (160)

Saadat Ansari Internal Medicine

Huntsville, Alabama, 35801, United States

Location

The Office of Iqbal Saeed MD, LLC

Huntsville, Alabama, 35805, United States

Location

AKDHC Medical Research Services, LLC*

Glendale, Arizona, 85306, United States

Location

Southwest Clinical Research Institute, LLC

Tempe, Arizona, 85281, United States

Location

Southwest Clinical Research Institute, LLC

Tempe, Arizona, 85284, United States

Location

North America Research Institute

Azusa, California, 91702, United States

Location

North American Research Institute / California Kidney Specialist

Azusa, California, 91702, United States

Location

Citrus Dialysis Center

Covina, California, 91723, United States

Location

California Institute of Renal Research

La Mesa, California, 91942, United States

Location

Capital Nephrology Clinical Research

Sacramento, California, 95825, United States

Location

California Kidney Specialists

San Dimas, California, 91773, United States

Location

American Institute of Research

Whittier, California, 90602, United States

Location

Whittier Internal Medicine Nephrology Medical Group

Whittier, California, 90602, United States

Location

North Valley Nephrology

Yuba City, California, 95991, United States

Location

Riverside Clinical Research

Edgewater, Florida, 32132, United States

Location

Palm Springs Research Institute

Hialeah, Florida, 33012, United States

Location

ASA Clinical Research, LLC

Jupiter, Florida, 33458, United States

Location

Lakeview Medical Research

Summerfield, Florida, 34491, United States

Location

Rockdale Medical Research Associates

Conyers, Georgia, 30094, United States

Location

Renal Physicians of Georgia

Macon, Georgia, 31217, United States

Location

Boise Kidney and Hypertension Institute

Meridian, Idaho, 83642, United States

Location

Chicago Clinical Research Institute, Inc.

Chicago, Illinois, 60616, United States

Location

Associates in Nephrology, SC

Evergreen Park, Illinois, 60805, United States

Location

Research by Design, LLC

Evergreen Park, Illinois, 60805, United States

Location

RenalCare Associates

Peoria, Illinois, 61603, United States

Location

Investigative Clinical Research of Indiana, LLC

Elwood, Indiana, 46036, United States

Location

Kansas Nephrology Research Institute, LLC

Wichita, Kansas, 67214, United States

Location

Four Rivers Clinical Research, Inc.

Paducah, Kentucky, 42003, United States

Location

Crescent City Clinical Research Center

Metairie, Louisiana, 70006, United States

Location

Northwest Louisiana Nephrology

Shreveport, Louisiana, 71101, United States

Location

Biolab Research, LLC

Rockville, Maryland, 20852, United States

Location

Alzohaili Medical Consultants

Dearborn, Michigan, 48124, United States

Location

Apex Medical Research, AMR, Inc.

Flint, Michigan, 48504, United States

Location

Apex Medical Research, MI, Inc.

Flint, Michigan, 48504, United States

Location

Clinical Research Consultants, LLC

Kansas City, Missouri, 64111, United States

Location

Lincoln Nephrology and Hypertension

Lincoln, Nebraska, 68510, United States

Location

Nebraska Nephrology Research Institute, LLC - Research Management, Inc.

Lincoln, Nebraska, 68510, United States

Location

Alliance Against Diabetes

Las Vegas, Nevada, 89101, United States

Location

Clinical Research Consortium

Las Vegas, Nevada, 89119, United States

Location

Jacobi Medical Center - Department of Medicine - Nephrology

The Bronx, New York, 10461, United States

Location

Mountain Kidney and Hypertension Associates, PA

Asheville, North Carolina, 28801, United States

Location

Trial Management Associates

Wilmington, North Carolina, 28401, United States

Location

Lake Medical Research

Willoughby Hills, Ohio, 44094, United States

Location

Northeast Clinical Research Center, LLC

Bethlehem, Pennsylvania, 18017, United States

Location

Preferred Primary Care Physicians, Inc.

Uniontown, Pennsylvania, 15401, United States

Location

Columbia Nephrology Associates, PA

Columbia, South Carolina, 29203, United States

Location

Carolina Nephrology, PA

Greenville, South Carolina, 29605, United States

Location

Palmetto Nephrology, PA

Orangeburg, South Carolina, 29118, United States

Location

South Carolina Nephrology & Hypertension Ctr, Inc

Orangeburg, South Carolina, 29118, United States

Location

South Carolina Nephrology and Hypertension Center

Orangeburg, South Carolina, 29118, United States

Location

Central Texas Kidney Associates

Austin, Texas, 78751, United States

Location

Research Management, Inc.

Austin, Texas, 78751, United States

Location

Diagnostic Clinic of Houston, PA

Houston, Texas, 77004, United States

Location

Houston Nephrology Research

Houston, Texas, 77024, United States

Location

Research Across America

Houston, Texas, 77054, United States

Location

Renal Associates, PA

San Antonio, Texas, 78215, United States

Location

San Antonio Kidney Disease Center Physicians Group, P.L.L.C.

San Antonio, Texas, 78229, United States

Location

Nephrology Associates of Northern Virginia, Inc.

Fairfax, Virginia, 22033, United States

Location

Nephrology Specialists, P.C.

Mechanicsville, Virginia, 23116, United States

Location

Clinical Research Associates of Tidewater

Norfolk, Virginia, 23507, United States

Location

Renal Remission & Hypertension Consultants, PLLC

Bremerton, Washington, 98310, United States

Location

Sound Medical Research

Port Orchard, Washington, 98366, United States

Location

Renal Remission and Hypertension Clinic

Silverdale, Washington, 98383, United States

Location

Renal Research Practice

Gosford, New South Wales, 2250, Australia

Location

John Hunter Hospital

Newcastle, New South Wales, 2305, Australia

Location

Department of Nephrology

New Lambton, Newcastle, 2305, Australia

Location

Pharmacy Department

New Lambton, Newcastle, 2305, Australia

Location

Melbourne Renal Research Group

Reservoir, Victoria, 3073, Australia

Location

Sheldon M Chumir Health Centre

Calgary, Alberta, T2N 0X7, Canada

Location

University of Alberta Hospital

Edmonton, Alberta, T6G 2B7, Canada

Location

Entralogix Clincal Research Inc.

Brampton, Ontario, L6Z 4N5, Canada

Location

Entralogix Clinical Research Inc.

Brampton, Ontario, L6Z 4N5, Canada

Location

London Health Sciences Centre

London, Ontario, N6A 5A5, Canada

Location

Entralogix Clinical Research Inc.

Oakville, Ontario, L6J 3M5, Canada

Location

N/A - formerly with Entralogix SMO

Toronto, Ontario, M4C 5T2, Canada

Location

Sunnybrook Health Sciences Center

Toronto, Ontario, M4N 3M5, Canada

Location

Centre de sante et de services sociaux champlain-Charles-Le Moyne

Greenfield Park, Quebec, J4V 2H1, Canada

Location

Centre de Dialyse de Bois de Boulogne

Montreal, Quebec, H3M 3E3, Canada

Location

Hopital de Sacre Coeur de Montreal

Montreal, Quebec, H4J 1C5, Canada

Location

Saskatoon Nephrology Group, Nurses Redisence

Saskatoon, Saskatchewan, S7M 2Z1, Canada

Location

Saskatoon Nephrology Group, Nurses Residence

Saskatoon, Saskatchewan, S7M 2Z1, Canada

Location

Saskatoon Nephrology Group

Saskatoon, Saskatchewan, S7M 2Z1, Canada

Location

Aarhus Universitetshospital (Aarhus Sygehus)

Aarhus, 8000, Denmark

Location

Rigshospitalet

Copenhagen Oe, 2100, Denmark

Location

Steno Diabetes Center

Gentofte Municipality, 2820, Denmark

Location

Queen Mary Hospital

Hong Kong, Hong Kong

Location

Division of Nephrology, Dept. of Medicine

Pokfulam, Hong Kong

Location

Division of Nephrology

Pokfulam, Hong Kong

Location

ICON Clinical Research

Quarry Bay, Hong Kong

Location

Prince of Wales Hospital

Shatin, N.T. 0, Hong Kong

Location

Apollo Hospitals

Hyderabad, Andhra Pradesh, 500096, India

Location

Gujarat Kidney Foundation

Ahmedabad, Gujarat, 380 007, India

Location

Shrushrut Clinical Research Association

Ahmedabad, Gujarat, 380 013, India

Location

P. D. Hinduja National Hospital and Medical Research Centre

Mumbai, Maharashtra, 400016, India

Location

Pfizer Centre

Mumbai, Maharashtra, 400102, India

Location

Deenanath Mangeshkar Hospital & Research Centre

Pune, Maharashtra, 411 004, India

Location

Diabetes Care and Research Centre

Pune, Maharashtra, 411 011, India

Location

KE.M Hospital Research Centre

Pune, Maharashtra, 411 011, India

Location

King Edward Memorial Hospital

Pune, Maharashtra, 411 011, India

Location

Jehangir Clinical Development Centre Pvt. Ltd.

Pune, Maharashtra, 411001, India

Location

Universiti Sains Malaysia

Kota Bharu, Kelantan, 16150, Malaysia

Location

Unit Kajian Klinikal, Hospital Universiti Sains Malaysia

Kubang Kerian, Kelantan, 16150,, Malaysia

Location

Hospital Taiping

Taiping, Perak, 34000, Malaysia

Location

Clinical Research Centre, Hospital Pulau Pinang

George Town, Pulau Pinang, 10990, Malaysia

Location

Hospital Pulau Pinang

George Town, Pulau Pinang, 10990, Malaysia

Location

Nephrology Clinic, Queen Elizabeth Hospital

Kota Kinabalu, Sabah, 88586, Malaysia

Location

Unit Hemodialisis, Hospital Serdang

Kajang, Selangor, 43000, Malaysia

Location

ICLE SC

Guadalajara, Jalisco, 44600, Mexico

Location

Comite Mexicano para la Prevencion de la Osteoporosis, A.C.

Mexico City, Mexico City, 06100, Mexico

Location

Instituto Nacional de Ciencias Medicas y Nutricion Salvador Zubiran (INCMNSZ)

Tlalpan, Mexico City, 14000, Mexico

Location

Hospital Central Dr Ignacio Morones Prieto Unidad Regional de Osteoporosis

San Luis Potosí City, San Luis Potosí, 78240, Mexico

Location

Hospital Angeles del Pedregal

Angeles Del Pedregal Cp., 10700, Mexico

Location

NZOZ "DIAGNOMED" S.C., Poradnia Nefrologiczna

Bielsko-Biala, 43-300, Poland

Location

Samodzielny Publiczny Szpital Kliniczny im Andrzeja Mieleckiego

Katowice, 40-027, Poland

Location

NZOZ PS "Medica"

Lublin, 20-538, Poland

Location

Centrum Medyczne "Osteomed" NZOZ, Lecznica Specjalistow

Warsaw, 02-256, Poland

Location

Centrum Medyczne "OSTEOMED" NZOZ

Warsaw, 02-256, Poland

Location

Centrum Medyczne "Osteomed"

Warsaw, 02-256, Poland

Location

Centrum Medyczne OSTEOMED NZOZ; Lecznica Specjalistaw

Warsaw, 02-256, Poland

Location

Miedzyleski Szpital Specjalistyczny w Warszawie

Warsaw, 4749, Poland

Location

SPZOZ Akademicki Szpital Kliniczny im. J. Mikulicza - Radeckiego

Wroclaw, 50-556, Poland

Location

Clinical Center of Serbia Institute for Endocrinology, Diabetes and Metabolic Diseases

Belgrade, 11 000, Serbia

Location

Clinic for Nephrology, Military Medical Academy

Belgrade, 11000, Serbia

Location

Clinical Center of Serbia

Belgrade, 11000, Serbia

Location

Clinical Hospital Center "Zvezdara"

Belgrade, 11000, Serbia

Location

Clinical Hospital Center Zvezdara

Belgrade, 11000, Serbia

Location

Clinic for Endocrinology, Clinical Center Nis

Niš, 18000, Serbia

Location

FNsP Bratislava, Nemocnica Stare Mesto

Bratislava, 813 69, Slovakia

Location

Nemocnice s poliklinikami n.o.

Levice, 934 01, Slovakia

Location

Fakultna nemocnica s poliklinikou J.A.Reimana Presov

Prešov, 081 81, Slovakia

Location

Vseobecna nemocnica Rimavska Sobota

Rimavská Sobota, 979 12, Slovakia

Location

Worthwhile Clinical Trials (WWCT), Lake View Hospital

Benoni, Gauteng, 1500, South Africa

Location

Dr. George Mukhari Hospital -University of Limpopo

Pretoria, Gauteng, 0204, South Africa

Location

Wits Clinical research

Johannesburg, Gauteng- South Africa, 2096, South Africa

Location

Centre for Diabetes and Endocrinology

Durban, KwaZulu-Natal, 4091, South Africa

Location

Latros International

Bloemfontein, 9301, South Africa

Location

Division of Nephrology and Hypertension, E13 Renal Unit

Cape Town, 7925, South Africa

Location

St Augustine's Hospital

Durban, 4001, South Africa

Location

Centre for Diabetes and Endocrinology

Durban, 4091, South Africa

Location

Centre for Diabetes and Endocrinology

Houghton, Johannesburg, 2198, South Africa

Location

Intercare Parow Medical and Dental Centre

Parow, 7500, South Africa

Location

Medi-Clinic Heart Hospital (Pretoria Heart Hospital)

Pretoria, 132, South Africa

Location

Pharmacy

Seongnam-si, Gyeonggi-do, 463-707, South Korea

Location

Seoul National University Bundang Hospital

Seongnam-si, Gyeonggi-do, 463-707, South Korea

Location

Clinical Trial Pharmacy

Seongnam-si, 463-707, South Korea

Location

Seoul National University Hospital

Seoul, 110-744, South Korea

Location

Samsung Medical Center, Department of Pharmacy

Seoul, 135-710, South Korea

Location

Samsung Medical Center,Sungkyunkwan Univ School of Medicine

Seoul, 135-710, South Korea

Location

Samsung Medical Center/Division of Nephrology

Seoul, 135-710, South Korea

Location

Boramae Medical Center/Division of Nephrology

Seoul, 156-707, South Korea

Location

SMG-SNU Boramae Medical Center

Seoul, 156-707, South Korea

Location

Sahlgrenska University Hospital Njurmottagningen

Gothenburg, 413 45, Sweden

Location

A+ Science City site

Stockholm, 111 57, Sweden

Location

Akademiska Sjukhuset

Uppsala, 751 85, Sweden

Location

Doncaster Royal Infirmary

Doncaster, South Yorkshire, DN2 5LT, United Kingdom

Location

Research Offices (5th Floor)

Coventry, CV2 2DX, United Kingdom

Location

University of Edinburgh

Edinburgh, EH16 4TJ, United Kingdom

Location

The Royal London Hospital Whitechapel

London, E1 1BB, United Kingdom

Location

Guy's and St Thomas' Foundation Trust

London, SE1 9RT, United Kingdom

Location

Northern General Hospital Campus

Sheffield, S5 7AU, United Kingdom

Location

Related Links

MeSH Terms

Conditions

Diabetic NephropathiesRenal Insufficiency, Chronic

Interventions

PF-00489791

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesDiabetes ComplicationsDiabetes MellitusEndocrine System DiseasesRenal InsufficiencyChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Results Point of Contact

Title
Pfizer ClinicalTrials.gov Call Center
Organization
Pfizer, Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 10, 2010

First Posted

September 13, 2010

Study Start

December 1, 2010

Primary Completion

July 1, 2013

Study Completion

August 1, 2013

Last Updated

March 12, 2019

Results First Posted

March 12, 2019

Record last verified: 2019-02

Data Sharing

IPD Sharing
Will share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

More information

Locations