NCT01193478

Brief Summary

The primary purpose of this study is to evaluate the safety, tolerability, pharmacokinetics and activity of escalating, multiple, oral doses of GS-5885 in subjects with chronic genotype 1 Hepatitis C Virus (HCV) infection. Each participant in the study will be sequestered in the clinic for the initial 5 days of the study.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
71

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started Aug 2010

Geographic Reach
1 country

13 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2010

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

August 31, 2010

Completed
2 days until next milestone

First Posted

Study publicly available on registry

September 2, 2010

Completed
4 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2011

Completed
11 months until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2011

Completed
Last Updated

January 21, 2013

Status Verified

January 1, 2013

Enrollment Period

5 months

First QC Date

August 31, 2010

Last Update Submit

January 18, 2013

Conditions

Keywords

Hepatitis CHCV RNAmultiple ascending doseNS5AGS-5885chronic genotype 1 HCV infection

Outcome Measures

Primary Outcomes (2)

  • Number of subjects reporting an adverse event or experiencing a laboratory abnormality

    Safety and tolerability assessments will be performed up to Study Day 14 following administration of multiple doses of GS-5885 or placebo for 3 days

  • Antiviral activity measures: measured by change in plasma HCV RNA levels form baseline

    Assessed up to Study Day 14 following administration of multiple doses of GS-5885 or placebo for 3 days

Secondary Outcomes (2)

  • Measure of GS-5885 plasma concentration over time

    Assessed up to Study Day 14 following administration of multiple doses of GS-5885 or placebo for 3 days

  • Emergence of viral resistance

    Up to 48 weeks following Study Day 14

Study Arms (6)

Cohort 1

ACTIVE COMPARATOR

GS-5885 (3 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Cohort 2

ACTIVE COMPARATOR

GS-5885 (10 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Cohort 3

ACTIVE COMPARATOR

GS-5885 (30 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Cohort 4

ACTIVE COMPARATOR

GS-5885 ( up to 90 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Cohort 5

ACTIVE COMPARATOR

GS-5885 (up to 90 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Cohort 6 (optional)

ACTIVE COMPARATOR

GS-5885 (up to 90 mg), once daily or matching placebo, once daily

Drug: GS-5885Drug: Placebo

Interventions

tablet, oral, 3 mg once daily for 3 days

Cohort 1

tablet, oral, once daily for 3 days

Cohort 1

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Chronically infected with HCV genotype 1
  • HCV treatment-naïve
  • Not co-infected with HIV or HBV
  • HCV RNA viral load of at least 100,000 IU/mL
  • BMI 19 to 35 kg/m2
  • Subject agrees to use highly effective contraception methods if female of childbearing potential or sexually active male.

You may not qualify if:

  • History of clinically-significant illness or any other major medical disorder that may interfere with subject treatment, assessment or compliance with the protocol
  • Decompensated liver disease or cirrhosis or evidence of hepatocellular carcinoma
  • Serological evidence of co-infection with human immunodeficiency virus (HIV), hepatitis B virus (HBV), or another HCV genotype
  • Subjects with known, current use of amphetamines and/or cocaine; subjects taking methadone or buprenorphine (opioid replacement therapy) or ongoing alcohol abuse

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (13)

Unknown Facility

Anaheim, California, 92801, United States

Location

Unknown Facility

Cypress, California, 90630, United States

Location

Unknown Facility

National City, California, 91950, United States

Location

Unknown Facility

Washington D.C., District of Columbia, 20010, United States

Location

Unknown Facility

DeLand, Florida, 32720, United States

Location

Unknown Facility

Miami, Florida, 33169, United States

Location

Unknown Facility

Orlando, Florida, 32809, United States

Location

Unknown Facility

St Louis, Missouri, 63104, United States

Location

Unknown Facility

Portland, Oregon, 97239, United States

Location

Unknown Facility

Philadelphia, Pennsylvania, 19139, United States

Location

Unknown Facility

Houston, Texas, 77030, United States

Location

Unknown Facility

San Antonio, Texas, 78215, United States

Location

Unknown Facility

Tacoma, Washington, 98418, United States

Location

Related Publications (1)

  • Wong KA, Worth A, Martin R, Svarovskaia E, Brainard DM, Lawitz E, Miller MD, Mo H. Characterization of Hepatitis C virus resistance from a multiple-dose clinical trial of the novel NS5A inhibitor GS-5885. Antimicrob Agents Chemother. 2013 Dec;57(12):6333-40. doi: 10.1128/AAC.02193-12. Epub 2013 Jul 22.

MeSH Terms

Conditions

Hepatitis C

Interventions

ledipasvir

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsHepatitis, Viral, HumanVirus DiseasesFlaviviridae InfectionsRNA Virus InfectionsHepatitisLiver DiseasesDigestive System Diseases

Study Officials

  • Diana Brainard, MD

    Gilead Sciences

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 31, 2010

First Posted

September 2, 2010

Study Start

August 1, 2010

Primary Completion

January 1, 2011

Study Completion

December 1, 2011

Last Updated

January 21, 2013

Record last verified: 2013-01

Locations