NCT01071850

Brief Summary

Evaluate the efficacy, safety, and tolerability of multiple doses of ASP1941 compared to placebo over 12 weeks of therapy in adult patients with type 2 diabetes mellitus.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
412

participants targeted

Target at P75+ for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started Mar 2010

Geographic Reach
5 countries

59 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 18, 2010

Completed
1 day until next milestone

First Posted

Study publicly available on registry

February 19, 2010

Completed
12 days until next milestone

Study Start

First participant enrolled

March 3, 2010

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 11, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 11, 2011

Completed
Last Updated

May 22, 2025

Status Verified

May 1, 2025

Enrollment Period

1.1 years

First QC Date

February 18, 2010

Last Update Submit

May 20, 2025

Conditions

Keywords

ASP1941MetforminType 2 diabetesdiabetes

Outcome Measures

Primary Outcomes (1)

  • Mean change from baseline in Hemoglobin A1c (HbA1c)

    12 weeks

Secondary Outcomes (3)

  • Mean change from baseline in fasting plasma glucose (FPG)

    12 weeks

  • Proportion of subjects achieving target goal of HbA1c <7.0%

    12 weeks

  • Proportion of subjects achieving target goal of HbA1c <6.5%

    12 weeks

Study Arms (6)

ASP1941 lowest dose

EXPERIMENTAL

oral tablet

Drug: ipragliflozin

ASP1941 low dose

EXPERIMENTAL

oral tablet

Drug: ipragliflozin

ASP1941 high dose

EXPERIMENTAL

oral tablet

Drug: ipragliflozin

ASP1941 highest dose

EXPERIMENTAL

oral tablet

Drug: ipragliflozin

Metformin

ACTIVE COMPARATOR

oral tablet

Drug: Metformin

Placebo

PLACEBO COMPARATOR

oral tablet

Drug: Placebo

Interventions

oral tablet

Also known as: ASP1941
ASP1941 high doseASP1941 highest doseASP1941 low doseASP1941 lowest dose

oral tablet

Metformin

oral tablet

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subject has been diagnosed with type 2 diabetes
  • Subject has a HbA1c value between 6.8 and 9.5%
  • Subject has never, is not currently taking anti-diabetic medication OR is receiving a single anti- diabetic agent or low-doses two anti-diabetic medications and is willing to discontinue them during the study
  • Subject is on a stable diet and exercise program
  • Female subject is not pregnant and agrees to use an acceptable form of contraception throughout the duration of the study

You may not qualify if:

  • Subject has type 1 diabetes mellitus
  • Subject is using insulin therapy
  • Subject has a serum creatinine higher than upper limit of normal
  • Subject has an ALT and/or AST value higher than 3 times upper limit of normal or a total bilirubin value more than 2 times upper limit of normal
  • Subject has persistent, uncontrolled severe hypertension as indicated by a
  • systolic blood pressure \>180 mmHg or a diastolic blood pressure of
  • \>110mmHg
  • Subject has had significant cardiovascular disease such as myocardial infarction or a vascular intervention (e.g., angioplasty or stent) in the last 3 months
  • Subject is known to have hepatitis or be a carrier of hepatitis B surface
  • antigen, hepatitis C virus antibody or is known positive for HIV1 and/or
  • HIV2
  • Subject has a history of lactic acidosis
  • Subject has a history of drug and alcohol abuse/dependency within last 12
  • months
  • Subject has had a malignancy in the last 5 years, except for successfully
  • +4 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (59)

Parkway Medical Center

Birmingham, Alabama, 35215, United States

Location

Winston Technology Research, LLC

Haleyville, Alabama, 35565, United States

Location

Desert Clinical Research

Mesa, Arizona, 85213, United States

Location

Central Phoenix Medical Clinic

Phoenix, Arizona, 85020, United States

Location

Paul W. Davis, MD, PA

Pine Bluff, Arkansas, 71603, United States

Location

Clinical Innovations, Inc.

Costa Mesa, California, 92626, United States

Location

Del Rosario Medical Clinic, Inc

Huntington Park, California, 90255, United States

Location

Torrance Clinical Research

Lomita, California, 90717, United States

Location

San Diego Managed Care Group Clinical Research

San Diego, California, 92128, United States

Location

Expresscare Clinical Research

Colorado Springs, Colorado, 80909, United States

Location

PAB Clinical Research

Brandon, Florida, 33511, United States

Location

Clinical Therapeutics Corp.

Coral Gables, Florida, 33131, United States

Location

A.G.A Clinical Trials DBA Neostart Group

Hialeah, Florida, 33012, United States

Location

Suncoast Clinical Research

New Port Richey, Florida, 34652, United States

Location

CSRA Partners in Health, Inc.

Augusta, Georgia, 30909, United States

Location

Atlanta Vascular Research Foundation, Atlanta Cardiology & Primary Care P.C.

Tucker, Georgia, 30084, United States

Location

Cedar Crosse Research Center

Chicago, Illinois, 60607, United States

Location

APEX Medical Research, AMR, Inc

Chicago, Illinois, 60616, United States

Location

MediSphere Medical Research

Evansville, Indiana, 47714, United States

Location

Bay West Endocrinology

Towson, Maryland, 21204, United States

Location

Prism Research

Saint Paul, Minnesota, 55114, United States

Location

PMG Research of Charlotte, LLC

Charlotte, North Carolina, 28209, United States

Location

PMG Research of Salisbury, LLC

Salisbury, North Carolina, 28144, United States

Location

Rapid Medical Research

Cleveland, Ohio, 44122, United States

Location

Primecare of Southeastern Ohio, Inc.

Zanesville, Ohio, 43701, United States

Location

Integris Family Care

Yukon, Oklahoma, 73099, United States

Location

Willamette Valley Clinical Studies

Eugene, Oregon, 97404, United States

Location

Fleetwood Clinical Research

Fleetwood, Pennsylvania, 19522, United States

Location

Southeastern Research Associates, Inc.

Taylors, South Carolina, 29687, United States

Location

PMG Research of Bristol, LLC

Bristol, Tennessee, 37620, United States

Location

Holston Medical Group

Kingsport, Tennessee, 37660, United States

Location

Southwind Medical Specialist

Memphis, Tennessee, 38125, United States

Location

Punzi Medical Center

Carrollton, Texas, 75006, United States

Location

Corpus Christi Family Wellness Center

Corpus Christi, Texas, 78414, United States

Location

Excel Clinical Research, LLC

Houston, Texas, 77081, United States

Location

Cetero Research

San Antonio, Texas, 78229, United States

Location

Aspen Clinical Research

Orem, Utah, 84058, United States

Location

BIOMELAB

Barranquilla, Colombia

Location

Centro de Reumatologia y ortopedia

Barranquilla, Colombia

Location

Fundacion de Caribe para le Investigacion Biomedica

Barranquilla, Colombia

Location

Dexa Diad Servicios Medicos

Bogotá, Colombia

Location

School of Medicine University of Rosario

Bogotá, Colombia

Location

Fundacion Cardiovascular de Columbia

Floridablanca Santander, Colombia

Location

Diacon Hospital

Bangalore, 560010, India

Location

Hormone Care and Research Centre

Ghaziabad, 201002, India

Location

TOTALL Diabetes Hormone Institute Pvt.Ltd.

Indore, 452001, India

Location

S R Kalla Memorial Gastro & General Hospital

Jaipur, 302001, India

Location

Bride, Bharti Hospital

Karnāl, 132001, India

Location

Amrita Institute of Medical Sciences and Research Centre, AIMS

Kerala, 682041, India

Location

Unidad Metabólica y Cardiovascular, SC.

Cuernavaca, 62250, Mexico

Location

Instituto Jaliscience de Investigacion Clinica

Guadalajara, 44100, Mexico

Location

Torre Medica Providencia

Guadalajara, 44670, Mexico

Location

Medical Care and Research

Mérida, 97070, Mexico

Location

CEDIME, Instituto Vascular

Mérida, 97129, Mexico

Location

Hospital Universitario Dr. Eleuterio Gonzalez

Monterrey, 66460, Mexico

Location

Cebu Doctors' University Hospital

Cebu, 6000, Philippines

Location

St. Paul's Hospital

Iloilo City, 5000, Philippines

Location

Amang Rodriguez Memorial Medical Center

Marikina City, 1800, Philippines

Location

San Juan De Dios Hospital

Pasay, 1300, Philippines

Location

Related Publications (2)

  • Kashiwagi A, Shestakova MV, Ito Y, Noguchi M, Wilpshaar W, Yoshida S, Wilding JPH. Safety of Ipragliflozin in Patients with Type 2 Diabetes Mellitus: Pooled Analysis of Phase II/III/IV Clinical Trials. Diabetes Ther. 2019 Dec;10(6):2201-2217. doi: 10.1007/s13300-019-00699-8. Epub 2019 Oct 12.

  • Fonseca VA, Ferrannini E, Wilding JP, Wilpshaar W, Dhanjal P, Ball G, Klasen S. Active- and placebo-controlled dose-finding study to assess the efficacy, safety, and tolerability of multiple doses of ipragliflozin in patients with type 2 diabetes mellitus. J Diabetes Complications. 2013 May-Jun;27(3):268-73. doi: 10.1016/j.jdiacomp.2012.11.005. Epub 2012 Dec 29.

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Diabetes Mellitus

Interventions

ipragliflozinMetformin

Condition Hierarchy (Ancestors)

Glucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

BiguanidesGuanidinesAmidinesOrganic Chemicals

Study Officials

  • Medical Director

    Astellas Pharma Global Development

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 18, 2010

First Posted

February 19, 2010

Study Start

March 3, 2010

Primary Completion

April 11, 2011

Study Completion

April 11, 2011

Last Updated

May 22, 2025

Record last verified: 2025-05

Data Sharing

IPD Sharing
Will not share

Access to anonymized individual participant level data will not be provided for this trial. Further details on Astellas' data sharing policy can be found at https://www.clinicaltrials.astellas.com/transparency/.

Locations