NCT01008059

Brief Summary

To evaluate two paradigms for simultaneous assessment of hepatic and intestinal CYP3A activity.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
6

participants targeted

Target at below P25 for not_applicable

Timeline
Completed

Started Oct 2009

Longer than P75 for not_applicable

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

October 1, 2009

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

November 3, 2009

Completed
2 days until next milestone

First Posted

Study publicly available on registry

November 5, 2009

Completed
6.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 1, 2016

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2016

Completed
2.7 years until next milestone

Results Posted

Study results publicly available

May 17, 2019

Completed
Last Updated

May 17, 2019

Status Verified

May 1, 2019

Enrollment Period

6.9 years

First QC Date

November 3, 2009

Results QC Date

February 16, 2018

Last Update Submit

May 15, 2019

Conditions

Outcome Measures

Primary Outcomes (1)

  • Area Under the Curve of Alfentanil Concentration vs. Time Extrapolated to Infinity

    AUC(0-inf)

    9 hours

Study Arms (1)

Alfentanil

EXPERIMENTAL

Alfentanil (0.5-1 mg IV bolus) followed 3 hours later or simultaneously by 1-4 mg oral deuterium-labeled (d3) alfentanil on each study visit.

Drug: Alfentanil

Interventions

No drug treatment before alfentanil

Alfentanil

Eligibility Criteria

Age18 Years - 40 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Male or non-pregnant female, 18-40 yr. old
  • Good general health with no remarkable medical conditions such as liver, kidney, heart, or lung failure
  • BMI between 20-33
  • Provide informed consent

You may not qualify if:

  • Known history of liver or kidney disease
  • Use of prescription or non prescription medications, herbals or foods known to be metabolized by or affect CYP3A (including oral birth control medications)
  • Females who are pregnant or nursing
  • Known history of drug or alcohol addiction (prior or present addiction or treatment for addiction)
  • History of bradycardia
  • Respiratory rate \<10
  • History of significant pulmonary disease
  • History of pre-existing medical condition predisposing to respiratory depression
  • Systolic blood pressure \<100 mgHg and diastolic blood pressure \<70mmHg

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Washington University/Barnes Jewish Hospital

St Louis, Missouri, 63110, United States

Location

MeSH Terms

Interventions

Alfentanil

Intervention Hierarchy (Ancestors)

FentanylPiperidinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Results Point of Contact

Title
Evan D. Kharasch, MD PhD
Organization
Washington University

Study Officials

  • Evan D Kharasch, MD, PhD

    Washington University School of Medicine

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
Yes

Study Design

Study Type
interventional
Phase
not applicable
Allocation
NA
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
SINGLE GROUP
Sponsor Type
OTHER
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 3, 2009

First Posted

November 5, 2009

Study Start

October 1, 2009

Primary Completion

September 1, 2016

Study Completion

September 1, 2016

Last Updated

May 17, 2019

Results First Posted

May 17, 2019

Record last verified: 2019-05

Locations