NCT01006603

Brief Summary

This study will evaluate the efficacy and tolerability of saxagliptin compared to glimepiride in elderly patients with type 2 diabetes mellitus who have inadequate glycaemic control on metformin monotherapy.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
957

participants targeted

Target at P75+ for phase_4 type-2-diabetes-mellitus

Timeline
Completed

Started Oct 2009

Typical duration for phase_4 type-2-diabetes-mellitus

Geographic Reach
13 countries

131 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

October 1, 2009

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

October 31, 2009

Completed
3 days until next milestone

First Posted

Study publicly available on registry

November 3, 2009

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2012

Completed
1.5 years until next milestone

Results Posted

Study results publicly available

November 28, 2013

Completed
Last Updated

November 28, 2013

Status Verified

September 1, 2013

Enrollment Period

2.7 years

First QC Date

October 31, 2009

Results QC Date

June 12, 2013

Last Update Submit

September 27, 2013

Conditions

Keywords

Type 2 Diabetes Mellituselderly patientssaxagliptinrandomiseddouble-blind

Outcome Measures

Primary Outcomes (1)

  • Proportion of Patients Reaching HbA1c <7% After 52 Weeks of Treatment Without Confirmed or Severe Hypoglycaemia.

    Defined as obtained on or before the 8th day after the last dosing day, as determined by central laboratory. Safety analysis set. Confirmed hypoglycaemia defined as: any event defined as either a symptomatic event with blood glucose level \<3 mmol/L (\<54 mg/dL) and no need for external assistance, or an asymptomatic blood glucose measurement \<3 mmol/L (\<54 mg/dL). Major (or severe) hypoglycaemia defined as: symptomatic events requiring external assistance due to severe impairment in consciousness or behaviour, with or without blood glucose level \<3 mmol/L (\<54 mg/dL), but with prompt recovery after glucose or glucagon administration. These events may be associated with sufficient neuroglycopenia to induce seizure or coma. Plasma glucose measurements may not be available during such an event, but neurological recovery, attributable to the restoration of plasma glucose to normal, was considered sufficient evidence that the event was induced by a low plasma glucose concentration.

    From week 0 to week 52.

Secondary Outcomes (6)

  • Proportion of Patients Having Experienced at Least One Hypoglycaemic Event (Confirmed or Severe) Over the 52-week Double-blind Treatment Period.

    From week 0 to week 52.

  • Change From Baseline to Week 52 in HbA1c.

    From week 0 to week 52.

  • Proportion of Patients Achieving a Therapeutic Glycaemic Response at Week 52 Defined as HbA1c <7.0%

    From week 0 to week 52

  • Change From Baseline to Week 52 in Fasting Plasma Glucose (FPG)

    From week 0 to week 52

  • Change From Baseline to Week 52 in Insulin

    From week 0 to week 52

  • +1 more secondary outcomes

Study Arms (2)

1

EXPERIMENTAL

Saxagliptin 5 mg

Drug: Saxagliptin

2

ACTIVE COMPARATOR

Glimepiride 1 - 6 mg

Drug: Glimepiride

Interventions

5 mg, oral tablet, once daily

Also known as: Onglyza
1

1, 2, 3, 4 or 6 mg, oral encapsulated tablet, once daily

Also known as: Amaryl
2

Eligibility Criteria

Age65 Years+
Sexall
Healthy VolunteersNo
Age GroupsOlder Adult (65+)

You may qualify if:

  • Provision of informed consent prior to any study specific procedures
  • Established clinical diagnosis of type 2 diabetes. Treatment with a stable metformin monotherapy, for at least 8 weeks prior to Visit 1
  • HbA1c ≥7.0% and ≤9.0%

You may not qualify if:

  • Type 1 diabetes, history of diabetic ketoacidosis or hyperosmolar non-ketonic coma. Current use of any injectable or oral antihyperglycemic agent excluding metformin.
  • Renal impairment as defined by a creatinine clearance \<60 mL/min
  • Individuals who, in the opinion of the investigator, in which participation in this study may pose a significant risk to the patient and could render the patient unable to successfully complete the study

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (131)

Research Site

Feldbach, Austria

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Graz, Austria

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Salzburg, Austria

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Vienna, Austria

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Aalborg, Denmark

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Ans, Denmark

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Kjellerup, Denmark

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Kolding, Denmark

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Nørresundby, Denmark

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Roskilde, Denmark

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Roslev, Denmark

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Viborg, Denmark

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Viby J, Denmark

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Værløse, Denmark

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Lahti, Finland, Finland

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Vantaa, Finland, Finland

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Harjavalta, Finland

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Helsinki, Finland

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Kuopio, Finland

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Kuusankoski, Finland

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Oulu, Finland

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Seinäjoki, Finland

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Sipoo, Finland

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Tampere, Finland

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Turku, Finland

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Vimpeli, Finland

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Châtellerault, France

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La Rochelle, France

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La Seyne-sur-Mer, France

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Laval, France

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Seysses, France

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Strasbourg, France

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Tiercé, France

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Hamburg, Hamburg, Germany

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Augsburg, Germany

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Darmstadt, Germany

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Dresden, Germany

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Essen, Germany

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Gelnhausen, Germany

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Hamburg, Germany

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Magdeburg, Germany

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Mayen, Germany

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München, Germany

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Neumünster, Germany

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Nuremberg, Germany

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Pirna, Germany

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Ratzeburg, Germany

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Reinfeld, Germany

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Sulzbach, Germany

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Athens, Greece, Greece

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Athens, Greece

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Nikaia, Greece

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Thessaloniki, Greece

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Ács, Hungary

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Balatonfüred, Hungary

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Budapest, Hungary

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Érd, Hungary

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Gyöngyös, Hungary

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Komárom, Hungary

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Milan, MI, Italy

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Palermo, PA, Italy

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Padua, PD, Italy

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Pordenone, PN, Italy

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Reggio Emilia, RE, Italy

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Chieti, Italy

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Napoli, Italy

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Roma, Italy

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Viterbo, Italy

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Durango, Durango, Mexico

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Guadalajara, Jalisco, Mexico

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Monterrey, Nuevo León, Mexico

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Aksdal, Norway

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Ålesund, Norway

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Elverum, Norway

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Halden, Norway

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Hamar, Norway

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Kirkenær, Norway

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Kongsvinger, Norway

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Larvik, Norway

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Lierskogen, Norway

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Nordlenangen, Norway

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Oslo, Norway

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Røa, Norway

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Sandvika, Norway

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Skedsmokorset, Norway

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Svelvik, Norway

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Sørumsand, Norway

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Trondheim, Norway

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Ulset, Norway

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Seville, Andalusia, Spain

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Zamora, Castille and León, Spain

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A Coruña, Galicia, Spain

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Begonte (lugo), Galicia, Spain

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Getafe, Madrid, Spain

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Madrid, Madrid, Spain

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San Sebastián de los Reyes, Madrid, Spain

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Oviedo, Principality of Asturias, Spain

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Alicante, Valencia, Spain

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Jönköping, Sweden, Sweden

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Finspång, Sweden

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Gävle, Sweden

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Gothenburg, Sweden

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Jarfalla, Sweden

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Lessebo, Sweden

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Lund, Sweden

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Ödeshög, Sweden

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Piteå, Sweden

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Rättvik, Sweden

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Stockholm, Sweden

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Trollhättan, Sweden

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Västervik, Sweden

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Fowey, Cornwall, United Kingdom

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Nr Penzance, Cornwall, United Kingdom

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Penzance, Cornwall, United Kingdom

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Barnstaple, Devon, United Kingdom

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Plymouth, Devon, United Kingdom

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Annan, Dumfries and Galloway, United Kingdom

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Canterbury, Kent, United Kingdom

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Whitstable, Kent, United Kingdom

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Frome, Somerset, United Kingdom

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Bradford-on-Avon, Wiltshire, United Kingdom

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Trowbridge, Wiltshire, United Kingdom

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Ayrshire, United Kingdom

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Bath, United Kingdom

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Cumbernauld, United Kingdom

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Dundee, United Kingdom

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Hamilton, United Kingdom

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Middlesex, United Kingdom

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Motherwell, United Kingdom

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Somerset, United Kingdom

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Wellingborough, United Kingdom

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Related Publications (2)

  • Perl S, Cook W, Wei C, Ohman P, Hirshberg B. Effects of Glimepiride versus Saxagliptin on beta-Cell Function and Hypoglycemia: A Post Hoc Analysis in Older Patients with Type 2 Diabetes Inadequately Controlled with Metformin. Clin Ther. 2016 Dec;38(12):2578-2588. doi: 10.1016/j.clinthera.2016.10.006. Epub 2016 Nov 4.

  • Schernthaner G, Duran-Garcia S, Hanefeld M, Langslet G, Niskanen L, Ostgren CJ, Malvolti E, Hardy E. Efficacy and tolerability of saxagliptin compared with glimepiride in elderly patients with type 2 diabetes: a randomized, controlled study (GENERATION). Diabetes Obes Metab. 2015 Jul;17(7):630-8. doi: 10.1111/dom.12461. Epub 2015 Apr 7.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

saxagliptinglimepiride

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Results Point of Contact

Title
Boaz Hirshberg , MSD
Organization
AstraZeneca

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 4
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 31, 2009

First Posted

November 3, 2009

Study Start

October 1, 2009

Primary Completion

June 1, 2012

Study Completion

June 1, 2012

Last Updated

November 28, 2013

Results First Posted

November 28, 2013

Record last verified: 2013-09

Locations