NCT01004081

Brief Summary

The purpose of this study is to assess the efficacy, safety and tolerability of 2 dosing regimens of BIIB021 in combination with exemestane in women whose HR+ breast cancer had progressed following treatment with a nonsteroidal aromatase inhibitor (AI).

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
54

participants targeted

Target at P25-P50 for phase_2 breast-cancer

Timeline
Completed

Started Nov 2009

Shorter than P25 for phase_2 breast-cancer

Geographic Reach
4 countries

34 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 18, 2009

Completed
1 month until next milestone

First Posted

Study publicly available on registry

October 29, 2009

Completed
3 days until next milestone

Study Start

First participant enrolled

November 1, 2009

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2011

Completed
Last Updated

October 2, 2015

Status Verified

December 1, 2011

Enrollment Period

1.9 years

First QC Date

September 18, 2009

Last Update Submit

September 17, 2015

Conditions

Keywords

Cancer of BreastCancer of the Breast

Outcome Measures

Primary Outcomes (1)

  • The primary objective of this study is to assess the efficacy of 2 dosing regimens of BIIB021 in combination with exemestane in women whose HR+ breast cancer had progressed following treatment with a nonsteroidal AI.

    As specified in protocol

Secondary Outcomes (1)

  • The secondary objective of this study is to evaluate the safety and tolerability of BIIB021 in combination with exemestane in this study population.

    As specified in protocol

Study Arms (2)

BIIB021 BID + exemestane

EXPERIMENTAL

BIIB021 100 mg BID + exemestane 25 mg QD

Drug: BIIB021Drug: exemestane (Aromasin)

BIIB021 TIW + exemestane

EXPERIMENTAL

BIIB021 450 mg TIW + exemestane 25 mg QD

Drug: BIIB021Drug: exemestane (Aromasin)

Interventions

BID orally for 28 days

Also known as: CNF2024
BIIB021 BID + exemestane

Daily in tablet form for 28 days

Also known as: Aromasin
BIIB021 BID + exemestaneBIIB021 TIW + exemestane

Eligibility Criteria

Age18 Years+
Sexfemale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Age 18 years of age
  • Must have histologically or cytologically confirmed estrogen receptor- positive or progesterone receptor-positive, incurable, locally advanced, or metastatic breast cancer.
  • Must have disease progression during treatment with a nonsteroidal AI for locally advanced or metastatic disease, or relapse during treatment or within 12 months of discontinuation of treatment in the adjuvant setting.
  • Must be a postmenopausal female.
  • Must have measurable or evaluable disease.
  • Measurable disease is defined as \>=1 lesion with a diameter of \>=10 mm
  • Evaluable disease is defined as bone lesions evaluable by plain X ray, CT scan, or MRI. Lesions identified only by radionuclide bone scan are not allowed.
  • One prior chemotherapy regimen for advanced mBC is allowed.
  • Prior radiotherapy is allowed.
  • Must be able to swallow and retain oral medication.
  • ECOG performance status of \<=2
  • Required laboratory values
  • Plasma cortisol and adrenocorticotropic hormone (ACTH) levels that are not suggestive of adrenal insufficiency unless on replacement therapy for known adrenal insufficiency.

You may not qualify if:

  • HER2 overexpressing tumor.
  • History of central nervous system (CNS) metastasis.
  • Previous treatment with exemestane or treatment with an Hsp90 inhibitor.
  • Use of proton pump inhibitors.
  • Known history of or positive test result for hepatitis B or C or HIV.
  • History of gastrectomy or major surgery to small intestine.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (34)

Research Site

Alabaster, Alabama, United States

Location

Research Site

Encinitas, California, 92024, United States

Location

Research Site

Encinitas, California, United States

Location

Research Site

Gilroy, California, United States

Location

Research Site

Long Beach, California, United States

Location

Research Site

Davie, Florida, United States

Location

Research Site

Orlando, Florida, United States

Location

Research Site

Rochester, Minnesota, United States

Location

Research Site

St Louis, Missouri, United States

Location

Research Site

Berkeley Heights, New Jersey, United States

Location

Research Site

New York, New York, United States

Location

Research Site

Fargo, North Dakota, United States

Location

Research Site

Columbus, Ohio, United States

Location

Research Site

Pittsburgh, Pennsylvania, United States

Location

Research Site

Nashville, Tennessee, United States

Location

Research Site

El Paso, Texas, United States

Location

Research Site

Houston, Texas, United States

Location

Research Site

San Antonio, Texas, 78229, United States

Location

Research Site

Lacey, Washington, United States

Location

Research Site

Waratah, New South Wales, Australia

Location

Research Site

Wollongong, New South Wales, Australia

Location

Research Site

Herston, Queensland, Australia

Location

Research Site

Redcliffe, Queensland, Australia

Location

Research Site

Hobart, Tasmania, Australia

Location

Research Site

Geelong, Victoria, Australia

Location

Research Site

Brasschaat, Belgium

Location

Research Site

Edegem, Belgium

Location

Research Site

Kortrijk, Belgium

Location

Research Site

Liège, Belgium

Location

Research Site

Mons, Belgium

Location

Research Site

Kuzmolovskiy, Russia

Location

Research Site

Moscow, Russia

Location

Research Site

Ryazan, Russia

Location

Research Site

Saint Petersburg, Russia

Location

MeSH Terms

Conditions

Breast Neoplasms

Interventions

6-chloro-9-(4-methoxy-3,5-dimethylpyridin-2-ylmethyl)-9H-purin-2-ylamineexemestane

Condition Hierarchy (Ancestors)

Neoplasms by SiteNeoplasmsBreast DiseasesSkin DiseasesSkin and Connective Tissue Diseases

Study Officials

  • Medical Director

    Biogen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 18, 2009

First Posted

October 29, 2009

Study Start

November 1, 2009

Primary Completion

October 1, 2011

Study Completion

October 1, 2011

Last Updated

October 2, 2015

Record last verified: 2011-12

Locations