NCT00918138

Brief Summary

The purpose of this study was to compare effect of Saxagliptin as add-on to Metformin on 24-hour mean weighted glucose (MWG) to the effect of uptitrating Metformin in subjects with T2DM inadequately controlled on metformin alone.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
219

participants targeted

Target at P25-P50 for phase_3 type-2-diabetes

Timeline
Completed

Started Aug 2009

Shorter than P25 for phase_3 type-2-diabetes

Geographic Reach
4 countries

21 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 9, 2009

Completed
2 days until next milestone

First Posted

Study publicly available on registry

June 11, 2009

Completed
2 months until next milestone

Study Start

First participant enrolled

August 1, 2009

Completed
9 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2010

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2010

Completed
1.4 years until next milestone

Results Posted

Study results publicly available

October 6, 2011

Completed
Last Updated

May 21, 2015

Status Verified

May 1, 2015

Enrollment Period

9 months

First QC Date

June 9, 2009

Results QC Date

September 2, 2011

Last Update Submit

May 4, 2015

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in 24-Hour Mean Weighted Glucose (MWG) at Week 4

    Adjusted mean change from baseline in MWG achieved with saxagliptin 5 mg plus metformin XR versus placebo plus metformin XR at Week 24. MWG was calculated as the area under the curve (AUC) for the full 24 hours expressed as average mg/dL. Glucose measurements were collected 30 minutes before and just prior to each meal (0 minutes) and 30, 60, 120, and 180 minutes after each meal (with 1 additional measurement at 240 minutes after the evening meal), midnight, 3 AM, and at end-of-domicile visit 24 hours after the first measurement. Mean change from baseline was adjusted for baseline value.

    Baseline, Week 4

Secondary Outcomes (2)

  • Change From Baseline to Week 4 in 2-hour Postprandial Glucose (PPG) (2 Hours After the Evening Meal)

    Baseline, Week 4

  • Change From Baseline Fasting Plasma Glucose (FPG) at Week 4, Obtained Immediately Before the Morning Meal

    Baseline, Week 4

Other Outcomes (2)

  • Participants With Confirmed Hypoglycemia Events During the Treatment Period

    AEs: up to last treatment day (LTD) +1 day or last visit day (LVD), whichever came last ; SAEs: up to LTD +30 days or LVD + 30 days, whichever came last. Mean duration of exposure=27.7 days for Saxa 5 mg + Met XR 1500 mg, and 28.3 days for Met 2000 mg.

  • Participants With Reported Hypoglycemic Adverse Events During Treatment Period

    AEs: up to last treatment day (LTD) +1 day or last visit day (LVD), whichever came last ; SAEs: up to LTD +30 days or LVD + 30 days, whichever came last. Mean duration of exposure=27.7 days for Saxa 5 mg + Met XR 1500 mg, and 28.3 days for Met 2000 mg.

Study Arms (2)

Saxagliptin + Metformin XR + matching Metformin XR placebo

EXPERIMENTAL

(Saxagliptin 5 mg plus Metformin XR 1500 plus matching Metformin XR 500 mg placebo)

Drug: SaxagliptinDrug: Metformin XRDrug: Placebo matching Metformin XR

Metformin XR + Metformin XR + matching Saxagliptin placebo

ACTIVE COMPARATOR

(Metformin XR 500 mg plus Metformin XR 1500 mg plus matching Saxagliptin 5 mg placebo)

Drug: Metformin XRDrug: Placebo matching Saxagliptin

Interventions

Tablets, Oral, 5 mg, once daily, 4 weeks

Also known as: BMS-477118, Onglyza
Saxagliptin + Metformin XR + matching Metformin XR placebo

Tablets, Oral, 1500 mg, once daily, 4 weeks

Also known as: Glucophage XR®
Metformin XR + Metformin XR + matching Saxagliptin placeboSaxagliptin + Metformin XR + matching Metformin XR placebo

Tablets, Oral, 0 mg, once daily, 4 weeks

Saxagliptin + Metformin XR + matching Metformin XR placebo

Tablets, Oral, 0 mg, once daily, 4 weeks

Metformin XR + Metformin XR + matching Saxagliptin placebo

Eligibility Criteria

Age18 Years - 78 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Type 2 diabetes
  • years of age
  • Taking stable dose of metformin immediate release (IR) or XR ≥850 mg and ≤1500 mg as monotherapy for at least 8 weeks prior to screening
  • Glycosylated hemoglobin A1C (A1C) 7.5-11.5% at screening
  • Fasting C-peptide: ≥1.0 ng/mL
  • FPG≥126 mg/dl obtained at the Day -7 visit
  • Body mass index (BMI): ≤ 40kg/m²
  • A1C ≥ 7.0% and ≤ 11.0% obtained at the Day -7 visit for randomization

You may not qualify if:

  • Women of childbearing potential unable or unwilling to use acceptable birth control
  • Women who are pregnant or breastfeeding
  • Significant cardiovascular history
  • Active liver disease
  • Renal impairment

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (21)

Dedicated Phase I, Inc.

Phoenix, Arizona, 85013, United States

Location

Pacific Sleep Medicine Services (Avastra Clinical Trials)

Redlands, California, 92373, United States

Location

Orange County Research Center

Tustin, California, 92780, United States

Location

Clinical Research Of South Florida

Coral Gables, Florida, 33134, United States

Location

Palm Springs Research Institute

Hialeah, Florida, 33012, United States

Location

Healthcare Clinical Data, Inc.

North Miami, Florida, 33161, United States

Location

River Birch Research Alliance, Llc

Blue Ridge, Georgia, 30513, United States

Location

Jasper Clinic, Inc.

Kalamazoo, Michigan, 49007, United States

Location

Clinilabs, Inc.

New York, New York, 10019, United States

Location

Medpace Clinical Pharmacology Unit

Cincinnati, Ohio, 45212, United States

Location

Clinical Trials Of Texas Inc.

San Antonio, Texas, 78229, United States

Location

Advanced Clinical Research

West Jordan, Utah, 84088, United States

Location

Local Institution

Buenos Aires, Buenos Aires, 1425, Argentina

Location

Local Institution

Capital Federal, Buenos Aires, 1429, Argentina

Location

Local Institution

Beersheba, 84101, Israel

Location

Local Institution

Holon, 58100, Israel

Location

Local Institution

Kfar Saba, 44281, Israel

Location

Local Institution

Safed, 13100, Israel

Location

Local Institution

Durango, Durango, 34000, Mexico

Location

Local Institution

Durango, Durango, 34075, Mexico

Location

Local Institution

Monterrey, Nuevo León, 64460, Mexico

Location

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

saxagliptinMetformin

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

BiguanidesGuanidinesAmidinesOrganic Chemicals

Results Point of Contact

Title
Boaz Hirschberg
Organization
AstraZeneca Pharmaceuticals

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 9, 2009

First Posted

June 11, 2009

Study Start

August 1, 2009

Primary Completion

May 1, 2010

Study Completion

May 1, 2010

Last Updated

May 21, 2015

Results First Posted

October 6, 2011

Record last verified: 2015-05

Locations