NCT00910065

Brief Summary

The objective of this study is to investigate whether intravenous administration (injected into a vein) of acetylsalicylic acid (Aspirin) in doses of 250 and 500 mg is superior to oral treatment of ACS with tablets containing 300 mg of Aspirin.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
270

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Mar 2011

Typical duration for phase_3

Geographic Reach
4 countries

37 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 28, 2009

Completed
1 day until next milestone

First Posted

Study publicly available on registry

May 29, 2009

Completed
1.8 years until next milestone

Study Start

First participant enrolled

March 1, 2011

Completed
3.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2014

Completed
3 months until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2014

Completed
Last Updated

June 25, 2015

Status Verified

June 1, 2015

Enrollment Period

3.1 years

First QC Date

May 28, 2009

Last Update Submit

June 24, 2015

Conditions

Keywords

Acute Coronary SyndromeACSAspirin

Outcome Measures

Primary Outcomes (1)

  • Concentration of Thromboxane B2 (TXB2) at 5 Minutes Post-dose

    5 minutes post-dose

Secondary Outcomes (5)

  • Concentration of Thromboxane B2 (TXB2) at 20 Minutes Post-dose

    20 minutes post-dose

  • Platelet Aggregation Inhibition (PAI) at 5 Minutes and 20 Minutes After Single Dose of Study Drug Administration Measured as Response to Treatment

    5 and 20 minutes post-dose

  • Serum Concentration of Prostacyclin Metabolite at 5 and 20 Minutes Post-dose

    5 and 20 minutes post-dose

  • Incidence of the Composite Clinical Endpoint of Cardiovascular Death, Stroke and Myocardial Infarction up to Day 30 After Single Dose of Study Drug Administration

    Post-randomization up to 30 days after single dose of study drug administration

  • Incidence of Post-randomization Deaths From all Causes, Cardiovascular Deaths, Myocardial Re/Infarctions and Ischemic Strokes Within 24 Hours, 7 Days And 30 Days After Single Dose of Study Drug Administration

    Post-randomization up to 24 hours, 7 days and 30 days after single dose of study drug administration

Study Arms (3)

Arm 1

EXPERIMENTAL
Drug: D,L-lysine acetylsalicylate (Aspirin, BAY81-8781) 500 mg IV

Arm 2

EXPERIMENTAL
Drug: D,L-lysine acetylsalicylate (Aspirin, BAY81-8781) 250 mg IV

Arm 3

ACTIVE COMPARATOR
Drug: Acetylsalicylic acid (Aspirin, BAYe4465) 300 mg Tablet

Interventions

Single IV dose of aspirin at a dose of 500 mg as bolus infusion injection in approximately 30 seconds through the vein on Day 1.

Arm 1

Single IV dose of aspirin at a dose of 250 mg as bolus infusion injection in approximately 30 seconds through the vein on Day 1.

Arm 2

Single oral dose of aspirin tablet at a dose of 300 mg on Day 1.

Arm 3

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Angina pectoris lasting for more than 20 minutes within the last 24 hours before study drug treatment (or equivalent acute symptoms such as increasing dyspnea, diaphoresis, nausea, abdominal/epigastric pain, syncope etc.)
  • ECG change suggestive for ischemia:
  • ST elevation or T-wave change or ST depression, new or presumed left bundle-branch block (LBBB)
  • Elevated troponin T level \> 0.01 ng/ml, levels according to local laboratory reference values
  • Risk factors for ACS such as known coronary artery disease (CAD), diabetes mellitus, impaired renal function, peripheral artery or cerebrovascular disease, current smoking.

You may not qualify if:

  • Treatment with acetylsalicylic acid (ASA) within 48 hours prior to study drug treatment
  • Treatment with glycoprotein IIa/IIIb inhibitors within 48 hours prior to study drug treatment and before the 20 minutes blood samples for thromboxane, prostacycline and platelet aggregation measurement have been taken
  • Thrombolytic therapy within 24 hours before study drug treatment
  • Obligation for tracheal intubation and mechanical ventilation
  • Contraindications to ASA treatment
  • Known haemorrhagic diathesis
  • Evidence of an active gastrointestinal or urogenital bleeding
  • Stroke within 3 months prior to study drug treatment
  • Major surgery including coronary artery bypass graft (CABG) within 6 weeks prior to study drug treatment
  • Known severe hepatic or renal insufficiency
  • Pregnant or breast-feeding women

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (37)

Unknown Facility

Guangzhou, Guangdong, 510080, China

Location

Unknown Facility

Guangzhou, Guangdong, 510100, China

Location

Unknown Facility

Guangzhou, Guangdong, 510120, China

Location

Unknown Facility

Guangzhou, Guangdong, 510405, China

Location

Unknown Facility

Changsha, Hunan, 410013, China

Location

Unknown Facility

Nanchang, Jiangxi, 330006, China

Location

Unknown Facility

Shenyang, Liaoning, 110004, China

Location

Unknown Facility

Shenyang, Liaoning, 110016, China

Location

Unknown Facility

Hangzhou, Zhejiang, 310016, China

Location

Unknown Facility

Beijing, 100029, China

Location

Unknown Facility

Beijing, 100037, China

Location

Unknown Facility

Shanghai, 200080, China

Location

Unknown Facility

Bad Krozingen, Baden-Wurttemberg, 79189, Germany

Location

Unknown Facility

Heidelberg, Baden-Wurttemberg, 69120, Germany

Location

Unknown Facility

Coburg, Bavaria, 96450, Germany

Location

Unknown Facility

Dachau, Bavaria, 85221, Germany

Location

Unknown Facility

Melsungen, Hesse, 34212, Germany

Location

Unknown Facility

Bonn, North Rhine-Westphalia, 53105, Germany

Location

Unknown Facility

Cologne, North Rhine-Westphalia, 50968, Germany

Location

Unknown Facility

Essen, North Rhine-Westphalia, 45147, Germany

Location

Unknown Facility

Mönchengladbach, North Rhine-Westphalia, 41063, Germany

Location

Unknown Facility

Soest, North Rhine-Westphalia, 59494, Germany

Location

Unknown Facility

Ludwigshafen am Rhein, Rhineland-Palatinate, 67063, Germany

Location

Unknown Facility

Mainz, Rhineland-Palatinate, 55131, Germany

Location

Unknown Facility

Worms, Rhineland-Palatinate, 67550, Germany

Location

Unknown Facility

Magdeburg, Saxony-Anhalt, 39112, Germany

Location

Unknown Facility

Berlin, State of Berlin, 12351, Germany

Location

Unknown Facility

Moscow, 109263, Russia

Location

Unknown Facility

Moscow, 115093, Russia

Location

Unknown Facility

Moscow, 115516, Russia

Location

Unknown Facility

Moscow, 117292, Russia

Location

Unknown Facility

Moscow, 119881, Russia

Location

Unknown Facility

Moscow, 125101, Russia

Location

Unknown Facility

Alicante, Alicante, 03010, Spain

Location

Unknown Facility

San Juan, Alicante, 03550, Spain

Location

Unknown Facility

Sabadell, Barcelona, 08208, Spain

Location

Unknown Facility

Valencia, Valencia, 46015, Spain

Location

Related Links

MeSH Terms

Conditions

Acute Coronary Syndrome

Interventions

AspirinTablets

Condition Hierarchy (Ancestors)

Myocardial IschemiaHeart DiseasesCardiovascular DiseasesVascular Diseases

Intervention Hierarchy (Ancestors)

SalicylatesHydroxybenzoatesPhenolsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDosage FormsPharmaceutical Preparations

Study Officials

  • Bayer Study Director

    Bayer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 28, 2009

First Posted

May 29, 2009

Study Start

March 1, 2011

Primary Completion

April 1, 2014

Study Completion

July 1, 2014

Last Updated

June 25, 2015

Record last verified: 2015-06

Locations