NCT00902369

Brief Summary

This will be a Phase II, multi-centre study consisting of 2 parts. Part 1: Clinical Pharmacology Study (drug-drug interaction between AK106-001616 and methotrexate) Part 2: Proof of Concept Study

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
130

participants targeted

Target at P50-P75 for phase_2 rheumatoid-arthritis

Timeline
Completed

Started May 2009

Shorter than P25 for phase_2 rheumatoid-arthritis

Geographic Reach
6 countries

12 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

May 1, 2009

Completed
13 days until next milestone

First Submitted

Initial submission to the registry

May 14, 2009

Completed
1 day until next milestone

First Posted

Study publicly available on registry

May 15, 2009

Completed
5 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2009

Completed
9 months until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2010

Completed
Last Updated

July 25, 2016

Status Verified

July 1, 2010

Enrollment Period

5 months

First QC Date

May 14, 2009

Last Update Submit

July 21, 2016

Conditions

Keywords

AK106-001616

Study Arms (3)

AK106-001616

EXPERIMENTAL
Drug: AK106-001616

Placebo

PLACEBO COMPARATOR

Part1: AK106-001616 and Placebo

Drug: Placebo

Active comparator

ACTIVE COMPARATOR

Part2: AK106-001616 and Active comparator

Drug: Active comparator

Interventions

Part1: Dose escalation Part2: Dose expansion

AK106-001616
Placebo
Active comparator

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Diagnosis of RA (class I to III)
  • Stable dose of methotrexate (at least 12 weeks)

You may not qualify if:

  • Pregnant or breastfeeding
  • Abnormal screening laboratory test values considered to be clinically significant

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (12)

Unknown Facility

Hlučín, Czechia

Location

Unknown Facility

Prague, Czechia

Location

Unknown Facility

Uherské Hradiště, Czechia

Location

Unknown Facility

Frankfurt am Main, Hesse, Germany

Location

Unknown Facility

Berlin, Germany

Location

Unknown Facility

Hamburg, Germany

Location

Unknown Facility

Budapest, Hungary

Location

Unknown Facility

Érd, Hungary

Location

Unknown Facility

Vilnius, Lithuania

Location

Unknown Facility

Bucharest, Romania

Location

Unknown Facility

Cambridge, Cambridgeshire, United Kingdom

Location

Unknown Facility

Sheffield, South Yorkshire, United Kingdom

Location

Related Publications (1)

  • Kozaki T, Tagashira M, Yamanishi K, Ellis B, Kayanoki T, Ooishi R, Sugiyama K, Matsuda S, Tsuruta K, Kohira T, Tsurui K. Evaluation of drug-drug interaction between the novel cPLA2 inhibitor AK106-001616 and methotrexate in rheumatoid arthritis patients. Xenobiotica. 2015;45(7):615-24. doi: 10.3109/00498254.2014.1000430. Epub 2015 Jan 12.

MeSH Terms

Conditions

Arthritis, Rheumatoid

Interventions

AK106-001616

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic DiseasesConnective Tissue DiseasesSkin and Connective Tissue DiseasesAutoimmune DiseasesImmune System Diseases

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 14, 2009

First Posted

May 15, 2009

Study Start

May 1, 2009

Primary Completion

October 1, 2009

Study Completion

July 1, 2010

Last Updated

July 25, 2016

Record last verified: 2010-07

Locations