NCT00881166

Brief Summary

Adult subjects with malignant disease appropriate for treatment with carboplatin/paclitaxel, carboplatin/etoposide, topotecan, docetaxel or erlotinib according to the standard dosing regimen will be enrolled in each treatment arm. Primary objective: Determine the MTD. Secondary objectives: Response rates, PK, quantify MP-470 on PK of SOC, and collect pharmacodynamic information. Evaluate the overall safety of MP-470 when co-administered with specific SOC treatments.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
101

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started Nov 2007

Typical duration for phase_1

Geographic Reach
1 country

5 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 1, 2007

Completed
1.4 years until next milestone

First Submitted

Initial submission to the registry

April 13, 2009

Completed
2 days until next milestone

First Posted

Study publicly available on registry

April 15, 2009

Completed
8 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 1, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2009

Completed
Last Updated

August 2, 2024

Status Verified

August 1, 2024

Enrollment Period

2.1 years

First QC Date

April 13, 2009

Last Update Submit

August 1, 2024

Conditions

Keywords

MP-470Multi-targeted Tyrosine Kinase InhibitorMalignant disease

Outcome Measures

Primary Outcomes (1)

  • Maximum tolerated dose (MTD)

    March 2010

Secondary Outcomes (3)

  • Response rate

    March 2010

  • Pharmacokinetics, pharmacodynamic effects on biomarker modulation.

    March 2010

  • Experience DLT

    March 2010

Study Arms (5)

1

EXPERIMENTAL

oral MP-470 + paclitaxel/carboplatin

Drug: MP-470 + paclitaxel/carboplatin

2

EXPERIMENTAL

oral MP-470 + carboplatin/etoposide

Drug: MP-470 + carboplatin/etoposide

3

EXPERIMENTAL

oral MP-470 + topotecan

Drug: MP-470 + topotecan

4

EXPERIMENTAL

oral MP-470 + docetaxel

Drug: MP-470 + docetaxel

5

EXPERIMENTAL

oral MP-470 + Erlotinib

Drug: MP-470 + erlotinib

Interventions

Topotecan 1.5 mg/m2 IV infusion over 30 minutes on Days 1-5

3

Docetaxel 75 mg/m2 IV infusion over 1 hour on Day 1

4

150 mg PO once daily at least 1 hour before or 2 hours after eating

5

Paclitaxel 200 mg/m2 IV infusion over 3 hours followed by carboplatin IV infusion over 1 hour to a target AUC of 6 mg∙min/mL on Day 1

1

Carboplatin IV infusion over 1 hour to target AUC of 5 mg min/mL on Day 1 followed by etoposide 100 mg/m2 IV infusion over 2 hours on Days 1-3

2

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Malignant disease appropriate for initiating treatment with carboplatin/paclitaxel, carboplatin/etoposide, topotecan, docetaxel, or erlotinib.
  • Must be able to read, understand, and sign the IRB approved Informed Consent Form.
  • At least 18 years old.
  • Eastern Cooperative Oncology Group (ECOG) performance status 0-2.
  • Adequate bone marrow function; normal renal and hepatic function, normal cardiac function.

You may not qualify if:

  • Any other active invasive malignancy except non-melanoma skin cancers or cervical carcinoma in situ.
  • History of significant cardiovascular disease such as uncontrolled or symptomatic arrhythmias, congestive heart failure and/or myocardial infarction.
  • Received any anticancer agent(s) within the past 3 weeks, including investigational agents, chemotherapy (6 weeks for nitrosoureas or mitomycin), immunotherapy, biologic or hormonal therapy other than LHRH agonists.
  • Received prior radiation therapy within the past 4 weeks.
  • Any serious, uncontrolled active infection that requires systemic treatment or known infection with HIV, HCV or HBV.
  • Patient requires treatment with immunosuppressive agents other than corticosteroids appropriate for the SOC chemotherapy regimen or those at stable doses for at least 2 weeks.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (5)

Premiere Oncology

Scottsdale, Arizona, 85258, United States

Location

Premiere Oncology

Santa Monica, California, 90404, United States

Location

Audie Murphy Veterans Memorial Hospital (VA)

San Antonio, Texas, 78229, United States

Location

CTRC at the UT Health Science Center at San Antonio

San Antonio, Texas, 78229, United States

Location

South Texas Accelerated Research Therapy (START)

San Antonio, Texas, 78229, United States

Location

Related Publications (1)

  • Mita M, Gordon M, Rosen L, Kapoor N, Choy G, Redkar S, Taverna P, Oganesian A, Sahai A, Azab M, Bristow R, Tolcher AW. Phase 1B study of amuvatinib in combination with five standard cancer therapies in adults with advanced solid tumors. Cancer Chemother Pharmacol. 2014 Jul;74(1):195-204. doi: 10.1007/s00280-014-2481-1. Epub 2014 May 22.

MeSH Terms

Interventions

amuvatinibTopotecanDocetaxelErlotinib HydrochloridePaclitaxelCarboplatinEtoposide

Intervention Hierarchy (Ancestors)

CamptothecinAlkaloidsHeterocyclic CompoundsTaxoidsCyclodecanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsDiterpenesTerpenesQuinazolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingCoordination ComplexesPodophyllotoxinTetrahydronaphthalenesNaphthalenesPolycyclic Aromatic HydrocarbonsHydrocarbons, AromaticPolycyclic CompoundsGlucosidesGlycosidesCarbohydrates

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 13, 2009

First Posted

April 15, 2009

Study Start

November 1, 2007

Primary Completion

December 1, 2009

Study Completion

December 1, 2009

Last Updated

August 2, 2024

Record last verified: 2024-08

Locations