NCT00754130

Brief Summary

The multiple dose study to assess the safety, tolerability, pharmacokinetics and pharmacodynamics of MK-0941 in Japanese patients with Type 2 Diabetes.

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
16

participants targeted

Target at below P25 for phase_1

Timeline
Completed

Started Sep 2008

Shorter than P25 for phase_1

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2008

Completed
15 days until next milestone

First Submitted

Initial submission to the registry

September 16, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 17, 2008

Completed
14 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2008

Completed
4 years until next milestone

Results Posted

Study results publicly available

October 3, 2012

Completed
Last Updated

March 12, 2015

Status Verified

February 1, 2015

Enrollment Period

1 month

First QC Date

September 16, 2008

Results QC Date

August 31, 2012

Last Update Submit

February 23, 2015

Conditions

Outcome Measures

Primary Outcomes (2)

  • Number of Participants Who Experienced at Least One Adverse Event (AE)

    An AE is defined as any unfavorable and unintended change in the structure, function, or chemistry of the body temporally associated with the use of the study drug, whether or not considered related to the use of the product. Participants were monitored for occurrence AEs for up to 8 days after last dose of study drug during Period 1 and for up to 14 days after last dose of study drug during Period 2.

    Up to 14 days after last dose of study drug

  • Number of Participants Who Discontinued Study Drug Due to an AE

    An AE is defined as any unfavorable and unintended change in the structure, function, or chemistry of the body temporally associated with the use of the study drug, whether or not considered related to the use of the product. Participants were monitored for occurrence AEs for up to 8 days after last dose of study drug during Period 1 and for up to 14 days after last dose of study drug during Period 2.

    Up to 14 days after last dose of study drug

Secondary Outcomes (6)

  • Plasma Pharmacokinetic Parameter: Area Under the Concentration-time Curve (AUC)(0-24hr) of MK-0941

    Up to 72 hours after study drug administration

  • Plasma Pharmacokinetic Parameter: Maximum Concentration (Cmax) of MK-0941

    Up to 72 hours after study drug administration

  • Plasma Pharmacokinetic Parameter: Time to Reach Cmax (Tmax) of MK-0941

    Up to 72 hours after study drug administration

  • Plasma Pharmacokinetic Parameter: Concentration of MK-0941 at 24 Hours (C24hr)

    Up to 72 hours after study drug administration

  • Plasma Pharmacokinetic Parameter: Apparent Terminal Elimination Half-life (t1/2) of MK-0941

    Up to 72 hours after study drug administration

  • +1 more secondary outcomes

Study Arms (6)

Placebo/MK-0941 20mg

EXPERIMENTAL

Participants received Placebo during Period 1 and MK-0941 20 mg during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: PlaceboDrug: MK-0941

MK-0941 5mg/Placebo

EXPERIMENTAL

Participants received MK-0941 5 mg during Period 1 and Placebo during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: PlaceboDrug: MK-0941

MK-0941 5mg/MK-0941 20mg

EXPERIMENTAL

Participants received MK-0941 5 mg during Period 1 and MK-0941 20 mg during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: MK-0941

Placebo/MK-0941 40mg

EXPERIMENTAL

Participants received Placebo during Period 1 and MK-0941 40 mg during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: PlaceboDrug: MK-0941

MK-0941 10mg/Placebo

EXPERIMENTAL

Participants received MK-0941 10 mg during Period 1 and Placebo during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: PlaceboDrug: MK-0941

MK-0941 10mg/MK-0941 40mg

EXPERIMENTAL

Participants received MK-0941 10 mg during Period 1 and MK-0941 40 mg during Period 2. There was a washout period of at least 8 days between the two treatment periods.

Drug: MK-0941

Interventions

Placebo tablets before every meal (q.a.c) Treatment period is 5 days.

MK-0941 10mg/PlaceboMK-0941 5mg/PlaceboPlacebo/MK-0941 20mgPlacebo/MK-0941 40mg

MK-0941 5 mg tablets q.a.c.; 10 mg tablets q.a.c.; 20 mg tablets q.a.c.; or 40 mg tablets q.a.c. Treatment period is 5 days.

MK-0941 10mg/MK-0941 40mgMK-0941 10mg/PlaceboMK-0941 5mg/MK-0941 20mgMK-0941 5mg/PlaceboPlacebo/MK-0941 20mgPlacebo/MK-0941 40mg

Eligibility Criteria

Age20 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Japanese Male or Female between 20 to 65 years of age
  • Diagnosis of Type 2 Diabetes
  • Patient being treated by diet and exercise alone

You may not qualify if:

  • Patient has a history of Type 1 Diabetes
  • Patient is being treated with glaucoma medications
  • Patient has donated blood or participated in another clinical study in the past 12 weeks
  • Patient is a regular user of any illicit drugs or has a history of drug, including alcohol, abuse

Contact the study team to confirm eligibility.

Sponsors & Collaborators

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

3-((6-(ethylsulfonyl)-3-pyridinyl)oxy)-5-(2-hydroxy-1-methylethoxy)-N-(1-methyl-1H-pyrazol-3-yl)benzamide

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Results Point of Contact

Title
Senior Vice President, Global Clinical Development
Organization
Merck Sharp & Dohme Corp

Study Officials

  • Medical Monitor

    Merck Sharp & Dohme LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 16, 2008

First Posted

September 17, 2008

Study Start

September 1, 2008

Primary Completion

October 1, 2008

Study Completion

October 1, 2008

Last Updated

March 12, 2015

Results First Posted

October 3, 2012

Record last verified: 2015-02