NCT00715676

Brief Summary

This study will evaluate the effect of a 1-year administration of the vitamin D analog 2-methylene-19-nor-(20S)-1alpha, 25-dihydroxyvitamin D3 (DP001) on bone mineral density (BMD), safety, and tolerability.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
157

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Mar 2007

Geographic Reach
1 country

9 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2007

Completed
1.4 years until next milestone

First Submitted

Initial submission to the registry

July 14, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

July 15, 2008

Completed
5 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 1, 2008

Completed
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2009

Completed
1 year until next milestone

Results Posted

Study results publicly available

January 11, 2010

Completed
Last Updated

January 11, 2010

Status Verified

December 1, 2009

Enrollment Period

1.8 years

First QC Date

July 14, 2008

Results QC Date

September 16, 2009

Last Update Submit

December 7, 2009

Conditions

Keywords

Osteoporosis2-methylene-19-nor-(20S)-1a, 25-dihydroxyvitamin D3Vitamin DBone Density Conservation AgentsBone Regeneration

Outcome Measures

Primary Outcomes (1)

  • Percent Change From Baseline in Lumbar Spine Bone Mineral Density (BMD) at Week 52

    Percent change in lumbar spine BMD (relative to baseline) at Week 52

    Baseline and Week 52

Secondary Outcomes (6)

  • Percent Change From Baseline in Hip Bone Mineral Density (BMD) at Week 52

    Baseline and Week 52

  • Percent Change From Baseline in Femoral Neck Bone Mineral Density (BMD) at Week 52

    Baseline and Week 52

  • Percent Change From Baseline in Trochanter Bone Mineral Density (BMD) at Week 52

    Baseline and Week 52

  • Change From Baseline in Serum Calcium Levels at Week 52

    Baseline and Week 52

  • Percent Change From Baseline in Serum Bone Markers at Week 26

    Baseline and Week 26

  • +1 more secondary outcomes

Study Arms (3)

Group 1

PLACEBO COMPARATOR
Drug: Placebo

Group 2

EXPERIMENTAL

220 ng

Drug: DP001

Group 3

EXPERIMENTAL

440 ng

Drug: DP001

Interventions

oral, once daily

Group 1
DP001DRUG

oral, once daily

Also known as: 2-methylene-19-nor-(20S)-1a, 25-dihydroxyvitamin D3, 2MD
Group 2Group 3

Eligibility Criteria

Age55 Years - 80 Years
Sexfemale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Postmenopausal female subjects, defined as amenorrheic for at least 5 years
  • Body Mass Index of 18 to 35
  • Osteopenic
  • Generally healthy
  • Informed consent

You may not qualify if:

  • History or evidence of acute or unstable chronic hematological, renal, endocrine, pulmonary, gastrointestinal, cardiovascular, psychiatric, or neurologic diseases
  • Current or recent treatment with any medications or products affecting vitamin D metabolism, calcium balance, bone turnover, or an investigational drug therapy
  • lead electrocardiogram demonstrating QTc (QT interval corrected for heart rate) \>450 milliseconds at screening
  • Abnormal creatinine clearance
  • Elevated urinary calcium levels
  • Vitamin D deficiency
  • Excessive dietary calcium or vitamin D intake
  • Current use of any illicit drug and/or history of alcohol abuse

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (9)

Boling Clinical Trials

Upland, California, 91786, United States

Location

Indiana School of Medicine University Hospital

Indianapolis, Indiana, 46202, United States

Location

Bethesda Health Research

Bethesda, Maryland, 20817, United States

Location

Creighton University Bone Metabolism Unit

Omaha, Nebraska, 68131, United States

Location

New Mexico Clinical Research and Osteoporosis Center

Albuquerque, New Mexico, 87106, United States

Location

Winthrop University Hospital Bone Mineral Research Center

Mineola, New York, 11501, United States

Location

Helen Hayes Hospital Clinical Research Center

West Haverstraw, New York, 10993, United States

Location

Altoona Center for Clinical Research

Duncansville, Pennsylvania, 16635, United States

Location

University of Wisconsin-Madison Osteoporosis Clinical Research

Madison, Wisconsin, 53705, United States

Location

Related Publications (3)

  • Ke HZ, Qi H, Crawford DT, Simmons HA, Xu G, Li M, Plum L, Clagett-Dame M, DeLuca HF, Thompson DD, Brown TA. A new vitamin D analog, 2MD, restores trabecular and cortical bone mass and strength in ovariectomized rats with established osteopenia. J Bone Miner Res. 2005 Oct;20(10):1742-55. doi: 10.1359/JBMR.050605. Epub 2005 Jun 13.

    PMID: 16160732BACKGROUND
  • Plum LA, Fitzpatrick LA, Ma X, Binkley NC, Zella JB, Clagett-Dame M, DeLuca HF. 2MD, a new anabolic agent for osteoporosis treatment. Osteoporos Int. 2006;17(5):704-15. doi: 10.1007/s00198-005-0036-3. Epub 2006 Feb 21.

    PMID: 16491322BACKGROUND
  • Shevde NK, Plum LA, Clagett-Dame M, Yamamoto H, Pike JW, DeLuca HF. A potent analog of 1alpha,25-dihydroxyvitamin D3 selectively induces bone formation. Proc Natl Acad Sci U S A. 2002 Oct 15;99(21):13487-91. doi: 10.1073/pnas.202471299. Epub 2002 Oct 8.

    PMID: 12374862BACKGROUND

MeSH Terms

Conditions

Osteoporosis

Condition Hierarchy (Ancestors)

Bone Diseases, MetabolicBone DiseasesMusculoskeletal DiseasesMetabolic DiseasesNutritional and Metabolic Diseases

Results Point of Contact

Title
Hector F. DeLuca, President and Chief Executive Officer
Organization
Deltanoid Pharmaceuticals

Study Officials

  • Wendy A Bedale, Ph.D.

    Deltanoid Pharmaceuticals

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
GT60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

July 14, 2008

First Posted

July 15, 2008

Study Start

March 1, 2007

Primary Completion

December 1, 2008

Study Completion

January 1, 2009

Last Updated

January 11, 2010

Results First Posted

January 11, 2010

Record last verified: 2009-12

Locations