NCT00518115

Brief Summary

This study is a placebo-controlled study in patients with Type 2 Diabetes Mellitus who are either taking no diabetes medication or who are taking metformin only. This study will investigate the safety, tolerability, and efficacy of Albiglutide (GSK716155) and will measure the levels of Albiglutide (GSK716155) in the bloodstream when it is given for 16 weeks. As a comparison, some subjects will receive exenatide instead of Albiglutide (GSK716155). The study will involve weekly visits for 17 weeks,and less frequent follow-up visits for an additional 10 weeks. Assessments include repeat blood sampling and monitoring of any side effects.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
361

participants targeted

Target at P75+ for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started Apr 2007

Geographic Reach
3 countries

163 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

April 1, 2007

Completed
5 months until next milestone

First Submitted

Initial submission to the registry

August 17, 2007

Completed
3 days until next milestone

First Posted

Study publicly available on registry

August 20, 2007

Completed
9 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2008

Completed
6.1 years until next milestone

Results Posted

Study results publicly available

June 23, 2014

Completed
Last Updated

December 16, 2016

Status Verified

November 1, 2016

Enrollment Period

1.1 years

First QC Date

August 17, 2007

Results QC Date

May 1, 2014

Last Update Submit

November 3, 2016

Conditions

Keywords

GLP-1,Type 2 Diabetes,pharmacokinetics,pharmacodynamics,GSK716155,metformin,exenatideType 2 Diabetes Mellitus

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Glycosylated Hemoglobin (HbA1c) at Week 16

    HbA1c is a form of hemoglobin that is measured primarily to identify the average plasma glucose concentration over a 2- to 3-month period. The Baseline HbA1c value is defined as the last non-missing value before the start of treatment. Change from Baseline in HbA1c was calculated as the value at Week 16 minus the value at Baseline. Based on ANCOVA: Change = treatment + Baseline HbA1c + prior therapy + gender + region. The last observation carried forward (LOCF) method was used to impute missing data, in which the last valid observation recorded on treatment (scheduled or unscheduled) was used to impute the missing measurement. For participants who had missing observations before their last observation on treatment, the closest previous non-missing on-treatment observation was carried forward to missing visits. If a participant had missing observation(s) immediately after Baseline, the Baseline observation was not carried forward and was left as missing.

    Baseline and Week 16

Secondary Outcomes (17)

  • Change From Baseline in HbA1c at Weeks 4, 5, 7, 8, 9, 12, 15, and 16

    Baseline and Weeks 4, 5, 7, 8, 9, 12, 15, and 16

  • Number of Participants Who Achieved Target Values for HbA1c <6.5% and >=6.5% to <7% at Weeks 4, 5, 7, 8, 9, 12, 15, and 16

    Weeks (W) 4, 5, 7, 8, 9, 12, 15, and 16

  • Change From Baseline in Waist Circumference at Week 16

    Baseline and Week 16

  • Change From Baseline in Body Weight at Week 16

    Baseline and Week 16

  • Percent Change From Baseline in Body Weight at Week 16

    Baseline and Week 16

  • +12 more secondary outcomes

Interventions

Albiglutide weekly subcutaneous injection or exenatide twice daily injection

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has type 2 diabetes mellitus as defined by the criteria of the American Diabetes Association and recognized by World Health Organization Expert Committee on the Diagnosis and Classification of Diabetes Mellitus \[American Diabetes Association, 2004a\] at least three months preceding screening
  • Has concurrent type 2 diabetes mellitus therapy: Must be diet and exercise treated; must not have taken antidiabetic medication for at least three months prior to prescreening or Monotherapy with metformin, with a history of a stable dose for at least three months before prescreening (not taking more than one oral antidiabetic agent)
  • Has HbA1c level at screening ≥7 and ≤10%
  • Is male or female 18 to 75 years of age, inclusive, at screening
  • Has body mass index ≥20 and ≤40 kg/m²
  • If subject is a smoker, must be able to abstain while in clinic at each visit
  • If female, is eligible to enter and participate throughout the study, including the follow-up period: 1) If of nonchildbearing potential (i.e. physiologically incapable of becoming pregnant {tubal ligation}, including any female who is postmenopausal \[\>1 year without menstrual period\]); or, 2) If of childbearing potential, has negative pregnancy tests at screening (serum) and at baseline (urine) and: 3) Has a male partner who is sterile prior to the female subject's entry into the study and is the sole sexual partner for that female subject, or 4) Uses double-barrier methods of contraception; condoms (with spermicide) and intrauterine devices are acceptable, or 5) Uses hormonal contraceptives (oral, depots, patches, etc) with double-barrier methods of contraception as outlined above, or, 6) Abstains from sexual intercourse, or 7) Is with a same-sex partner and does not participate in bisexual activities where there is any risk of pregnancy
  • Signs and dates informed consent before any study-related procedures are performed

You may not qualify if:

  • Has metabolic disease including but not limited to: 1) Diagnosis of type 1 diabetes mellitus, 2) Uncorrected thyroid dysfunction (NOTE: subjects with hypothyroidism on a stable dose of thyroid replacement therapy for at least three months prior to screening, and who have a screening thyroid-stimulating hormone within the limits of normal may participate)
  • Has qualitative changes in lifestyle that, in the opinion of the investigator, would affect the subject's weight or disease status
  • Had previous use of insulin within one month prior to screening, or more than seven total days of insulin treatment within three months prior to screening
  • Has fasting serum triglycerides ≥800mg/dL or 9mmol/L at screening (Visit 2). Subjects receiving lipid-lowering therapy must have been on the same dose of therapy for the past three months. Fasting is defined as no food/drink for at least eight hours prior to sampling
  • If female, is currently lactating, pregnant, or actively trying to become pregnant
  • Has significant renal disease as manifested by one or more of the following: 1) Creatinine clearance \<60mL/min. (estimated from serum creatinine and demographic data using the modification of diet in renal disease calculation; refer to the SPM/ISFM), 2) Urine albumin excretion ≥500 µg/mL on a urine spot check, 3) Known loss of a kidney either by surgical ablation, injury, or disease
  • Has history of significant comorbid diseases active within the last six months (e.g., gastrointestinal disease)
  • Has history of pancreatitis within five years prior to randomization
  • Has a documented history of chronic or advanced hepatobiliary disease including a history of, or positive laboratory results for, hepatitis at screening (Visit 2), and/or clinically significant hepatic enzyme elevation including: 1) Any two of the following enzymes greater than 1.5 times the upper limit of normal (ULN) value: - alanine aminotransferase (ALT), - aspartate aminotransferase (AST), - alkaline phosphatase (ALP), 2) Any one of the above enzymes two times greater than the ULN value AND total or direct bilirubin \>1.5 times the ULN
  • Has a history of alcohol or substance abuse within the past year, as determined by the investigator or a positive urine drug screen at screening (Visit 2) or during treatment: 1) Unwilling to refrain from the use of excessive alcohol or illicit drugs and adhere to other protocol-stated restrictions while participating in the study, 2) History of alcohol abuse defined as an average weekly intake of greater than 21 units or an average daily intake of greater than three units (males) or defined as an average weekly intake of greater than 14 units or an average daily intake of greater than two units (females). One unit is equivalent to a half-pint of beer or one measure of spirits or one glass of wine, 2) The investigator should exercise their medical judgment to determine if a urine drug screen is indicated
  • Is currently taking prohibited concomitant medications listed in Section 6.6.2
  • Has clinically significant anemia (i.e., hemoglobin \<12.0g/dL or \<120.0g/L for males and \<11.0g/dL or \<110.0g/L for females) or any other abnormal hematological profile that is considered by the investigator to be clinically significant
  • Has known allergy to any formulation excipients, or history of drug or other allergy, which, in the opinion of the responsible study physician, contradicts participation
  • Received treatment with an investigational drug or participated in any other clinical trial during the previous 30 days
  • Has prior use of investigational agents with long half-lives of greater than seven days within the three months prior to screening
  • +3 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (163)

GSK Investigational Site

Anniston, Alabama, 36207, United States

Location

GSK Investigational Site

Birmingham, Alabama, 35233, United States

Location

GSK Investigational Site

Mobile, Alabama, 36617, United States

Location

GSK Investigational Site

Bull Shoals, Arizona, 72619, United States

Location

GSK Investigational Site

Glendale, Arizona, 85306, United States

Location

GSK Investigational Site

Jonesboro, Arizona, 72401, United States

Location

GSK Investigational Site

Phoenix, Arizona, 85032, United States

Location

GSK Investigational Site

Harrisburg, Arkansas, 72432, United States

Location

GSK Investigational Site

Jonesboro, Arkansas, 72401, United States

Location

GSK Investigational Site

Little Rock, Arkansas, 72205, United States

Location

GSK Investigational Site

Little Rock, Arkansas, 72211-3733, United States

Location

GSK Investigational Site

Searcy, Arkansas, 72143, United States

Location

GSK Investigational Site

Castro Valley, California, 94546, United States

Location

GSK Investigational Site

Culver City, California, 90232, United States

Location

GSK Investigational Site

Fullerton, California, 92835, United States

Location

GSK Investigational Site

Garden Grove, California, 92843, United States

Location

GSK Investigational Site

Huntington Beach, California, 92646, United States

Location

GSK Investigational Site

Huntington Beach, California, 92648, United States

Location

GSK Investigational Site

Huntington Park, California, 90255, United States

Location

GSK Investigational Site

Lake Forest, California, 92630, United States

Location

GSK Investigational Site

Loma Linda, California, 92354, United States

Location

GSK Investigational Site

Los Angeles, California, 90022, United States

Location

GSK Investigational Site

Orange, California, 92868, United States

Location

GSK Investigational Site

Redwood City, California, 94062, United States

Location

GSK Investigational Site

Reedley, California, 93654, United States

Location

GSK Investigational Site

Riverside, California, 92506, United States

Location

GSK Investigational Site

Sacramento, California, 95823, United States

Location

GSK Investigational Site

Torrance, California, 90503, United States

Location

GSK Investigational Site

Van Buys, California, 91405, United States

Location

GSK Investigational Site

Ventura, California, 93003, United States

Location

GSK Investigational Site

Victorville, California, 92395, United States

Location

GSK Investigational Site

Denver, Colorado, 80220, United States

Location

GSK Investigational Site

Trumbull, Connecticut, 06611, United States

Location

GSK Investigational Site

Bradenton, Florida, 34205, United States

Location

GSK Investigational Site

Clearwater, Florida, 33756, United States

Location

GSK Investigational Site

Fort Lauderdale, Florida, 33316, United States

Location

GSK Investigational Site

Gainesville, Florida, 32601, United States

Location

GSK Investigational Site

Jacksonville, Florida, 32204, United States

Location

GSK Investigational Site

Marianna, Florida, 32446, United States

Location

GSK Investigational Site

Miami, Florida, 33144, United States

Location

GSK Investigational Site

Oviedo, Florida, 32765, United States

Location

GSK Investigational Site

Palm Harbor, Florida, 34684, United States

Location

GSK Investigational Site

Plantation, Florida, 33317, United States

Location

GSK Investigational Site

Tallahassee, Florida, 32308, United States

Location

GSK Investigational Site

Tampa, Florida, 33603, United States

Location

GSK Investigational Site

Winter Haven, Florida, 33881, United States

Location

GSK Investigational Site

Winter Park, Florida, 32789, United States

Location

GSK Investigational Site

Athens, Georgia, 30606, United States

Location

GSK Investigational Site

Atlanta, Georgia, 30308, United States

Location

GSK Investigational Site

Atlanta, Georgia, 30312, United States

Location

GSK Investigational Site

Atlanta, Georgia, 30338, United States

Location

GSK Investigational Site

Augusta, Georgia, 30909, United States

Location

GSK Investigational Site

Columbus, Georgia, 31904, United States

Location

GSK Investigational Site

Decatur, Georgia, 30032, United States

Location

GSK Investigational Site

Perry, Georgia, 31069, United States

Location

GSK Investigational Site

Suwanee, Georgia, 30024, United States

Location

GSK Investigational Site

Tucker, Georgia, 30084, United States

Location

GSK Investigational Site

Honolulu, Hawaii, 96813, United States

Location

GSK Investigational Site

Meridian, Idaho, 83642, United States

Location

GSK Investigational Site

Aurora, Illinois, 60504, United States

Location

GSK Investigational Site

Evergreen Park, Illinois, 60805, United States

Location

GSK Investigational Site

La Grange, Illinois, 60525, United States

Location

GSK Investigational Site

Libertyville, Illinois, 60048, United States

Location

GSK Investigational Site

Oak Brook, Illinois, 60523, United States

Location

GSK Investigational Site

Watseka, Illinois, 60970, United States

Location

GSK Investigational Site

Anderson, Indiana, 46011, United States

Location

GSK Investigational Site

Indianapolis, Indiana, 46256, United States

Location

GSK Investigational Site

South Bend, Indiana, 46601, United States

Location

GSK Investigational Site

South Bend, Indiana, 46628, United States

Location

GSK Investigational Site

Ames, Iowa, 50010, United States

Location

GSK Investigational Site

Dubuque, Iowa, 52002, United States

Location

GSK Investigational Site

Kansas City, Kansas, 66160, United States

Location

GSK Investigational Site

Topeka, Kansas, 66606, United States

Location

GSK Investigational Site

Lexington, Kentucky, 40504, United States

Location

GSK Investigational Site

Covington, Louisiana, 70433, United States

Location

GSK Investigational Site

Lacombe, Louisiana, 70433, United States

Location

GSK Investigational Site

Metairie, Louisiana, 70006, United States

Location

GSK Investigational Site

Haverhill, Massachusetts, 01831-2451, United States

Location

GSK Investigational Site

Caro, Michigan, 48723, United States

Location

GSK Investigational Site

Dearborn, Michigan, 48126, United States

Location

GSK Investigational Site

Kalamazoo, Michigan, 49048, United States

Location

GSK Investigational Site

Picayune, Mississippi, 39446, United States

Location

GSK Investigational Site

Rolling Fork, Mississippi, 39159, United States

Location

GSK Investigational Site

City of Saint Peters, Missouri, 63376, United States

Location

GSK Investigational Site

Jefferson City, Missouri, 65109, United States

Location

GSK Investigational Site

Springfield, Missouri, 65807, United States

Location

GSK Investigational Site

Billings, Montana, 59101, United States

Location

GSK Investigational Site

Lincoln, Nebraska, 68516, United States

Location

GSK Investigational Site

North Platte, Nebraska, 69101, United States

Location

GSK Investigational Site

Omaha, Nebraska, 68152, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89106, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89128, United States

Location

GSK Investigational Site

Buffalo, New York, 14209, United States

Location

GSK Investigational Site

Glens Falls, New York, 12801, United States

Location

GSK Investigational Site

Rochester, New York, 14609, United States

Location

GSK Investigational Site

Syracuse, New York, 13210, United States

Location

GSK Investigational Site

Williamsville, New York, 14221, United States

Location

GSK Investigational Site

Asheville, North Carolina, 28801, United States

Location

GSK Investigational Site

Chadbourn, North Carolina, 28431, United States

Location

GSK Investigational Site

Charlotte, North Carolina, 28204, United States

Location

GSK Investigational Site

Charlotte, North Carolina, 28227, United States

Location

GSK Investigational Site

Greensboro, North Carolina, 27455, United States

Location

GSK Investigational Site

Mint Hill, North Carolina, 28227, United States

Location

GSK Investigational Site

Raleigh, North Carolina, 27609, United States

Location

GSK Investigational Site

Wilmington, North Carolina, 28401, United States

Location

GSK Investigational Site

Winston-Salem, North Carolina, 27103, United States

Location

GSK Investigational Site

Bismarck, North Dakota, 58503, United States

Location

GSK Investigational Site

Bismarck, North Dakota, 58504, United States

Location

GSK Investigational Site

Fargo, North Dakota, 58104, United States

Location

GSK Investigational Site

Fargo, North Dakota, 58122, United States

Location

GSK Investigational Site

Grand Forks, North Dakota, 58201, United States

Location

GSK Investigational Site

Cleveland, Ohio, 44122, United States

Location

GSK Investigational Site

Columbus, Ohio, 43235, United States

Location

GSK Investigational Site

Toledo, Ohio, 43606, United States

Location

GSK Investigational Site

Oklahoma City, Oklahoma, 73104, United States

Location

GSK Investigational Site

Bend, Oregon, 97701, United States

Location

GSK Investigational Site

Bensalem, Pennsylvania, 19020, United States

Location

GSK Investigational Site

Harrisburg, Pennsylvania, 17112, United States

Location

GSK Investigational Site

Morrisville, Pennsylvania, 19067, United States

Location

GSK Investigational Site

Uniontown, Pennsylvania, 15401, United States

Location

GSK Investigational Site

Watertown, South Dakota, 57201, United States

Location

GSK Investigational Site

Bristol, Tennessee, 37620, United States

Location

GSK Investigational Site

Clarksville, Tennessee, 37043, United States

Location

GSK Investigational Site

Johnson City, Tennessee, 37604, United States

Location

GSK Investigational Site

Knoxville, Tennessee, 37923, United States

Location

GSK Investigational Site

Memphis, Tennessee, 38119, United States

Location

GSK Investigational Site

Milan, Tennessee, 38358, United States

Location

GSK Investigational Site

Nashville, Tennessee, 37203, United States

Location

GSK Investigational Site

Cleburne, Texas, 76033, United States

Location

GSK Investigational Site

Dallas, Texas, 75230, United States

Location

GSK Investigational Site

Euless, Texas, 76040, United States

Location

GSK Investigational Site

Houston, Texas, 77006, United States

Location

GSK Investigational Site

Houston, Texas, 77030, United States

Location

GSK Investigational Site

Houston, Texas, 77056, United States

Location

GSK Investigational Site

Houston, Texas, 77070, United States

Location

GSK Investigational Site

Houston, Texas, 77082, United States

Location

GSK Investigational Site

LaPorte, Texas, 77571, United States

Location

GSK Investigational Site

Lewisville, Texas, 75067, United States

Location

GSK Investigational Site

Longview, Texas, 75605, United States

Location

GSK Investigational Site

Midland, Texas, 79707, United States

Location

GSK Investigational Site

Missouri City, Texas, 77459, United States

Location

GSK Investigational Site

Pasadena, Texas, 77504, United States

Location

GSK Investigational Site

Pearland, Texas, 77584, United States

Location

GSK Investigational Site

Pharr, Texas, 78577, United States

Location

GSK Investigational Site

Round Rock, Texas, 78664, United States

Location

GSK Investigational Site

San Antonio, Texas, 78205, United States

Location

GSK Investigational Site

San Marcos, Texas, 78666, United States

Location

GSK Investigational Site

Spring, Texas, 77379, United States

Location

GSK Investigational Site

Sugar Land, Texas, 77478, United States

Location

GSK Investigational Site

The Woodlands, Texas, 77381, United States

Location

GSK Investigational Site

Tomball, Texas, 77375, United States

Location

GSK Investigational Site

Salt Lake City, Utah, 84107, United States

Location

GSK Investigational Site

South Burlington, Vermont, 05403, United States

Location

GSK Investigational Site

Chester, Virginia, 23836, United States

Location

GSK Investigational Site

Manassas, Virginia, 20110, United States

Location

GSK Investigational Site

Salem, Virginia, 24153, United States

Location

GSK Investigational Site

Madison, Washington, 53717, United States

Location

GSK Investigational Site

Spokane, Washington, 99204, United States

Location

GSK Investigational Site

Concepción, Región Del Biobio, 4070038, Chile

Location

GSK Investigational Site

Buin, Región Metro de Santiago, 9500645, Chile

Location

GSK Investigational Site

Santiago, Región Metro de Santiago, 7500010, Chile

Location

GSK Investigational Site

Santiago, Región Metro de Santiago, 8320268, Chile

Location

GSK Investigational Site

Santo Domingo, Dominican Republic

Location

Related Publications (2)

  • Rosenstock J, Reusch J, Bush M, Yang F, Stewart M; Albiglutide Study Group. Potential of albiglutide, a long-acting GLP-1 receptor agonist, in type 2 diabetes: a randomized controlled trial exploring weekly, biweekly, and monthly dosing. Diabetes Care. 2009 Oct;32(10):1880-6. doi: 10.2337/dc09-0366. Epub 2009 Jul 10.

    PMID: 19592625BACKGROUND
  • Young MA, Wald JA, Matthews JE, Scott R, Hodge RJ, Zhi H, Reinhardt RR. Clinical pharmacology of albiglutide, a GLP-1 receptor agonist. Postgrad Med. 2014 Nov;126(7):84-97. doi: 10.3810/pgm.2014.11.2836.

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

rGLP-1 proteinExenatide

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

PeptidesAmino Acids, Peptides, and ProteinsVenomsComplex MixturesToxins, BiologicalBiological Factors

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 17, 2007

First Posted

August 20, 2007

Study Start

April 1, 2007

Primary Completion

May 1, 2008

Study Completion

May 1, 2008

Last Updated

December 16, 2016

Results First Posted

June 23, 2014

Record last verified: 2016-11

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Clinical Study Report (GLP110125)Access
Study Protocol (GLP110125)Access
Statistical Analysis Plan (GLP110125)Access
Informed Consent Form (GLP110125)Access
Individual Participant Data Set (GLP110125)Access
Dataset Specification (GLP110125)Access
Annotated Case Report Form (GLP110125)Access

Locations