NCT00196989

Brief Summary

This Phase 2 dose-ranging study will evaluate the efficacy, safety and tolerability of a range of doses of GW677954 compared with placebo over sixteen weeks of treatment in subjects with T2DM (Type 2 Diabetes Mellitus).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
448

participants targeted

Target at P75+ for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started Sep 2005

Typical duration for phase_2 diabetes-mellitus-type-2

Geographic Reach
12 countries

142 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2005

Completed
12 days until next milestone

First Submitted

Initial submission to the registry

September 13, 2005

Completed
7 days until next milestone

First Posted

Study publicly available on registry

September 20, 2005

Completed
1.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2007

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 1, 2007

Completed
Last Updated

March 23, 2017

Status Verified

March 1, 2017

Enrollment Period

1.6 years

First QC Date

September 13, 2005

Last Update Submit

March 21, 2017

Conditions

Keywords

EfficacyPPARpanType 2 Diabetes MellitusPhase IIbSafetyPharmacokineticsGW677954PharmacodynamicsTolerabilityDose-Ranging

Outcome Measures

Primary Outcomes (1)

  • Percentage change from Baseline (Day 1) in glycated hemoglobin (HbA1c) levels at Week 16 as a measure of improvement in glucose control

    Improvement in glucose control was measured by means of reduction in glycated hemoglobin (Hb) levels in blood.

    Week (W) 16

Secondary Outcomes (27)

  • Percentage change from Baseline (Day 1) in fasting HbA1c levels at Weeks 4, 8 and 12

    Weeks 4, 8, and 12

  • Change from Baseline (Day 1) in fasting plasma glucose (FPG) at Weeks 1, 2, 4, 6, 8, 12 and 16

    W1, W2, W4, W6, W8, W12, and W16

  • Change from Baseline (Day 1) in fasting fructosamine at Weeks 2 and 4

    Baseline (Day 1), W2, W4

  • Percentage of participants achieving target HbA1c levels at Weeks 4, 8, 12, and 16

    Weeks 4, 8, 12, and 16

  • Percentage of participants achieving a decrease in HbA1c of >= 0.7% from Baseline (Day 1) at Weeks 4, 8, 12 and 16

    Baseline (Day 1), Weeks 4, 8, 12, and 16

  • +22 more secondary outcomes

Interventions

Also known as: Pioglitazone

Eligibility Criteria

Age18 Years - 70 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects with T2DM as defined by the criteria of the ADA and/or recognized by WHO Expert Committee on the Diagnosis and Classification of Diabetes Mellitus \[American Diabetes Association, 2004\], for at least 3 months preceding screening (see Section 15.3, Appendix 3:, "Diagnosis and Classification of Diabetes Mellitus").
  • To be eligible for Randomization into the trial, a subject must satisfy all of the following glycemic criteria:
  • HbA1c level via central laboratory at the pre-screening visit
  • If HbA1c ≥ 8.0% but ≤ 10.0%: subject may proceed to Randomization;
  • If HbA1c ≥ 7.8% but \< 8.0%, subject not eligible to proceed, but may be retested once to establish eligibility (or lack thereof). If HbA1c level ≥ 8.0% upon retest, subject is eligible to proceed; otherwise they should be withdrawn.
  • If HbA1c \< 7.8%, subject not eligible to proceed (no retest allowed).
  • FPG level via central laboratory at the pre-screening visit must be \< 270 mg/dL (15.0 mmol/L). FPG may be retested within a week to confirm eligibility (or lack thereof).
  • Concurrent T2DM therapy:
  • Diet and/or exercise treated: Must not have taken antidiabetic medication for at least 2 months prior to the pre-screening visit, OR
  • Metformin monotherapy: Subjects entering the study on metformin must be on the same dose, formulation and regimen of metformin for at least 2 months prior to the pre-screening visit, AND
  • TZDs and insulin are excluded in the 3 months prior to the Screening visit for all subjects.
  • Males and females who are 18 to 70 years of age inclusive at the time of Screening.
  • If female, eligible to enter and participate in this study:
  • If of non-childbearing potential (i.e., physiologically incapable of becoming pregnant (tubal ligation), including any female who is post-menopausal \[\>1 year without menstrual period\]); or,
  • If of child-bearing potential, has a negative pregnancy test at Screening (serum), at Randomization (urine) and:
  • +8 more criteria

You may not qualify if:

  • Metabolic Disease including:
  • Diagnosis of Type 1 diabetes mellitus
  • Uncorrected thyroid dysfunction. (NOTE: subjects with hypothyroidism on a stable dose of thyroid replacement therapy for at least 1 month prior to Screening, and who have a screening thyroid stimulating hormone (TSH) within the upper limit of normal may participate).
  • Significant weight gain or loss (defined as \> 5% of total body weight) within the 3 months prior to Screening.
  • Previous use of insulin for treatment of hyperglycemia within 3 months of Screening.
  • History of recent clinically significant cardiovascular disease including:
  • History or ECG evidence of prior myocardial infarction within 6 months prior to Screening.
  • Current unstable angina or history of unstable angina in past 6 months.
  • Coronary revascularization including percutaneous transluminal coronary angioplasty (PTCA) or coronary artery bypass graft (CABG) surgery that is either planned or occurred in the 6 months prior to Screening.
  • Clinically significant arrhythmia or valvular heart disease.
  • Congestive heart failure (CHF) with New York Heart Association (NYHA) Class II-IV symptoms (see Section 15.4, Appendix 4).
  • Blood pressure \> 160/100 mmHg or resting heart rate \> 100 bpm. Note: subjects using antihypertensives \[e.g., beta blockers, angiotensin converting enzyme (ACE) inhibitors, angiotensin II antagonists, calcium channel blockers and diuretics\] must be on stable doses during the 30 days prior to Screening and during the trial.
  • Has a QTc interval (Bazett's) \> 440 msec in males and \> 450 msec in females at Screening.
  • Clinically significant ECG abnormalities which, in the opinion of the Investigator, may affect the interpretation of safety data, or which otherwise, contraindicates participation in a clinical trial with a new chemical entity.
  • History of chronic pancreatitis.
  • +40 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (143)

GSK Investigational Site

Birmingham, Alabama, 35205, United States

Location

GSK Investigational Site

Northport, Alabama, 35476, United States

Location

GSK Investigational Site

Chandler, Arizona, 85224, United States

Location

GSK Investigational Site

Phoenix, Arizona, 85006, United States

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GSK Investigational Site

Phoenix, Arizona, 85032, United States

Location

GSK Investigational Site

Alhambra, California, 91801, United States

Location

GSK Investigational Site

Artesia, California, 90701, United States

Location

GSK Investigational Site

Huntington Beach, California, 92648, United States

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GSK Investigational Site

Inglewood, California, 90301, United States

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GSK Investigational Site

Irvine, California, 92618, United States

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GSK Investigational Site

La Jolla, California, 92037, United States

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GSK Investigational Site

Long Beach, California, 90806, United States

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GSK Investigational Site

Los Angeles, California, 90057, United States

Location

GSK Investigational Site

Los Angeles, California, 90095, United States

Location

GSK Investigational Site

Northridge, California, 91325, United States

Location

GSK Investigational Site

Norwalk, California, 90650, United States

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GSK Investigational Site

Pasadena, California, 91105, United States

Location

GSK Investigational Site

Sacramento, California, 95825, United States

Location

GSK Investigational Site

San Diego, California, 92128, United States

Location

GSK Investigational Site

San Diego, California, 92177, United States

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GSK Investigational Site

Santa Monica, California, 90404, United States

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GSK Investigational Site

Tustin, California, 92780, United States

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GSK Investigational Site

Vista, California, 92084, United States

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GSK Investigational Site

West Hills, California, 91307, United States

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GSK Investigational Site

Denver, Colorado, 80220, United States

Location

GSK Investigational Site

Norwich, Connecticut, 06360, United States

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GSK Investigational Site

Hollywood, Florida, 33021, United States

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GSK Investigational Site

Hollywood, Florida, 33023, United States

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GSK Investigational Site

Largo, Florida, 33773, United States

Location

GSK Investigational Site

Miami, Florida, 33156, United States

Location

GSK Investigational Site

Saint Cloud, Florida, 34769, United States

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GSK Investigational Site

Sarasota, Florida, 34239, United States

Location

GSK Investigational Site

Atlanta, Georgia, 30342, United States

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GSK Investigational Site

Duluth, Georgia, 30097, United States

Location

GSK Investigational Site

Honolulu, Hawaii, 96813, United States

Location

GSK Investigational Site

Springfield, Illinois, 62701, United States

Location

GSK Investigational Site

Indianapolis, Indiana, 46260, United States

Location

GSK Investigational Site

West Yarmouth, Massachusetts, 02673, United States

Location

GSK Investigational Site

St Louis, Missouri, 63110, United States

Location

GSK Investigational Site

St Louis, Missouri, 63141, United States

Location

GSK Investigational Site

Henderson, Nevada, 89014, United States

Location

GSK Investigational Site

Henderson, Nevada, 89015, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89106, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89119, United States

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GSK Investigational Site

Las Vegas, Nevada, 89128, United States

Location

GSK Investigational Site

Pahrump, Nevada, 89048, United States

Location

GSK Investigational Site

Albuquerque, New Mexico, 87102, United States

Location

GSK Investigational Site

Santa Fe, New Mexico, 87505, United States

Location

GSK Investigational Site

New York, New York, 10024, United States

Location

GSK Investigational Site

New York, New York, 10032, United States

Location

GSK Investigational Site

Greensboro, North Carolina, 27401, United States

Location

GSK Investigational Site

Cleveland, Ohio, 44195, United States

Location

GSK Investigational Site

Franklin, Ohio, 45005, United States

Location

GSK Investigational Site

Philadelphia, Pennsylvania, 19107, United States

Location

GSK Investigational Site

East Providence, Rhode Island, 02914, United States

Location

GSK Investigational Site

Greer, South Carolina, 29651, United States

Location

GSK Investigational Site

Simpsonville, South Carolina, 29681, United States

Location

GSK Investigational Site

Cite, Tennessee, 37604, United States

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GSK Investigational Site

Kingsport, Tennessee, 37660, United States

Location

GSK Investigational Site

Dallas, Texas, 75246, United States

Location

GSK Investigational Site

San Antonio, Texas, 78229, United States

Location

GSK Investigational Site

Tyler, Texas, 75708, United States

Location

GSK Investigational Site

Salt Lake City, Utah, 84109, United States

Location

GSK Investigational Site

West Jordan, Utah, 84084, United States

Location

GSK Investigational Site

Virginia Beach, Virginia, 23451, United States

Location

GSK Investigational Site

Edmonds, Washington, 98026, United States

Location

GSK Investigational Site

Everett, Washington, 98208, United States

Location

GSK Investigational Site

Monroe, Washington, 98272, United States

Location

GSK Investigational Site

Wauwatosa, Wisconsin, 53226, United States

Location

GSK Investigational Site

Buenos Aires, Buenos Aires, 1425, Argentina

Location

GSK Investigational Site

Capital Federal, Buenos Aires, 1181, Argentina

Location

GSK Investigational Site

Capital Federal, Buenos Aires, C1221ACI, Argentina

Location

GSK Investigational Site

Córdoba, Córdoba Province, 5000, Argentina

Location

GSK Investigational Site

San Juan, 5400, Argentina

Location

GSK Investigational Site

Miranda, New South Wales, 2228, Australia

Location

GSK Investigational Site

Carina Heights, Queensland, 4152, Australia

Location

GSK Investigational Site

Spring Hill, Queensland, 4000, Australia

Location

GSK Investigational Site

Adelaide, South Australia, 5000, Australia

Location

GSK Investigational Site

Keswick, South Australia, 5035, Australia

Location

GSK Investigational Site

Port Lincoln, South Australia, 5606, Australia

Location

GSK Investigational Site

Box Hill, Victoria, 3128, Australia

Location

GSK Investigational Site

Ringwood East, Victoria, 3135, Australia

Location

GSK Investigational Site

Langley, British Columbia, V3A 4H9, Canada

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GSK Investigational Site

Winnipeg, Manitoba, R3E 3P4, Canada

Location

GSK Investigational Site

St. John's, Newfoundland and Labrador, A1E 2C2, Canada

Location

GSK Investigational Site

Halifax, Nova Scotia, B3K 5R3, Canada

Location

GSK Investigational Site

Brampton, Ontario, L6T 3J1, Canada

Location

GSK Investigational Site

Greater Sudbury, Ontario, P3A 1Y8, Canada

Location

GSK Investigational Site

London, Ontario, N5W 6A2, Canada

Location

GSK Investigational Site

Mississauga, Ontario, L5A 1N1, Canada

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GSK Investigational Site

Ottawa, Ontario, K1H 1A2, Canada

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GSK Investigational Site

Smiths Falls, Ontario, K7A 4W8, Canada

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GSK Investigational Site

Thornhill, Ontario, L4J 8L7, Canada

Location

GSK Investigational Site

Toronto, Ontario, M4R 2G4, Canada

Location

GSK Investigational Site

Toronto, Ontario, M9W 4L6, Canada

Location

GSK Investigational Site

Waterloo, Ontario, N2J 1C4, Canada

Location

GSK Investigational Site

Bonaventure, Quebec, G0C 1E0, Canada

Location

GSK Investigational Site

Granby, Quebec, J2G 8Z9, Canada

Location

GSK Investigational Site

Laval, Quebec, H7T 2P5, Canada

Location

GSK Investigational Site

Longueuil, Quebec, J4N 1L6, Canada

Location

GSK Investigational Site

Montreal, Quebec, H4N 2W2, Canada

Location

GSK Investigational Site

Québec, Quebec, G1W 4R4, Canada

Location

GSK Investigational Site

Saint-Marc-des-Carrieres, Quebec, G0A 4B0, Canada

Location

GSK Investigational Site

Sainte-Foy, Quebec, G1V 1V6, Canada

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GSK Investigational Site

Sainte-Foy, Quebec, G1V 4G2, Canada

Location

GSK Investigational Site

Sainte-Foy, Quebec, G1V 4G5, Canada

Location

GSK Investigational Site

Sherbrooke, Quebec, J1G 5K2, Canada

Location

GSK Investigational Site

Bogotá, Colombia

Location

GSK Investigational Site

San José, Provincia de San José, Costa Rica

Location

GSK Investigational Site

Cheb, 350 02, Czechia

Location

GSK Investigational Site

České Budějovice, 370 87, Czechia

Location

GSK Investigational Site

Olomouc, 779 00, Czechia

Location

GSK Investigational Site

Prague, 10000, Czechia

Location

GSK Investigational Site

Prague, 128 08, Czechia

Location

GSK Investigational Site

Prague, 15030, Czechia

Location

GSK Investigational Site

Prague, 158 00, Czechia

Location

GSK Investigational Site

Quito, Ecuador

Location

GSK Investigational Site

Cēsis, LV4100, Latvia

Location

GSK Investigational Site

Daugavpils, LV5417, Latvia

Location

GSK Investigational Site

Riga, LV 1002, Latvia

Location

GSK Investigational Site

Riga, LV1024, Latvia

Location

GSK Investigational Site

Tukums, LV 3100, Latvia

Location

GSK Investigational Site

Tijuana, Baja California Norte, 22320, Mexico

Location

GSK Investigational Site

Durango, Durango, 3400, Mexico

Location

GSK Investigational Site

Pachuca, Hidalgo, 42039, Mexico

Location

GSK Investigational Site

Cuernavaca, Morelos, 62420, Mexico

Location

GSK Investigational Site

Monterrey, Nuevo León, 64570, Mexico

Location

GSK Investigational Site

Mexico City, 11650, Mexico

Location

GSK Investigational Site

Auckland, 1309, New Zealand

Location

GSK Investigational Site

Auckland, 1311, New Zealand

Location

GSK Investigational Site

Christchurch, 8001, New Zealand

Location

GSK Investigational Site

Rotorua, 3201, New Zealand

Location

GSK Investigational Site

Tauranga, 3001, New Zealand

Location

GSK Investigational Site

Lima, Lima Province, Lima 14, Peru

Location

GSK Investigational Site

Lima, Lima Province, Lima 27, Peru

Location

GSK Investigational Site

San Isidro, Lima region, Lima 27, Peru

Location

GSK Investigational Site

Lima, Lima 1, Peru

Location

GSK Investigational Site

Moscow, 117 036, Russia

Location

GSK Investigational Site

Perm, 614600, Russia

Location

GSK Investigational Site

Samara, 443067, Russia

Location

GSK Investigational Site

Tyumen, 625023, Russia

Location

GSK Investigational Site

Ufa, 450000, Russia

Location

GSK Investigational Site

Yaroslavl, 150062, Russia

Location

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

Pioglitazone

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

ThiazolidinedionesThiazolesSulfur CompoundsOrganic ChemicalsAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 13, 2005

First Posted

September 20, 2005

Study Start

September 1, 2005

Primary Completion

April 1, 2007

Study Completion

April 1, 2007

Last Updated

March 23, 2017

Record last verified: 2017-03

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Clinical Study Report (ADG20001)Access
Informed Consent Form (ADG20001)Access
Dataset Specification (ADG20001)Access
Statistical Analysis Plan (ADG20001)Access
Individual Participant Data Set (ADG20001)Access
Annotated Case Report Form (ADG20001)Access
Study Protocol (ADG20001)Access

Locations