NCT00460512

Brief Summary

The purpose of this study is to explore tolerability, safety and effectiveness of flexibly dosed paliperidone extended release (ER) in participants with schizophrenia (psychiatric disorder with symptoms of emotional instability, detachment from reality, often with delusions and hallucinations, and withdrawal into the self) previously unsuccessfully treated with an oral antipsychotic medication.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,814

participants targeted

Target at P75+ for phase_3 schizophrenia

Timeline
Completed

Started Apr 2007

Longer than P75 for phase_3 schizophrenia

Geographic Reach
21 countries

228 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 13, 2007

Completed
3 days until next milestone

First Posted

Study publicly available on registry

April 16, 2007

Completed
9 days until next milestone

Study Start

First participant enrolled

April 25, 2007

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 22, 2009

Completed
11.1 years until next milestone

Study Completion

Last participant's last visit for all outcomes

March 4, 2020

Completed
Last Updated

April 27, 2025

Status Verified

April 1, 2025

Enrollment Period

1.7 years

First QC Date

April 13, 2007

Last Update Submit

April 25, 2025

Conditions

Keywords

SchizophreniaFlexible dosingNon-acute patientsAntipsychoticAtypicalINVEGA

Outcome Measures

Primary Outcomes (2)

  • Percentage of Participants With at Least 20 Percent Improvement in Total Positive and Negative Syndrome Scale (PANSS) Score in Those Participants who Transitioned due to Lack of Efficacy

    The PANSS is a 30-item scale to assess the neuropsychiatric symptoms of schizophrenia (psychiatric disorder with symptoms of emotional instability, detachment from reality, often with delusions and hallucinations, and withdrawal into the self). The PANSS provides a total score and scores for 3 subscales, the positive subscale (7 items), the negative subscale (7 items), and the general psychopathology subscale (16 items), each item scored on a scale of 1 (absent) to 7 (extreme). The total score ranges from 30 to 210 and higher score indicates greater severity.

    Endpoint (up to Week 26)

  • Change From Baseline in Positive and Negative Syndrome Scale (PANSS) Total Score at Endpoint (up to Week 26)

    The PANSS is a 30-item scale to assess the neuropsychiatric symptoms of schizophrenia. The PANSS provides a total score and scores for 3 subscales, the positive subscale (7 items), the negative subscale (7 items), and the general psychopathology subscale (16 items), each item scored on a scale of 1 (absent) to 7 (extreme). The total score ranges from 30 to 210 and higher score indicates greater severity.

    Baseline and endpoint (up to Week 26)

Secondary Outcomes (9)

  • Percentage of Participants With at Least 20 Percent Improvement in Total Positive and Negative Syndrome Scale (PANSS) Score

    Endpoint (up to Week 26)

  • Change From Baseline in Positive and Negative Syndrome Scale (PANSS) Subscale Scores at Endpoint (up to Week 26)

    Baseline and endpoint (up to Week 26)

  • Change From Baseline in Positive and Negative Syndrome Scale (PANSS) Marder Subscale Scores at Endpoint (up to Week 26)

    Baseline and endpoint (up to Week 26)

  • Change From Baseline in Clinical Global Impression-Severity (CGI-S) Score at Endpoint (up to Week 26)

    Baseline and endpoint (up to Week 26)

  • Change From Baseline in Total Personal and Social Performance (PSP) Score at Endpoint (up to Week 26)

    Baseline and endpoint (up to Week 26)

  • +4 more secondary outcomes

Study Arms (1)

Paliperidone Extended Release (ER)

EXPERIMENTAL
Drug: Paliperidone ER

Interventions

Paliperidone ER tablet in dose range of 3 to12 milligram (mg) per day was given orally for 6 months as per Investigator's discretion to participants who transitioned to Paliperidone ER from other oral antipsychotics due to lack of efficacy, lack of tolerability, lack of compliance or other reasons.

Paliperidone Extended Release (ER)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participant meets the Diagnostic and Statistical Manual of Mental Disorders (Edition 4) criteria for schizophrenia
  • Participant is previously non-acute (on the same antipsychotic medication used for the treatment of schizophrenia and Clinical Global Impression-Severity \[CGI-S\] change less than or equal to 1 in the past 4 weeks before enrollment) and has been given an adequate dose of an appropriate oral antipsychotic for an adequate period of time prior to enrollment, but previous treatment is considered unsuccessful due to one or more of the following reasons: lack of effectiveness, lack of tolerability or safety, lack of compliance and/or other reasons to switch to another antipsychotic medication
  • Participant is healthy on the basis of a physical examination and vital signs at screening
  • Female participants must be postmenopausal for at least 1 year, surgically sterile, abstinent, or, if sexually active, agree to practice an effective method of birth control before entry and throughout the study
  • Participants must be willing and able to fill out self-administered questionnaires

You may not qualify if:

  • Participants on clozapine, any conventional depot neuroleptic or risperidone long-acting injection during the last 3 months
  • Participants with serious unstable medical condition, including known clinically relevant laboratory abnormalities
  • Participants with history or current symptoms of tardive dyskinesia (twitching or jerking movements that you cannot control in your face, tongue, or other parts of your body) and neuroleptic malignant syndrome (high fever, rigid muscles, shaking, confusion, sweating more than usual, increased heart rate or blood pressure, or muscle pain or weakness)
  • Participants judged to be at high risk for adverse events, violence or self-harm
  • Participants with a current use or known history (over the past 6 months) of substance dependence according to Diagnostic and Statistical Manual of Mental Disorders (Edition 4) Criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (231)

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Antwerp, Belgium

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Bertrix, Belgium

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Dave, Belgium

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Diest, Belgium

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Duffel, Belgium

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Kortenberg, Belgium

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Liège, Belgium

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Montignies-sur-Sambre, Belgium

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Mortsel, Belgium

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Roeselare, Belgium

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Saint Denijs-Westrem, Belgium

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Saint-Servais, Belgium

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Sint-Truiden, Belgium

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Tielt, Belgium

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Waregem, Belgium

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Bulgaria, Bulgaria

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Sofia, Bulgaria

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Tzerova Korya, Bulgaria

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Osijek, Croatia

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Rijeka, Croatia

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Split, Croatia

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Zagreb, Croatia

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Aalborg, Denmark

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Elsinore, Denmark

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Risskov, Denmark

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Viby J, Denmark

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Ekenäs, Finland

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Helsinki, Finland

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Raahe, Finland

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Tampere, Finland

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Bar-le-Duc, France

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Bordeaux, France

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Bourg-en-Bresse, France

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Bully-les-Mines, France

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Caen, France

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Chambéry, France

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Clermont-Ferrand, France

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Créteil, France

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Dijon, France

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Dole, France

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Henin Baumont, France

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Jarnac, France

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La Roche-sur-Yon, France

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La Seyne-sur-Mer, France

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Mont-Saint-Martin, France

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Montpellier, France

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Nîmes, France

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Paris, France

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Pau, France

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Rennes, France

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Roubaix, France

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Saint-Avé, France

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Saint-Cyr-au-Mont-d'Or, France

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Saint-Germain-en-Laye, France

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Villejuif, France

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Aalen, Germany

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Achim, Germany

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Augsburg, Germany

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Bamberg, Germany

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Bergfelde, Germany

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Bergheim, Germany

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Berlin, Germany

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Bochum, Germany

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Butzbach, Germany

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Chemnitz, Germany

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Coesfeld, Germany

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Cologne, Germany

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Darmstadt, Germany

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Dillingen, Germany

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Dresden, Germany

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Duisburg, Germany

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Düsseldorf, Germany

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Ebensfeld, Germany

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Eberbach, Germany

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Ellwangen, Germany

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Elmshorn, Germany

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Essen, Germany

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Ettlingen, Germany

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Freiburg im Breisgau, Germany

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Gelnhausen, Germany

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Gelsenkirchen, Germany

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Giessen, Germany

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Göttingen, Germany

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Haina, Germany

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Halle, Germany

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Hamburg, Germany

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Hanover, Germany

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Hattingen, Germany

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Hemer, Germany

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Hemmoor, Germany

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Heppenheim an der Bergstrasse, Germany

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Idar-Oberstein, Germany

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Jena, Germany

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Kaufbeuren, Germany

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Königsbrück, Germany

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Krefeld, Germany

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Leipzig, Germany

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Liebenburg, Germany

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Lüdenscheid, Germany

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Mainz, Germany

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Mannheim, Germany

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Mittweida, Germany

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München, Germany

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Münster, Germany

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Naumburg, Germany

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Norden, Germany

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Nuremberg, Germany

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Ober-Ramstadt, Germany

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Oldenburg, Germany

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Oranienburg, Germany

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Ostfildern, Germany

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Potsdam, Germany

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Rostock, Germany

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Saalfeld, Germany

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Salzgitter, Germany

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Schlüchtern, Germany

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Siegen, Germany

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Spremberg, Germany

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Stralsund, Germany

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Straubing, Germany

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Ulm, Germany

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Viersen, Germany

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Wasserburg, Germany

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Wiesbaden, Germany

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Wiesloch, Germany

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Wilhelmshaven, Germany

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Wismar, Germany

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Würzburg, Germany

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Athens, Greece

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Chios, Greece

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Heraklion, Greece

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Larissa, Greece

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Thessalonikis, Greece

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Balassagyarmat, Hungary

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Budapest, Hungary

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Kecskemét, Hungary

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Sopron, Hungary

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Bat Yam, Israel

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Be'er Ya'acov, Israel

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Jerusalem, Israel

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Pardesiyya, Israel

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Daugavpils, Latvia

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Jelgava, Latvia

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Liepāja, Latvia

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Riga, Latvia

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Strenči, Latvia

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Kaunas, Lithuania

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Panevezys, Lithuania

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Vilnius, Lithuania

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Assen, Netherlands

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Beilen, Netherlands

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Bennebroek, Netherlands

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Enschede, Netherlands

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Groningen, Netherlands

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Hoofddorp, Netherlands

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Leeuwarden, Netherlands

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The Hague, Netherlands

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Tilburg, Netherlands

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Zwolle, Netherlands

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Bydgoszcz, Poland

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Gdynia Na, Poland

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Krakow Na, Poland

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Lubliniec, Poland

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Skorzewo Na, Poland

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Angra do Heroísmo, Portugal

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Braga, Portugal

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Castelo Viegas, Portugal

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Coimbra, Portugal

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Lisbon, Portugal

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Porto, Portugal

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Kazan', Russia

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Krasnodar, Russia

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Moscow, Russia

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Moscow Russia, Russia

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Saint Peterburg Na, Russia

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Saint Petersburg, Russia

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Saratov, Russia

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Yaroslavl, Russia

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Belgrade, Serbia

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Kragujevac, Serbia

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Novi Sad, Serbia

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Alicante, Spain

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Barcelona, Spain

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Bunyola Illes Balears, Spain

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Burgos, Spain

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Oviedo, Spain

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Pontevedra, Spain

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Sama de Langreo Asturias, Spain

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Valencia, Spain

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Zamora, Spain

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Zaragoza, Spain

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Bromma, Sweden

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Gothenburg, Sweden

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Hudiksvall, Sweden

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Karlskrona, Sweden

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Malmo, Sweden

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Mölndal, Sweden

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Norrtälje, Sweden

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Nyköping, Sweden

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Simrishamn, Sweden

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Skövde, Sweden

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Solna, Sweden

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Trollhättan, Sweden

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Västra Frölunda, Sweden

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Aarau, Switzerland

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Basel, Switzerland

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Basel Bs, Switzerland

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Biel/Bienne, Switzerland

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Geneva, Switzerland

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Lenzburg, Switzerland

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Liestal, Switzerland

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Marsens, Switzerland

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Montreux, Switzerland

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Münsingen, Switzerland

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Oetwil, Switzerland

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Riehen, Switzerland

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Sarnen, Switzerland

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Solothurn, Switzerland

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Viganello, Switzerland

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Zurich, Switzerland

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Ankara, Turkey (Türkiye)

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Denizli, Turkey (Türkiye)

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Diyarbakır, Turkey (Türkiye)

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Gaziantep, Turkey (Türkiye)

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Izmir, Turkey (Türkiye)

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Barnet, United Kingdom

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Birmingham, United Kingdom

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Clacton-on-Sea, United Kingdom

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Devon, United Kingdom

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Exeter, United Kingdom

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Glasgow, United Kingdom

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Related Publications (1)

  • Schreiner A, Lahaye M, Peuskens J, Naber D, Dilbaz N, Millet B, Franco MA, Rancans E, Turczynski J, Smeraldi E, Lara E, Neznanov NG. Paliperidone extended-release in patients with non-acute schizophrenia previously unsuccessfully treated with other oral antipsychotics. Expert Opin Pharmacother. 2014 Apr;15(5):593-603. doi: 10.1517/14656566.2014.884071. Epub 2014 Feb 3.

MeSH Terms

Conditions

Schizophrenia

Interventions

Paliperidone Palmitate

Condition Hierarchy (Ancestors)

Schizophrenia Spectrum and Other Psychotic DisordersMental Disorders

Intervention Hierarchy (Ancestors)

IsoxazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrimidines

Study Officials

  • Janssen-Cilag International NV Clinical Trial

    Janssen-Cilag International NV

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 13, 2007

First Posted

April 16, 2007

Study Start

April 25, 2007

Primary Completion

January 22, 2009

Study Completion

March 4, 2020

Last Updated

April 27, 2025

Record last verified: 2025-04

Locations