NCT00411866

Brief Summary

The purposes of this study are to determine if there is a difference in how SB-773812 is distributed through the bloodstream before and after multiple doses of ketoconazole have been given and to determine if there is a difference in how safe and well tolerated SB-773812 is when given on its own and given with ketoconazole.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
36

participants targeted

Target at P25-P50 for phase_1 schizophrenia

Timeline
Completed

Started Oct 2006

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

October 13, 2006

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

December 13, 2006

Completed
2 days until next milestone

First Posted

Study publicly available on registry

December 15, 2006

Completed
10 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 10, 2007

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 10, 2007

Completed
Last Updated

August 3, 2017

Status Verified

August 1, 2017

Enrollment Period

12 months

First QC Date

December 13, 2006

Last Update Submit

August 2, 2017

Conditions

Keywords

safetypharmacokinetics,

Outcome Measures

Primary Outcomes (1)

  • Blood sampling over period of 336 hours post dosing with SB-773812

    over period of 336 hours post dosing

Secondary Outcomes (1)

  • Safety: ECG, vital signs, adverse events, clinical labs over 48 hours post SB-773812 dosing.

    over 48 hours post SB-773812 dosing.

Study Arms (2)

Subjects receiving ketoconazole for 8 days

EXPERIMENTAL

In Session 1, subjects will receive a single oral dose of SB-773812 20 milligrams (mg), followed by 21 days-washout. In Session 2, subjects will receive once daily oral dose of ketoconazole 400 mg repeated for 8 days. On day 5, single oral dose of SB-773812 20 mg will be dosed concomitantly with ketoconazole.

Drug: SB773812Drug: Ketoconazole

Subjects receiving ketoconazole for 14 days

EXPERIMENTAL

In Session 1, subjects will receive a single oral dose of SB-773812 (20mg), followed by 21 days-washout. In Session 2, subjects will receive once daily oral dose of ketoconazole 400 mg repeated for 12 days. On day 5, single oral dose of SB-773812 20 mg will be dosed concomitantly with ketoconazole.

Drug: SB773812Drug: Ketoconazole

Interventions

SB-773812 20 mg will be available as white round film coated tablets.

Subjects receiving ketoconazole for 14 daysSubjects receiving ketoconazole for 8 days

Ketoconazole will be available as 200mg tablets.

Also known as: SB773812
Subjects receiving ketoconazole for 14 daysSubjects receiving ketoconazole for 8 days

Eligibility Criteria

Age18 Years - 55 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy
  • Body Weight \>/=50kg and BMI 18.5-29.9 kg/m2 inclusive
  • Normal 12-lead ECG, physical examination and lab screen

You may not qualify if:

  • A history of psychiatric illness,
  • A history or presence gastro-intestinal,
  • A hepatic or renal disease or orthostatic hypotension.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

GSK Investigational Site

Dundee, DD1 9SY, United Kingdom

Location

Related Links

MeSH Terms

Conditions

Schizophrenia

Interventions

Ketoconazole

Condition Hierarchy (Ancestors)

Schizophrenia Spectrum and Other Psychotic DisordersMental Disorders

Intervention Hierarchy (Ancestors)

PiperazinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
DIAGNOSTIC
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 13, 2006

First Posted

December 15, 2006

Study Start

October 13, 2006

Primary Completion

October 10, 2007

Study Completion

October 10, 2007

Last Updated

August 3, 2017

Record last verified: 2017-08

Locations