NCT00330369

Brief Summary

This is a research study of a new experimental drug called darusentan. Darusentan is not currently approved by the U.S. Food and Drug Administration (FDA) for use in the United States, which means that a doctor cannot prescribe this drug. The purpose of this study is to determine if darusentan is effective in reducing systolic blood pressure in subjects with resistant systolic hypertension, despite treatment with full doses of three or more antihypertensive drugs, including a diuretic.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
352

participants targeted

Target at P50-P75 for phase_3 hypertension

Timeline
Completed

Started Jun 2006

Typical duration for phase_3 hypertension

Geographic Reach
11 countries

115 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 24, 2006

Completed
2 days until next milestone

First Posted

Study publicly available on registry

May 26, 2006

Completed
6 days until next milestone

Study Start

First participant enrolled

June 1, 2006

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2009

Completed
Last Updated

March 18, 2014

Status Verified

February 1, 2014

Enrollment Period

2.6 years

First QC Date

May 24, 2006

Last Update Submit

February 19, 2014

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change from baseline in trough sitting systolic and diastolic blood pressure measured by sphygmomanometry

    Baseline to Week 14

Secondary Outcomes (3)

  • Change from baseline in mean 24-hour systolic and diastolic ambulatory blood pressure

    Baseline to Week 14

  • Percentage of subjects to reach systolic blood pressure goal

    Week 14

  • Change from baseline in estimated glomerular filtration rate (eGFR)

    Baseline to Week 14

Study Arms (4)

Darusentan Placebo

PLACEBO COMPARATOR

Placebo to match darusentan for 2-week placebo run-in period, followed by placebo to match darusentan administered orally once daily for 14 weeks

Drug: Darusentan Placebo

Darusentan 50 mg

EXPERIMENTAL

Placebo to match darusentan for 2-week placebo run-in period, followed by darusentan 50 mg administered orally once daily for 14 weeks

Drug: DarusentanDrug: Darusentan Placebo

Darusentan 100 mg

EXPERIMENTAL

Placebo to match darusentan for 2-week placebo run-in period, followed by darusentan 100 mg administered orally once daily for 14 weeks

Drug: DarusentanDrug: Darusentan Placebo

Darusentan 300 mg

EXPERIMENTAL

Placebo to match darusentan for 2-week placebo run-in period, followed by darusentan 300 mg administered orally once daily for 14 weeks

Drug: DarusentanDrug: Darusentan Placebo

Interventions

Darusentan administered orally once daily

Also known as: LU 135252
Darusentan 100 mgDarusentan 300 mgDarusentan 50 mg

Placebo to match darusentan administered orally once daily

Darusentan 100 mgDarusentan 300 mgDarusentan 50 mgDarusentan Placebo

Eligibility Criteria

Age35 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects who are competent to provide written consent
  • Aged 35 to 80 years
  • Subjects with diabetes and/or chronic kidney disease must have a mean systolic blood pressure ≥130 mmHg
  • All other subjects must have a mean systolic blood pressure ≥140 mmHg
  • Receiving and adhering to full doses of appropriate guideline-recommended antihypertensive drugs from three different classes of antihypertensive agents, including a diuretic
  • Female subjects of non-childbearing potential (i.e., post-menopausal for at lest 2 years; surgically sterile)

You may not qualify if:

  • Average sitting systolic blood pressure ≥180 mmHg or diastolic blood pressure ≥110 mmHg
  • Serum ALT or AST \>2 x the upper limit of the normal range (ULN)
  • Subjects who have experienced myocardial infarction, unstable angina pectoris, or a cerebrovascular accident (CVA) within 6 month; or sick sinus syndrome or second or third degree atrioventricular block, atrial fibrillation or recurrent atrial tachyarrhythmia, recurrent ventricular tachycardia, or symptomatic bradycardia
  • Implanted pacemakers or implanted cardioverter defibrillator (ICD)
  • Symptomatic congestive heart failure requiring treatment
  • Hemodynamically significant valvular heart disease
  • Type I diabetes mellitus
  • Hemodialysis or peritoneal dialysis; or history of renal transplant
  • Diagnosis or recurrence of malignancy within the past 3 years
  • Sleep apnea, unless a recent sleep study demonstrates arterial oxygen saturation greater than or equal to 90%
  • Subjects who perform alternating shift or night work
  • Subjects who have participated in a clinical study involving another investigational drug or device within 4 weeks prior to Screening

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (115)

UAB Hypertension Program

Birmingham, Alabama, 35294, United States

Location

Comprehensive Heart Failure Center

Mobile, Alabama, 36608, United States

Location

Canyon Clinical Research

Tucson, Arizona, 85712, United States

Location

Chrishard Medical Group

Inglewood, California, 90301, United States

Location

VA Medical Center - WLA

Los Angeles, California, 90073, United States

Location

Sacramento Heart and Vascular

Sacramento, California, 95825, United States

Location

Apex Research Institute

Santa Ana, California, 92705, United States

Location

Complete Renal Care

Denver, Colorado, 80220, United States

Location

Connecticut Clinical Research, LLC

Bridgeport, Connecticut, 06606, United States

Location

MedStar Diabetes Institute at Washington Hospital Center

Washington D.C., District of Columbia, 20010, United States

Location

Deerfield Beach Cardiology Associates

Deerfield Beach, Florida, 33442, United States

Location

White-Wilson Medical Center

Fort Walton Beach, Florida, 32569, United States

Location

AMK Research

Gainsville, Florida, 32601, United States

Location

A.G.A. Clinical Trials

Hialeah, Florida, 33012, United States

Location

Jacksonville Center for Clinical

Jacksonville, Florida, 32216, United States

Location

Ricardo A. Bedoya, Cardiology

Jupiter, Florida, 33458, United States

Location

International Research Association

Miami, Florida, 33156, United States

Location

Cardiovascular Center of Sarasota

Sarasota, Florida, 34239, United States

Location

Tampa Bay Nephrology

Tampa, Florida, 33603, United States

Location

Metabolic Research Institute, Inc.

West Palm Beach, Florida, 33401, United States

Location

Global Research Partners

Calhoun, Georgia, 30701, United States

Location

Kula Research

Honolulu, Hawaii, 96816, United States

Location

Chicago Heart & Vein Clinic

Elk Grove Village, Illinois, 60007, United States

Location

Evanston Northwestern Healthcare

Evanston, Illinois, 60201, United States

Location

Clinical Investigation Specialists, Inc.

Gurnee, Illinois, 60031, United States

Location

Midwest Heart Foundation

Lombard, Illinois, 60148, United States

Location

American Clinical Research LLC

Marrero, Louisiana, 70072, United States

Location

Medical Research Institute

Slidell, Louisiana, 70458, United States

Location

Maine Research Associates

Auburn, Maine, 04210, United States

Location

Cardiovascular Consultants of Maine

Scarborough, Maine, 04074, United States

Location

MODEL Clinical Research

Baltimore, Maryland, 21204, United States

Location

Maryland Medical Research/Og Medical Center

Oxon Hill, Maryland, 20745, United States

Location

Clinical Associates

Reisterstown, Maryland, 21136, United States

Location

Rockville Internal Medicine Group

Rockville, Maryland, 20854, United States

Location

Professional Clinical Research

Benzonia, Michigan, 49616, United States

Location

Nephrology and Hypertension / Hurley Medical Center

Flint, Michigan, 48503, United States

Location

Professional Clinical Research

Interlochen, Michigan, 49643, United States

Location

Specialty Medical Center

Pahrump, Nevada, 89048, United States

Location

Bronx VA Medical Center / Mt. Sinai

The Bronx, New York, 10468, United States

Location

Physicians East, PA

Greenville, North Carolina, 27834, United States

Location

The Lindner Clinical Trial Center

Cincinnati, Ohio, 45219, United States

Location

West Coast Cardiology Associates

Fairview Park, Ohio, 44125, United States

Location

COR Clinical Research

Oklahoma City, Oklahoma, 73003, United States

Location

Southwest Cardiology Associates

Oklahoma City, Oklahoma, 73109, United States

Location

Sooner Clinical Research

Oklahoma City, Oklahoma, 73112, United States

Location

Castlerock Clinical Research Consultants

Tulsa, Oklahoma, 74136, United States

Location

Hillsboro Cardiology, PC

Hillsboro, Oregon, 97123, United States

Location

Northeast Clinical Research Centers, Inc.

Allentown, Pennsylvania, 18103, United States

Location

Heritage Cardiology Associates

Camp Hill, Pennsylvania, 17011, United States

Location

Brandywine Clinical Research

Downingtown, Pennsylvania, 19335, United States

Location

Green and Seidner Family Practice Associates

Lansdale, Pennsylvania, 19446, United States

Location

Temple University Hospital

Philadelphia, Pennsylvania, 19140, United States

Location

RI Hospital

Providence, Rhode Island, 02903, United States

Location

Neem Research Group, Inc.

Columbia, South Carolina, 29201, United States

Location

Internal Medicine & Industrial Medicine

DeSoto, Texas, 75115, United States

Location

T&R Clinical, P.A.

Fort Worth, Texas, 76117, United States

Location

Pri-Med Care

Lewisville, Texas, 75067, United States

Location

Texas Tech University Health Sciences Center

Lubbock, Texas, 79430, United States

Location

Diabetes Center of the Southwest

Midland, Texas, 79705, United States

Location

The Bracane Company

Plano, Texas, 75093, United States

Location

Innovative Clinical Trials

San Antonio, Texas, 78229, United States

Location

Burke Internal Medicine, Inc.

Burke, Virginia, 22015, United States

Location

Manassas Clinical Research Center

Manassas, Virginia, 20110, United States

Location

McGuire VA Medical Center

Richmond, Virginia, 22015, United States

Location

Peninsula Inernal Medicine

Gig Harbor, Washington, 98335, United States

Location

Liberty Research Center

Tacoma, Washington, 98405, United States

Location

CAMC Clinical Trials Center

Charleston, West Virginia, 25304, United States

Location

CIMEL

Buenos Aires, Argentina

Location

DIM (Clinica Privada)

Buenos Aires, Argentina

Location

Fundapres

Buenos Aires, Argentina

Location

Hospital Britanico de Buenos Aires

Buenos Aires, Argentina

Location

Hospital Jose Maria Ramos Meijia

Buenos Aires, Argentina

Location

Hospital Municipal bernardo Houssay

Buenos Aires, Argentina

Location

Medeos

Buenos Aires, Argentina

Location

Sanatorio Municipal Dr. Julio Mendez

Buenos Aires, Argentina

Location

Clinica Chutro SRL

Córdoba, Argentina

Location

Hospital San Roque

Córdoba, Argentina

Location

Hospital Governador Israel Pinheiro

Belo Horizonte, Brazil

Location

Hospital Socor

Belo Horizonte, Brazil

Location

Centro Medico de Campinas

Campinas, Brazil

Location

Hospital de Clinicas da Universidade Federal do Parana

Curitiba, Brazil

Location

Hospital das Clinicas

Goiânia, Brazil

Location

Clinica de Exames

Maceió, Brazil

Location

Instituto de Molestias

São José do Rio Preto, Brazil

Location

Centro Integrado Hospital do Rim e Hipertensao

São Paulo, Brazil

Location

Centro integrado hospital

São Paulo, Brazil

Location

Hospital das Clinicas da Faculdade de Medicina da USP

São Paulo, Brazil

Location

Cambridge Cardiac Care Center

Cambridge, Ontario, N3H 3R8, Canada

Location

Clinical Research Solutions

Kitchener, Ontario, N2G 1G5, Canada

Location

Bispebjerg Hospital

Copenhagen, Denmark

Location

Hvidovre Hospital

Hvidovre, Denmark

Location

CIC Hopital Jeanne D'Arc

Dommartin-lès-Toul, France

Location

CHU de Grenoble

Grenoble, France

Location

CHU la Timone Service de cardiologie

Marseille, France

Location

CHU Victor Provo

Roubaix, France

Location

Hôpital Civil, Service HTA maladies vasculaires

Strasbourg, France

Location

Kerckhoff-Klinik Forschungs GmbH

Bad Nauheim, Germany

Location

Charité Campus Buch

Berlin, Germany

Location

St Josefs-Hospital

Cloppenburg, Germany

Location

Medizinische Hochschule Hannover

Hanover, Germany

Location

Universitätsklinikum Schleswig-Holstein

Lübeck, Germany

Location

Azienda Ospedaliera University of Padua Policlinico

Padua, Italy

Location

Hospital Universitario de Santiago

A Coruña, Spain

Location

Fundacio Puigvert

Barcelona, Spain

Location

Hospital Clinic i Provincial

Barcelona, Spain

Location

Hospital del Mar

Barcelona, Spain

Location

Hospital Clínico San Cecilio

Granada, Spain

Location

Hospital Clínico de San Carlos

Madrid, Spain

Location

Hospital Universitario 12 de Octobre

Madrid, Spain

Location

Hospital Carlos Haya

Málaga, Spain

Location

Cardiovascular Research, Karolinska Institue

Stockholm, Sweden

Location

Stonehill Medical Centre

Bolton, United Kingdom

Location

Townhead Surgery

Scotland, United Kingdom

Location

Avenue Surgery

Wiltshire, United Kingdom

Location

Hathaway Medical Centre

Wiltshire, United Kingdom

Location

Related Publications (1)

  • Weber MA, Black H, Bakris G, Krum H, Linas S, Weiss R, Linseman JV, Wiens BL, Warren MS, Lindholm LH. A selective endothelin-receptor antagonist to reduce blood pressure in patients with treatment-resistant hypertension: a randomised, double-blind, placebo-controlled trial. Lancet. 2009 Oct 24;374(9699):1423-31. doi: 10.1016/S0140-6736(09)61500-2. Epub 2009 Sep 11.

Related Links

MeSH Terms

Conditions

Hypertension

Interventions

darusentan

Condition Hierarchy (Ancestors)

Vascular DiseasesCardiovascular Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 24, 2006

First Posted

May 26, 2006

Study Start

June 1, 2006

Primary Completion

January 1, 2009

Study Completion

January 1, 2009

Last Updated

March 18, 2014

Record last verified: 2014-02

Locations