NCT00266240

Brief Summary

This study will evaluate the efficacy, safety, tolerability, and pharmacokinetics of oral GK Activator (2), compared to placebo, in patients with type 2 diabetes mellitus. The anticipated time on study treatment is less than 3 months, and the target sample size is 100-500 individuals.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
267

participants targeted

Target at P75+ for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started Nov 2005

Typical duration for phase_2 diabetes-mellitus-type-2

Geographic Reach
7 countries

44 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 1, 2005

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

December 15, 2005

Completed
1 day until next milestone

First Posted

Study publicly available on registry

December 16, 2005

Completed
1.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2007

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2007

Completed
Last Updated

November 2, 2016

Status Verified

November 1, 2016

Enrollment Period

1.5 years

First QC Date

December 15, 2005

Last Update Submit

November 1, 2016

Conditions

Outcome Measures

Primary Outcomes (1)

  • HbA1c mean change from baseline, compared to placebo.

    Week 12

Secondary Outcomes (3)

  • Additional parameters of glycemic and lipid control.

    Week 12

  • AEs, laboratory parameters.

    Throughout study

  • Pharmacokinetic and exposure-response relationship

    Throughout study

Study Arms (5)

1

EXPERIMENTAL
Drug: GK Activator (2)

2

EXPERIMENTAL
Drug: GK Activator (2)

3

EXPERIMENTAL
Drug: GK Activator (2)

4

EXPERIMENTAL
Drug: GK Activator (2)

5

PLACEBO COMPARATOR
Drug: Placebo

Interventions

Escalating doses po bid

1234

po bid

5

Eligibility Criteria

Age30 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • adult patients 30-75 years of age;
  • type 2 diabetes mellitus for \>3 months before screening;
  • treatment-naive, inadequately controlled diabetes despite diet and exercise, or inadequately controlled diabetes in patients on monotherapy or combination therapy (maximum of 2 oral anti-hyperglycemic medications).

You may not qualify if:

  • type 1 diabetes mellitus;
  • women who are pregnant, breast-feeding or not using adequate contraceptive methods.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (44)

Unknown Facility

Tucson, Arizona, 85723, United States

Location

Unknown Facility

Pine Bluff, Arkansas, 71603, United States

Location

Unknown Facility

Chula Vista, California, 91911, United States

Location

Unknown Facility

Spring Valley, California, 91978, United States

Location

Unknown Facility

West Hills, California, 91307, United States

Location

Unknown Facility

Hollywood, Florida, 33021, United States

Location

Unknown Facility

Atlanta, Georgia, 30308, United States

Location

Unknown Facility

Binghamton, New York, 13901, United States

Location

Unknown Facility

Fayetteville, North Carolina, 28304, United States

Location

Unknown Facility

Statesville, North Carolina, 28625, United States

Location

Unknown Facility

Winston-Salem, North Carolina, 27103, United States

Location

Unknown Facility

Springdale, Ohio, 45246, United States

Location

Unknown Facility

Oklahoma City, Oklahoma, 73112, United States

Location

Unknown Facility

Medford, Oregon, 97504, United States

Location

Unknown Facility

Beaver, Pennsylvania, 15009, United States

Location

Unknown Facility

Tipton, Pennsylvania, 16684, United States

Location

Unknown Facility

Mt. Pleasant, South Carolina, 29464, United States

Location

Unknown Facility

Plano, Texas, 75093, United States

Location

Unknown Facility

Renton, Washington, 98055, United States

Location

Unknown Facility

Dimitrovgrad, 6400, Bulgaria

Location

Unknown Facility

Pleven, 5800, Bulgaria

Location

Unknown Facility

Rousse, 7002, Bulgaria

Location

Unknown Facility

Sofia, 1233, Bulgaria

Location

Unknown Facility

Sofia, 1303, Bulgaria

Location

Unknown Facility

Sofia, 1431, Bulgaria

Location

Unknown Facility

Sofia, 1606, Bulgaria

Location

Unknown Facility

Zagreb, 10000, Croatia

Location

Unknown Facility

Guatemala City, 01015, Guatemala

Location

Unknown Facility

Budapest, 1083, Hungary

Location

Unknown Facility

Budapest, 1088, Hungary

Location

Unknown Facility

Győr, 9024, Hungary

Location

Unknown Facility

Kecskemét, 6000, Hungary

Location

Unknown Facility

Chihuahua City, 31238, Mexico

Location

Unknown Facility

Cuernavaca, 62250, Mexico

Location

Unknown Facility

Durango, 34070, Mexico

Location

Unknown Facility

Mexico City, 06700, Mexico

Location

Unknown Facility

Mexico City, 11650, Mexico

Location

Unknown Facility

Mexico City, 14050, Mexico

Location

Unknown Facility

Mexico City, 14610, Mexico

Location

Unknown Facility

Bialystok, 15-276, Poland

Location

Unknown Facility

Gdansk, 80-757, Poland

Location

Unknown Facility

Gorzów, 66-400, Poland

Location

Unknown Facility

Krakow, 31-121, Poland

Location

Unknown Facility

Wroclaw, 50-088, Poland

Location

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Study Officials

  • Clinical Trials

    Hoffmann-La Roche

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 15, 2005

First Posted

December 16, 2005

Study Start

November 1, 2005

Primary Completion

May 1, 2007

Study Completion

May 1, 2007

Last Updated

November 2, 2016

Record last verified: 2016-11

Locations