NCT00105079

Brief Summary

This 2 arm study will evaluate the efficacy, safety and tolerability of saquinavir/ritonavir or lopinavir/ritonavir in combination with emtricitabine/tenofovir in patients with human immunodeficiency virus type 1 (HIV-1) infection who have received no prior HIV treatment. Patients will be randomized to receive either saquinavir/ritonavir 1000/100mg oral (po) twice daily (bid) + emtricitabine/tenofovir 200/300mg po once daily (qd), or lopinavir/ritonavir 400/100mg po bid + emtricitabine/tenofovir 200/300mg po qd. The anticipated time on study treatment is 3-12 months, and the target sample size is 100-500 individuals.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
337

participants targeted

Target at P25-P50 for phase_3 hiv-infections

Timeline
Completed

Started Apr 2005

Geographic Reach
5 countries

44 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 4, 2005

Completed
3 days until next milestone

First Posted

Study publicly available on registry

March 7, 2005

Completed
25 days until next milestone

Study Start

First participant enrolled

April 1, 2005

Completed
2.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2007

Completed
11 months until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2008

Completed
3.3 years until next milestone

Results Posted

Study results publicly available

November 2, 2011

Completed
Last Updated

November 2, 2011

Status Verified

September 1, 2011

Enrollment Period

2.3 years

First QC Date

March 4, 2005

Results QC Date

March 29, 2011

Last Update Submit

September 23, 2011

Conditions

Outcome Measures

Primary Outcomes (1)

  • Number of Patients With Human Immunodeficiency Virus Type 1 (HIV-1) Ribonucleic Acid (RNA) Viral Load <50 Copies/mL

    The primary objective of this study was to evaluate the efficacy of saquinavir/ritonavir BID plus emtricitabine/tenofovir QD versus lopinavir/ritonavir BID plus emtricitabine/tenofovir QD in treatment-naïve HIV-1 infected adults. Blood samples for HIV-1 RNA viral load measurement were collected at the Week 48 clinic visit. The number of participants with HIV-1 RNA results \<50 copies/mL is reported.

    Week 48

Secondary Outcomes (5)

  • Number of Patients With HIV-1 RNA Viral Load <50 and <400 Copies/mL

    Week 48

  • Change From Baseline in HIV-1 RNA Viral Load

    Baseline to Week 48

  • Change From Baseline in Cluster Differentiation Antigen 4 Positive (CD4+) Lymphocyte Count

    Baseline to Week 48

  • Number of Participants Assessed for Adverse Events (AEs)

    reported up to 28 days after the last dose of study treatment. (Up to 52 weeks)

  • Number of Patients Who Discontinued Treatment Due to Abnormal Laboratory Parameters

    baseline and all study visits (Up to Week 52)

Study Arms (2)

saquinavir/ritonavir

EXPERIMENTAL

saquinavir mesylate 1000 mg twice daily (BID) + ritonavir 100 mg BID + emtricitabine/tenofovir disoproxil fumarate 200/300 mg orally every day for 48 weeks.

Drug: saquinavir [Invirase]Drug: Emtricitabine/tenofovir disoproxil fumarateDrug: Ritonavir

lopinavir/ritonavir

ACTIVE COMPARATOR

lopinavir/ritonavir 400/100 mg BID + emtricitabine/tenofovir disoproxil fumarate 200/300 mg orally every day for 48 weeks.

Drug: Lopinavir/ritonavirDrug: Emtricitabine/tenofovir disoproxil fumarate

Interventions

1000 milligram (mg) Oral (po) twice daily (bid)

Also known as: Invirase
saquinavir/ritonavir

Lopinavir/ritonavir 400/100 mg po bid

Also known as: Kaletra
lopinavir/ritonavir

Emtricitabine/tenofovir disoproxil fumarate 200/300 mg po qd

Also known as: Truvada
lopinavir/ritonavirsaquinavir/ritonavir

100 mg po bid

Also known as: Norvir
saquinavir/ritonavir

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • adult patients \>=18 years of age;
  • chronic HIV-1 infection;
  • treatment-naive;
  • HIV-1 RNA viral load \>=10,000copies/mL;
  • women of childbearing potential must have a negative pregnancy test, and must use reliable contraception for the duration of the study and for 90 days after the last dose of study medication.

You may not qualify if:

  • females who are pregnant or breastfeeding;
  • active hepatitis B infection;
  • previous treatment with antiretroviral medication;
  • patients who have received an investigational drug within the last 4 weeks.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (44)

Unknown Facility

Hobson City, Alabama, 36201, United States

Location

Unknown Facility

Tucson, Arizona, 85745, United States

Location

Unknown Facility

Berkeley, California, 94705, United States

Location

Unknown Facility

Los Angeles, California, 90028, United States

Location

Unknown Facility

Washington D.C., District of Columbia, 20009, United States

Location

Unknown Facility

Jacksonville, Florida, 32204, United States

Location

Unknown Facility

Miami, Florida, 33136, United States

Location

Unknown Facility

Orlando, Florida, 32803, United States

Location

Unknown Facility

Vero Beach, Florida, 32960, United States

Location

Unknown Facility

Atlanta, Georgia, 30309, United States

Location

Unknown Facility

Macon, Georgia, 31201, United States

Location

Unknown Facility

Chicago, Illinois, 60613, United States

Location

Unknown Facility

Ypsilanti, Michigan, 48197, United States

Location

Unknown Facility

St Louis, Missouri, 63139, United States

Location

Unknown Facility

Newark, New Jersey, 07102, United States

Location

Unknown Facility

New York, New York, 10011, United States

Location

Unknown Facility

Huntersville, North Carolina, 28078, United States

Location

Unknown Facility

Philadelphia, Pennsylvania, 19107, United States

Location

Unknown Facility

Houston, Texas, 77004, United States

Location

Unknown Facility

Hamilton, Ontario, L8N 3Z5, Canada

Location

Unknown Facility

Ottawa, Ontario, K1H 8L6, Canada

Location

Unknown Facility

Toronto, Ontario, M4N 3M5, Canada

Location

Unknown Facility

Toronto, Ontario, M5B 1L6, Canada

Location

Unknown Facility

Toronto, Ontario, M5G 2C4, Canada

Location

Unknown Facility

Montreal, Quebec, H2L 4P9, Canada

Location

Unknown Facility

Montreal, Quebec, H2L 5B1, Canada

Location

Unknown Facility

Montreal, Quebec, H2X 2P4, Canada

Location

Unknown Facility

Avignon, 84902, France

Location

Unknown Facility

Lyon, 69288, France

Location

Unknown Facility

Lyon, 69437, France

Location

Unknown Facility

Marseille, 13009, France

Location

Unknown Facility

Marseille, 13385, France

Location

Unknown Facility

Nantes, 44035, France

Location

Unknown Facility

Nice, 06202, France

Location

Unknown Facility

Paris, 75010, France

Location

Unknown Facility

Paris, 75014, France

Location

Unknown Facility

Paris, 75651, France

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Unknown Facility

Rouen, 73031, France

Location

Unknown Facility

Strasbourg, 67091, France

Location

Unknown Facility

Suresnes, 92150, France

Location

Unknown Facility

Toulouse, 31052, France

Location

Unknown Facility

Tourcoing, 59208, France

Location

Unknown Facility

Ponce, 00717-1563, Puerto Rico

Location

Unknown Facility

Bangkok, 10330, Thailand

Location

MeSH Terms

Conditions

HIV Infections

Interventions

SaquinavirLopinavirlopinavir-ritonavir drug combinationEmtricitabine, Tenofovir Disoproxil Fumarate Drug CombinationRitonavir

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsVirus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

IsoquinolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic CompoundsQuinolinesPyrimidinonesPyrimidinesHeterocyclic Compounds, 1-RingTenofovirOrganophosphonatesOrganophosphorus CompoundsOrganic ChemicalsEmtricitabineDeoxycytidineCytidinePyrimidine NucleosidesAdeninePurinesDeoxyribonucleosidesNucleosidesNucleic Acids, Nucleotides, and NucleosidesDrug CombinationsPharmaceutical PreparationsThiazolesSulfur CompoundsAzoles

Results Point of Contact

Title
Medical Communications
Organization
Hoffman-LaRoche

Study Officials

  • Clinical Trials

    Hoffmann-La Roche

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 4, 2005

First Posted

March 7, 2005

Study Start

April 1, 2005

Primary Completion

August 1, 2007

Study Completion

July 1, 2008

Last Updated

November 2, 2011

Results First Posted

November 2, 2011

Record last verified: 2011-09

Locations