NCT06045221

Brief Summary

The main purpose of this study is to assess efficacy and safety of orforglipron compared with oral semaglutide in participants with Type 2 diabetes and inadequate glycemic control with metformin.The study will last around 61 weeks.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
1,698

participants targeted

Target at P75+ for phase_3 type-2-diabetes

Timeline
Completed

Started Sep 2023

Typical duration for phase_3 type-2-diabetes

Geographic Reach
6 countries

131 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 13, 2023

Completed
8 days until next milestone

First Posted

Study publicly available on registry

September 21, 2023

Completed
1 day until next milestone

Study Start

First participant enrolled

September 22, 2023

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 22, 2025

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 22, 2025

Completed
Last Updated

September 22, 2025

Status Verified

September 1, 2025

Enrollment Period

1.9 years

First QC Date

September 13, 2023

Last Update Submit

September 19, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change from Baseline in Hemoglobin A1c (HbA1c)

    Baseline, Week 52

Secondary Outcomes (20)

  • Change from Baseline in HbA1c

    Baseline, Week 52

  • Percentage of Participants Who Achieved HbA1c <7.0% 53 millimole/mole (mmol/mol)

    Week 52

  • Percentage of Participants Who Achieved HbA1c ≤6.5% (48 mmol/mol)

    Week 52

  • Percentage Change from Baseline in Body Weight

    Baseline, Week 52

  • Change from Baseline in Body Weight

    Baseline, Week 52

  • +15 more secondary outcomes

Study Arms (4)

Orforglipron Dose 1

EXPERIMENTAL

Participants will receive orforglipron orally.

Drug: Orforglipron

Orforglipron Dose 2

EXPERIMENTAL

Participants will receive orforglipron orally.

Drug: Orforglipron

Semaglutide Dose 1

ACTIVE COMPARATOR

Participants will receive semaglutide orally.

Drug: Semaglutide

Semaglutide Dose 2

ACTIVE COMPARATOR

Participants will receive semaglutide orally.

Drug: Semaglutide

Interventions

Administered orally

Also known as: LY3502970
Orforglipron Dose 1Orforglipron Dose 2

Administered orally

Semaglutide Dose 1Semaglutide Dose 2

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have Type 2 Diabetes
  • Have HbA1c ≥7.0% (53 mmol/mol) to ≤10.5% (91 mmol/mol), as determined by the central laboratory at screening.
  • Have been on stable diabetes treatment with metformin ≥1500 milligram (mg)/day during the 90 days prior to screening and maintained through randomization.
  • Are of stable body weight (±5%) for at least 90 days prior to screening and agree to not initiate an intensive diet or exercise program during the study with the intent of reducing body weight, other than the lifestyle and/or dietary measures for diabetes treatment

You may not qualify if:

  • Have Type 1 Diabetes
  • Are currently receiving or planning to receive treatment for diabetic retinopathy and/or macular edema, for example, laser photocoagulation or intravitreal injections of anti-vascular endothelial growth factor inhibitors.
  • Have a history of ketoacidosis or hyperosmolar state or coma within the last 6 months prior to screening, or between screening and randomization.
  • Have a New York Heart Association functional classification IV congestive heart failure.
  • Have an estimated glomerular filtration rate (eGFR) \<45 milliliter/minute (mL/min)/1.73 square meter (m²) or lower than the country-specific threshold for discontinuing metformin therapy per local label as determined by the central laboratory at screening.
  • Have a serum calcitonin level of ≥35 nanogram/Liter (ng/L), as determined by the central laboratory at screening.
  • Have a history of an active or untreated malignancy or are in remission from a clinically significant malignancy for less than 5 years.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (131)

Absolute Clinical Research

Phoenix, Arizona, 85051, United States

Location

San Fernando Valley Health Institute

Canoga Park, California, 91304, United States

Location

Neighborhood Healthcare Institute of Health

Escondido, California, 92025, United States

Location

Velocity Clinical Research, Gardena

Gardena, California, 90247, United States

Location

Biopharma Informatic, LLC

Los Angeles, California, 90035, United States

Location

Velocity Clinical Research, Westlake

Los Angeles, California, 90057, United States

Location

Infinity Clinical Research - Norco

Norco, California, 92860, United States

Location

Valley Clinical Trials, Inc.

Northridge, California, 91325, United States

Location

Norcal Endocrinology & Internal Medicine

San Ramon, California, 94583, United States

Location

Encompass Clinical Research

Spring Valley, California, 91978, United States

Location

University Clinical Investigators, Inc.

Tustin, California, 92780, United States

Location

New West Physicians Clinical Research

Golden, Colorado, 80401, United States

Location

Connecticut Clinical Research - Cromwell

Cromwell, Connecticut, 06416, United States

Location

Clinical Research of West Florida, Inc. (Clearwater)

Clearwater, Florida, 33765, United States

Location

South Florida Clinical Research Institute

Margate, Florida, 33063, United States

Location

Miami Dade Medical Research Institute, LLC

Miami, Florida, 33176, United States

Location

West Orange Endocrinology

Ocoee, Florida, 34761, United States

Location

Latin Clinical Trial Center Florida

Tamarac, Florida, 33321, United States

Location

Clinical Research of West Florida

Tampa, Florida, 33606, United States

Location

Metabolic Research Institute, Inc.

West Palm Beach, Florida, 33401, United States

Location

Balanced Life Health Care Solutions/SKYCRNG

Lawrenceville, Georgia, 30046, United States

Location

Clinical Research Atlanta

Stockbridge, Georgia, 30281, United States

Location

North Georgia Clinical Research

Woodstock, Georgia, 30189, United States

Location

Northwest Clinical Trials

Boise, Idaho, 83704, United States

Location

Family First Medical Center

Idaho Falls, Idaho, 83404, United States

Location

American Health Network of Indiana, LLC - Greenfield

Greenfield, Indiana, 46140, United States

Location

Velocity Clinical Research, Valparaiso

Valparaiso, Indiana, 46383, United States

Location

Cotton O'Neil Diabetes & Endocrinology

Topeka, Kansas, 66606, United States

Location

Tekton Research, Inc

Wichita, Kansas, 67218, United States

Location

DelRicht Research

New Orleans, Louisiana, 70115, United States

Location

Joslin Diabetes Center

Boston, Massachusetts, 02215, United States

Location

Revival Research Institute, LLC

Dearborn, Michigan, 48126, United States

Location

SKY Integrative Medical Center/SKYCRNG

Ridgeland, Mississippi, 39157, United States

Location

Kansas City Research Institute

Kansas City, Missouri, 64131, United States

Location

Logan Health Research

Kalispell, Montana, 59901, United States

Location

Wr-Crcn, Llc

Las Vegas, Nevada, 89106, United States

Location

Premier Research

Trenton, New Jersey, 08611, United States

Location

Albany Medical College, Division of Community Endocrinology

Albany, New York, 12203, United States

Location

Ellipsis Research Group - Brooklyn - 7th Street

Brooklyn, New York, 11215, United States

Location

Great Lakes Medical Research, LLC

Westfield, New York, 14787, United States

Location

PharmQuest Life Sciences, LLC

Greensboro, North Carolina, 27408, United States

Location

Lucas Research, Inc

Morehead City, North Carolina, 28557, United States

Location

Accellacare - Piedmont

Statesville, North Carolina, 28625, United States

Location

Wake Forest University Baptist Medical Center (WFUBMC)

Winston-Salem, North Carolina, 27104, United States

Location

Aventiv Research Inc

Columbus, Ohio, 43213, United States

Location

Tekton Research, Inc

Moore, Oklahoma, 73160, United States

Location

Alliance for Multispecialty Research, LLC

Norman, Oklahoma, 73069, United States

Location

The Corvallis Clinic, P.C.

Corvallis, Oregon, 97330, United States

Location

Heritage Valley Medical Group, Inc.

Beaver, Pennsylvania, 15009, United States

Location

Preferred Primary Care Physicians, Preferred Clinical Research (Ofc 18)

Pittsburgh, Pennsylvania, 15236, United States

Location

The Research Center of The Upstate

Greenville, South Carolina, 29607, United States

Location

New Phase Research and Development

Knoxville, Tennessee, 37909, United States

Location

Clinical Neuroscience Solutions Inc.

Memphis, Tennessee, 38119, United States

Location

Velocity Clinical Research, Austin

Austin, Texas, 78759, United States

Location

Velocity Clinical Research, Dallas

Dallas, Texas, 75230, United States

Location

Diabetes and Thyroid Center of Ft. Worth

Fort Worth, Texas, 76132, United States

Location

Juno Research

Houston, Texas, 77040, United States

Location

Endocrine Ips, Pllc

Houston, Texas, 77079, United States

Location

Clear Brook Medical Associates

Houston, Texas, 77089, United States

Location

Southern Endocrinology Associates

Mesquite, Texas, 75149, United States

Location

Texas Valley Clinical Research

Weslaco, Texas, 78596, United States

Location

Synexus Clinical Research US, Inc.

Salt Lake City, Utah, 84106, United States

Location

Eastside Research Associates

Redmond, Washington, 98052, United States

Location

Rainier Clinical Research Center

Renton, Washington, 98057, United States

Location

Centro de Investigaciones Metabólicas (CINME)

Ciudad Autónoma de Buenos Aires, Buenos Aires, 1056, Argentina

Location

CIMeL

Lanús, Buenos Aires, B1824KAJ, Argentina

Location

Centro de Investigaciones Médicas Mar del Plata

Mar del Plata, Buenos Aires, 7600, Argentina

Location

Policlinica Red OMIP

Mar del Plata, Buenos Aires, 7600, Argentina

Location

Consultorio de Investigación Clínica EMO SRL

Buenos Aires, Buenos Aires F.D., 1405, Argentina

Location

CIPREC

Buenos Aires, Buenos Aires F.D., C1061AAS, Argentina

Location

Centro Médico Viamonte

Buenos Aires, Buenos Aires F.D., C1120AAC, Argentina

Location

Instituto Centenario

CABA, Buenos Aires F.D., 1204, Argentina

Location

Centro de Salud e Investigaciones Médicas

Santa Rosa, La Pampa Province, 6300, Argentina

Location

INECO Neurociencias Oroño

Rosario, Santa Fe Province, 2000, Argentina

Location

Instituto de Especialidades de la Salud Rosario

Rosario, Santa Fe Province, 2000, Argentina

Location

Instituto Médico Catamarca IMEC

Rosario, Santa Fe Province, 2000, Argentina

Location

Instituto Médico Fundación Grupo Colaborativo Rosario Investigación y Prevención Medica

Rosario, Santa Fe Province, 2000, Argentina

Location

Fundacion Estudios Clinicos

Rosario, Santa Fe Province, S2000DEJ, Argentina

Location

Instituto de Investigaciones Clínicas Córdoba

Córdoba, 5000, Argentina

Location

Instituto Médico DAMIC

Córdoba, 5003DCE, Argentina

Location

Sanatorio Norte

Santiago del Estero, 4200, Argentina

Location

Beijing Pinggu District Hospital

Beijing, Beijing Municipality, 101200, China

Location

Chongqing General Hospital

Chongqing, Chongqing Municipality, 400014, China

Location

Shunde Hospital of Southern Medical Univesity

Foshan, Guangdong, 528399, China

Location

Huizhou Municipal Central Hospital

Huizhou, Guangdong, 516001, China

Location

The Fourth Hospital of Harbin Medical University

Harbin, Heilongjiang, 150001, China

Location

The First Affiliated Hospital of Henan University of Science &Technology

Luoyang Shi, Henan, 471003, China

Location

Nanyang First People's Hospital

Nanyang, Henan, 473014, China

Location

The Second Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, 450014, China

Location

Nanjing First Hospital

Nanjing, Jiangsu, 210006, China

Location

The Second Affiliated Hospital of Nanjing Medical University

Nanjing, Jiangsu, 210011, China

Location

Affiliated Hospital of Jiangsu University

Zhenjiang, Jiangsu, 212000, China

Location

Jiangxi Pingxiang People's Hospital

Pingxiang, Jiangxi, 337055, China

Location

Dalian Municipal Central Hospital Affiliated of Dalian Medical University

Dalian, Liaoning, 116033, China

Location

Jinan Central Hospital

Jinan, Shandong, 250013, China

Location

Shanghai Sixth People's Hospital

Shanghai, Shanghai Municipality, 200030, China

Location

Pudong New Area People's Hospital Shanghai

Shanghai, Shanghai Municipality, 201200, China

Location

West China Hospital of Sichuan University

Chengdu, Sichuan, 610041, China

Location

First Affiliated Hospital of Kunming Medical University

Kunming, Yunnan, 650032, China

Location

Zhejiang Hospital

Hangzhou, Zhejiang, 310013, China

Location

Huzhou Central Hospital

Huzhou, Zhejiang, 313000, China

Location

The First Affiliated Hospital of Wenzhou Medical University

Wenzhou, Zhejiang, 325000, China

Location

Mikannohana Clinic, Diabetes, Endocrinology and Metabolism

Matsuyama, Ehime, 116099, Japan

Location

Manda Memorial Hospital

Sapporo, Hokkaido, 060-0062, Japan

Location

Nakamoto Internal Medicine Clinic

Mito, Ibaraki, 310-0826, Japan

Location

Nakakinen clinic

Naka, Ibaraki, 311-0113, Japan

Location

Ohishi Internal Medicine Clinic

Tsuchiura, Ibaraki, 300-0835, Japan

Location

Takai Internal Medicine Clinic

Kamakura-shi, Kanagawa, 247-0056, Japan

Location

Shiraiwa Medical Clinic

Kashihara, Osaka, 582-0005, Japan

Location

Medical Corporation Sato Medical clinic

Ootaku, Tokyo, 143-0015, Japan

Location

Gifu University Hospital

Gifu, 501-1112, Japan

Location

Centro de Investigacion Medica Integral

Guadalajara, Jalisco, 44160, Mexico

Location

Instituto Jalisciense de Investigacion en Diabetes y Obesidad

Guadalajara, Jalisco, 44600, Mexico

Location

CICEJ Centro de Investigación Clínica Endocrinológica de Jalisco S.C

Guadalajara, Jalisco, 44670, Mexico

Location

Private Practice - Dr. Arechavaleta Granell Maria del Rosario

Guadalajara, Jalisco, 44670, Mexico

Location

Virgen Cardiovascular Research SC

Guadalajara, Jalisco, 44670, Mexico

Location

Centro de Investigacion Medica de Occidente, S.C.

Zapopan, Jalisco, 44260, Mexico

Location

Caimed Investigacion En Salud S.A. de C.V.

Mexico City, Mexico City, 06760, Mexico

Location

Centro Especializado En Diabetes, Obesidad Y Prevencion De Enfermedades Cardiovasculares

Mexico City, Mexico City, 11650, Mexico

Location

Cardiolink Clin Trials

Monterrey, Nuevo León, 64060, Mexico

Location

Unidad biomedica avanzada monterrey

Monterrey, Nuevo León, 64460, Mexico

Location

Clínica García Flores SC

Monterrey, Nuevo León, 64610, Mexico

Location

Eukarya PharmaSite

Monterrey, Nuevo León, 64718, Mexico

Location

Hospital Universitario "Dr. Jose Eleuterio Gonzalez"

Monterrey, Nuevo León, 66460, Mexico

Location

Centro de investigación y control metabólico

San Nicolás de los Garza, Nuevo León, 66465, Mexico

Location

Centro Para El Desarrollo de La Medicina Y de Asistencia Medica Especializada S.C.

Culiacán, Sinaloa, 80230, Mexico

Location

Lahoja. Asociacion Para La Investigacion Y La Farmacovigilancia

Durango, 34000, Mexico

Location

Isis Clinical Research Center

Guaynabo, PR, 00968, Puerto Rico

Location

Mgcendo Llc

San Juan, PR, 00921, Puerto Rico

Location

Research and Cardiovascular Corp.

Ponce, 00717, Puerto Rico

Location

Latin Clinical Trial Center

San Juan, 00909, Puerto Rico

Location

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

orforglipronsemaglutide

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Study Officials

  • Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

    Eli Lilly and Company

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 13, 2023

First Posted

September 21, 2023

Study Start

September 22, 2023

Primary Completion

August 22, 2025

Study Completion

August 22, 2025

Last Updated

September 22, 2025

Record last verified: 2025-09

Data Sharing

IPD Sharing
Will share

Anonymized individual patient level data will be provided in a secure access environment upon approval of a research proposal and a signed data sharing agreement.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
Data are available 6 months after the primary publication and approval of the indication studied in the US and European Union (EU), whichever is later. Data will be indefinitely available for requesting.
Access Criteria
A research proposal must be approved by an independent review panel and researchers must sign a data sharing agreement.
More information

Locations