NCT05892393

Brief Summary

This phase I trial tests the safety of \[89Zr\]DFO-YS5 positron emission tomography (PET) imaging and how well it works to detect CD46 positive cancer cells in patients with multiple myeloma. \[89Zr\]DFO-YS5 is an imaging agent called a radiopharmaceutical tracer. A radiopharmaceutical tracer uses a small amount of radioactive material that is injected into a vein to help image different areas of the body. \[89Zr\]DFO-YS5 targets a specialized protein called CD46, which is in certain multiple myeloma cancer cells, and \[89Zr\]DFO-YS5 PET scans may improve detection of multiple myeloma.

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
20

participants targeted

Target at P25-P50 for phase_1 multiple-myeloma

Timeline
4mo left

Started Jun 2023

Geographic Reach
1 country

1 active site

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress90%
Jun 2023Sep 2026

First Submitted

Initial submission to the registry

May 26, 2023

Completed
12 days until next milestone

First Posted

Study publicly available on registry

June 7, 2023

Completed
9 days until next milestone

Study Start

First participant enrolled

June 16, 2023

Completed
3.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2026

Expected
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2026

Last Updated

November 12, 2025

Status Verified

August 1, 2025

Enrollment Period

3.1 years

First QC Date

May 26, 2023

Last Update Submit

November 7, 2025

Conditions

Outcome Measures

Primary Outcomes (3)

  • Sensitivity of metastatic lesion

    Defined as the rate of lesions with positive uptake when compared against 18F-fluorodeoxyglucose (FDG) PET/computed tomography (CT) positivity. Sensitivity estimated based on lesion level without considering the location of the lesions or the possible intracorrelation of the lesions from the same patient by point estimate with its 95% confidence interval.

    Up to 1 week

  • Median maximum standardized uptake value (SUVmax)

    The median and range of standardized uptake value maximum (SUVmax) (across all metastatic lesions per participant) in each study cohort will be descriptively reported using mediastinal blood pool and normal organ background uptake values.

    Up to 1 week

  • Median Standardized Uptake Value averaged across lesions (SUVmax-avg)

    The median and range of SUVmax-average across all lesions in each study cohort will be descriptively reported using mediastinal blood pool and normal organ background uptake values.

    Up to 1 week

Secondary Outcomes (4)

  • Proportion of participants reporting treatment-related Adverse Events

    Up to 35 days

  • Average organ uptake of [89Zr]DFO-YS5

    Up to 1 week

  • Descriptive patterns of intra-tumoral uptake of [89Zr]DFO-YS5

    Up to 1 week

  • Dosimetry measurements (Cohort B only)

    Up to 1 week

Study Arms (2)

Cohort A ([89Zr]DFO-YS5, single scan

EXPERIMENTAL

Participants receive \[89Zr\]DFO-YS5 IV and undergo a single PET/CT or PET/MRI scan 5-7 days post-injection. Participants also receive fludeoxyglucose F-18 IV and undergo PET/CT or PET/MRI scan within 28 days prior to day 1

Drug: Zirconium Zr 89-DFO-YS5Procedure: Positron Emission Tomography / Computed Tomography (PET/CT)Procedure: Positron Emission Tomography / Magnetic Resonance Imaging (PET/MRI)Other: Fludeoxyglucose F-18

Cohort B ([89Zr]DFO-YS5, multiple scans

EXPERIMENTAL

Participants receive \[89Zr\]DFO-YS5 IV and undergo four PET/CT or PET/MRI scans on days 1, 2, 3-4, and 5-7 post-injection. Participants also receive fludeoxyglucose F-18 IV and undergo PET/CT or PET/MRI scan within 28 days prior to day 1

Drug: Zirconium Zr 89-DFO-YS5Procedure: Positron Emission Tomography / Computed Tomography (PET/CT)Procedure: Positron Emission Tomography / Magnetic Resonance Imaging (PET/MRI)Other: Fludeoxyglucose F-18

Interventions

Given IV

Also known as: (89)Zr-DFO-YS5, 89Zr DFO-YS5
Cohort A ([89Zr]DFO-YS5, single scanCohort B ([89Zr]DFO-YS5, multiple scans

Positron emission tomography-computed tomography is a nuclear medicine technique which combines, in a single gantry, a positron emission tomography scanner and an x-ray computed tomography scanner, to acquire sequential images from both devices in the same session, which are combined into a single superposed image

Also known as: PET/CT
Cohort A ([89Zr]DFO-YS5, single scanCohort B ([89Zr]DFO-YS5, multiple scans

Positron emission tomography-magnetic resonance imaging is a hybrid imaging technology that incorporates magnetic resonance imaging soft tissue morphological imaging and positron emission tomography functional imaging.

Also known as: PET/MRI
Cohort A ([89Zr]DFO-YS5, single scanCohort B ([89Zr]DFO-YS5, multiple scans

Given IV

Also known as: Fludeoxyglucose (18F)
Cohort A ([89Zr]DFO-YS5, single scanCohort B ([89Zr]DFO-YS5, multiple scans

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants must have histologically or cytologically confirmed multiple myeloma by International Myeloma Working Group (IMWG) diagnostic criteria
  • At least one positive myelomatous lesion found on 18F-FDG PET/CT or PET/MRI. A positive lesion is defined as uptake greater than liver on FDG PET, based on the Italian myeloma criteria for PET use (IMPeTUs) criteria
  • Age \>= 18 years
  • Total bilirubin =\< 1.5 X institutional upper limit of normal (ULN)
  • Aspartate aminotransferase (AST) =\< 3 X ULN
  • Alanine aminotransferase (ALT) =\< 3 X ULN
  • Creatinine clearance \>= 60 mL/min, calculated using the Cockcroft-Gault equation or serum creatinine \<= 1.5x the institutional upper limit of normal.
  • Ability to understand a written informed consent document, and the willingness to sign it

You may not qualify if:

  • Any condition that, in the opinion of the principal investigator, would impair the participants' ability to comply with study procedures or interfere with the safety of the investigational regimen
  • Individuals who are pregnant or breastfeeding/chestfeeding.
  • \- Breast-feeding/chest-feeding should be discontinued before administration of \[89ZR\]DFO-YS5.
  • Females of childbearing potential must have a negative urine or serum pregnancy test (i.e., human chorionic gonadotropin test) within 72 hours prior to administration of \[89ZR\]-DFO-YS5.
  • \- If the urine pregnancy test is positive or equivocal, a confirmatory serum pregnancy test is required. In such cases, the individual must be excluded from participation if the serum pregnancy result is positive.
  • \- A female is considered to be of childbearing potential (regardless of sexual orientation, having undergone a tubal ligation, or remaining celibate by choice), unless it is documented that the individual meets either of the following two criteria: (1) has reached a postmenopausal state ( \>= 12 continuous months of amenorrhea with no identified cause other than menopause); or (2) has undergone surgical sterilization (i.e., hysterectomy and/or bilateral oophorectomy for removal of uterus and/or ovaries).
  • Individuals who are pregnant or breastfeeding/chestfeeding are excluded because there is an unknown but potential risk for adverse effects in the unborn/nursing child secondary to treatment of the study participant with \[89ZR\]-DFO-YS5

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

University of California, San Francisco

San Francisco, California, 94143, United States

RECRUITING

MeSH Terms

Conditions

Multiple Myeloma

Interventions

Magnetic Resonance SpectroscopyFluorodeoxyglucose F18

Condition Hierarchy (Ancestors)

Neoplasms, Plasma CellNeoplasms by Histologic TypeNeoplasmsHemostatic DisordersVascular DiseasesCardiovascular DiseasesParaproteinemiasBlood Protein DisordersHematologic DiseasesHemic and Lymphatic DiseasesHemorrhagic DisordersLymphoproliferative DisordersImmunoproliferative DisordersImmune System Diseases

Intervention Hierarchy (Ancestors)

Spectrum AnalysisChemistry Techniques, AnalyticalInvestigative TechniquesDeoxyglucoseDeoxy SugarsCarbohydrates

Study Officials

  • Robert Flavell, MD, PhD

    University of California, San Francisco

    PRINCIPAL INVESTIGATOR

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
DIAGNOSTIC
Intervention Model
SINGLE GROUP
Sponsor Type
OTHER
Responsible Party
SPONSOR INVESTIGATOR
PI Title
Principal Investigator

Study Record Dates

First Submitted

May 26, 2023

First Posted

June 7, 2023

Study Start

June 16, 2023

Primary Completion (Estimated)

August 1, 2026

Study Completion (Estimated)

September 1, 2026

Last Updated

November 12, 2025

Record last verified: 2025-08

Data Sharing

IPD Sharing
Will not share

Locations