NCT05587309

Brief Summary

The objective of the Healing Phase of the study is to evaluate the safety and efficacy of up to 8 weeks of once daily oral administration of BLI5100 versus a PPI control in healing EE. The objective of the Maintenance Phase of the study is to evaluate the safety and efficacy of 24 weeks of once daily oral administration of BLI5100 (low or high dose) versus a PPI control in the maintenance of healed EE.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
1,250

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Oct 2022

Typical duration for phase_3

Geographic Reach
1 country

122 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 17, 2022

Completed
3 days until next milestone

First Posted

Study publicly available on registry

October 20, 2022

Completed
10 days until next milestone

Study Start

First participant enrolled

October 30, 2022

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 16, 2025

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 16, 2025

Completed
Last Updated

September 24, 2025

Status Verified

September 1, 2025

Enrollment Period

2.6 years

First QC Date

October 17, 2022

Last Update Submit

September 19, 2025

Conditions

Outcome Measures

Primary Outcomes (2)

  • Healing Phase: Percentage of patients with complete healing by Week 8.

    8 Weeks

  • Maintenance Phase: Percentage of patients who maintain complete healing through Week 24.

    24 Weeks

Secondary Outcomes (2)

  • Healing Phase: Percentage of 24-hour heartburn-free days through Week 8.

    8 Weeks

  • Maintenance Phase: Percentage of 24-hour heartburn-free days through Week 24.

    24 Weeks

Study Arms (5)

Healing Phase - BLI5100

EXPERIMENTAL

During the Healing Phase, patients will take BLI5100 once daily, orally, for up to 8 weeks.

Drug: BLI5100

Healing Phase - PPI Control

ACTIVE COMPARATOR

During the Healing Phase, patients will take a PPI control once daily, orally, for up to 8 weeks.

Drug: PPI Control

Maintenance Phase - BLI5100 Low Dose

EXPERIMENTAL

During the Maintenance Phase, patients will take BLI5100 low dose once daily, orally, for 24 weeks.

Drug: BLI5100

Maintenance Phase - BLI5100 High Dose

EXPERIMENTAL

During the Maintenance Phase, patients will take BLI5100 high dose once daily, orally, for 24 weeks.

Drug: BLI5100

Maintenance Phase - PPI Control

ACTIVE COMPARATOR

During the Maintenance Phase, patients will take a PPI control once daily, orally, for 24 weeks.

Drug: PPI Control

Interventions

Orally via tablet

Healing Phase - BLI5100Maintenance Phase - BLI5100 High DoseMaintenance Phase - BLI5100 Low Dose

Orally via tablet

Healing Phase - PPI ControlMaintenance Phase - PPI Control

Eligibility Criteria

Age18 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Aged ≥18 years at the time of signing informed consent;
  • Have experienced both heartburn and regurgitation within 7 days prior to the Screening Visit;
  • Current evidence of EE of LA grades A to D based on an upper GI endoscopy;
  • Able to understand and comply with the protocol requirements;
  • Willing and able to provide written informed consent at Screening;
  • A female of reproductive potential defined as a non-post-menopausal female who has not had a bilateral oophorectomy or medically documented ovarian failure; or If a female of childbearing potential, agrees to use an acceptable form of birth control and avoid egg donation from the Screening Visit until 6 months after the last dose of study drug.
  • If a male, agrees to use an acceptable form of birth control from the Screening Visit until 3 months after the last dose of study drug.
  • If a male, agrees to abstain from sperm donation through 3 months after administration of the last dose of study drug.

You may not qualify if:

  • Unable to undergo an upper GI endoscopy;
  • Presence of esophageal stricture, gastroesophageal varix (including post sclerotherapy or ligation), untreated Barrett's esophagus, gastric bleeding, infection, tumor, or gastric or duodenal ulcer on the upper GI endoscopy;
  • o Note: Patients with diagnosis of Schatzki's ring (mucosal tissue ring around lower esophageal sphincter) are eligible to participate.
  • Alarm symptoms such as odynophagia, severe dysphagia, upper GI bleeding, weight loss, anemia, or hematochezia within 4 weeks prior to Screening, unless the presumed malignancy is ruled out;
  • History of eosinophilic esophagitis, achalasia, or other primary esophageal motility disorder; functional heartburn; physiochemical trauma (including radiation, mucosal resection, or cryotherapy); or documented history of delayed gastric emptying;
  • History of a connective tissue disorder associated with GI symptoms (eg, scleroderma or systemic lupus erythematous) or inflammatory bowel disease;
  • History of acid-suppressive, esophageal, or gastric surgery;
  • o Note: This is not applicable to appendectomy, cholecystectomy, or endoscopic excision of benign tumor.
  • History of malignancy within the past 5 years (with the exception of resected basal cell or squamous cell carcinoma of the skin);
  • o Note: This is not applicable to patients who had complete response or pathological complete response and whose tumor had not recurred for at least 5 years from the date of last treatment, or patients whose tumor had been removed by endoscopic resection without any findings indicating recurrence of the tumor within 3 years.
  • History of an allergic disease, or hypersensitivity or intolerance to the active ingredient or excipients of the study drug;
  • History of alcoholism, chronic opiate use, or substance addiction in the 12 months before Screening or a positive urine drug screen for opiates or substances of abuse;
  • Note: Patients on prescribed opioids are eligible to participate if they have been on a stable dose for \>3 months prior to Screening.
  • Note: Retesting of a positive urine drug screen requires Medical Monitor approval. Positive urine drug screen for all drugs will require verification of prescription for the positive tested substance.
  • Presence of manic-depression, anxiety disorder, panic disorder, somatoform disorder, personality disorder, or other psychological disorder;
  • +18 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (122)

Research Site 145

Homewood, Alabama, 35209, United States

Location

Research Site 24

Huntsville, Alabama, 35801, United States

Location

Research Site 132

Peoria, Arizona, 85381, United States

Location

Research Site 150

Peoria, Arizona, 85381, United States

Location

Research Site 62

Phoenix, Arizona, 85018, United States

Location

Research Site 27

Tucson, Arizona, 85712, United States

Location

Research Site 87

Little Rock, Arkansas, 72211, United States

Location

Research Site 117

North Little Rock, Arkansas, 72117, United States

Location

Research Site 51

Arcadia, California, 91006, United States

Location

Research Site 66

Bell Gardens, California, 90201, United States

Location

Research Site 156

Camarillo, California, 93012, United States

Location

Research Site 19

Canoga Park, California, 91304, United States

Location

Research Site 94

Chula Vista, California, 91910, United States

Location

Research Site 10

Huntington Park, California, 90255, United States

Location

Research Site 55

La Mesa, California, 91942, United States

Location

Research Site 72

Los Angeles, California, 90017, United States

Location

Research Site 14

San Diego, California, 92120, United States

Location

Research Site 85

Santa Ana, California, 92703, United States

Location

Research Site 13

Santa Ana, California, 92704, United States

Location

Research Site 41

Santa Maria, California, 93458, United States

Location

Research Site 54

Westlake, California, 90057, United States

Location

Research Site 89

Littleton, Colorado, 80120, United States

Location

Research Site 147

Bristol, Connecticut, 06010, United States

Location

Research Site 74

Boca Raton, Florida, 33434, United States

Location

Research Site 108

Cooper City, Florida, 33024, United States

Location

Research Site 91

Doral, Florida, 33172, United States

Location

Research Site 03

Hialeah, Florida, 33013, United States

Location

Research Site 78

Homestead, Florida, 33030, United States

Location

Research Site 09

Lake City, Florida, 32055, United States

Location

Research Site 23

Maitland, Florida, 32751, United States

Location

Research Site 38

Miami, Florida, 33134, United States

Location

Research Site 43

Miami, Florida, 33136, United States

Location

Research Site 67

Miami, Florida, 33155, United States

Location

Research Site 92

Miami, Florida, 33173, United States

Location

Research Site 31

Miami, Florida, 33185, United States

Location

Research Site 71

Miami, Florida, 33186, United States

Location

Research Site 42

Miami Lakes, Florida, 33014, United States

Location

Research Site 17

New Port Richey, Florida, 34653, United States

Location

Research Site 90

Ocoee, Florida, 34761, United States

Location

Research Site 107

Orlando, Florida, 32087, United States

Location

Research Site 05

Palmetto Bay, Florida, 33157, United States

Location

Research Site 95

St. Petersburg, Florida, 33709, United States

Location

Research Site 11

Sunrise, Florida, 33351, United States

Location

Research Site 46

Viera, Florida, 32940, United States

Location

Research Site 153

Atlanta, Georgia, 30329, United States

Location

Research Site 04

Marietta, Georgia, 30060, United States

Location

Research Site 59

Sandy Springs, Georgia, 30328, United States

Location

Research Site 151

Boise, Idaho, 83706, United States

Location

Research Site 101

Idaho Falls, Idaho, 83404, United States

Location

Research Site 143

Glenview, Illinois, 60026, United States

Location

Research Site 01

Gurnee, Illinois, 60031, United States

Location

Research Site 141

Gurnee, Illinois, 60031, United States

Location

Research Site 02

Oak Lawn, Illinois, 60453, United States

Location

Research Site 135

South Bend, Indiana, 46635, United States

Location

Research Site 125

Covington, Louisiana, 70433, United States

Location

Research Site 45

Houma, Louisiana, 70363, United States

Location

Research Site 12

Marrero, Louisiana, 70072, United States

Location

Research Site 124

Metairie, Louisiana, 70006, United States

Location

Research Site 48

Metairie, Louisiana, 70006, United States

Location

Research Site 34

New Orleans, Louisiana, 70127, United States

Location

Research Site 25

West Monroe, Louisiana, 71291, United States

Location

Research Site 93

Chesterfield, Michigan, 48047, United States

Location

Research Site 148

Plymouth, Minnesota, 55446, United States

Location

Research Site 140

Flowood, Mississippi, 39232, United States

Location

Research Site 111

Chesterfield, Missouri, 63005, United States

Location

Research Site 137

Columbia, Missouri, 65201, United States

Location

Research Site 138

Kansas City, Missouri, 64128, United States

Location

Research Site 159

Henderson, Nevada, 89052, United States

Location

Research Site 160

Las Vegas, Nevada, 28919, United States

Location

Research Site 73

Las Vegas, Nevada, 33030, United States

Location

Research Site 06

Las Vegas, Nevada, 89106, United States

Location

Research Site 163

Las Vegas, Nevada, 89106, United States

Location

Research Site 127

Las Vegas, Nevada, 89128, United States

Location

Research Site 64

Reno, Nevada, 89511, United States

Location

Research Site 129

Englewood, New Jersey, 07631, United States

Location

Research Site 130

Freehold, New Jersey, 07728, United States

Location

Research Site 131

Jackson, New Jersey, 08527, United States

Location

Research Site 35

Brooklyn, New York, 11235, United States

Location

Research Site 07

Great Neck, New York, 11023, United States

Location

Research Site 28

Hartsdale, New York, 10530, United States

Location

Research Site 58

New York, New York, 10021, United States

Location

Research Site 49

New York, New York, 10033, United States

Location

Research Site 40

Rochester, New York, 14609, United States

Location

Research Site 75

Fayetteville, North Carolina, 84092, United States

Location

Research Site 155

High Point, North Carolina, 27260, United States

Location

Research Site 69

Mount Airy, North Carolina, 27030, United States

Location

Research Site 116

Salisbury, North Carolina, 28144, United States

Location

Research Site 158

Columbus, Ohio, 43212, United States

Location

Research Site 20

Columbus, Ohio, 43213, United States

Location

Research Site 88

Columbus, Ohio, 43215, United States

Location

Research Site 109

Mentor, Ohio, 44060, United States

Location

Research Site 118

Springboro, Ohio, 45066, United States

Location

Research Site 110

Westlake, Ohio, 44145, United States

Location

Research Site 157

Anderson, South Carolina, 29621, United States

Location

Research Site 61

North Charleston, South Carolina, 29405, United States

Location

Research Site 128

Hermitage, Tennessee, 37076, United States

Location

Research Site 114

Kingsport, Tennessee, 37663, United States

Location

Research Site 60

Nashville, Tennessee, 37203, United States

Location

Research Site 103

Nashville, Tennessee, 37211, United States

Location

Research Site 50

Shelbyville, Tennessee, 37160, United States

Location

Research Site 100

Bellaire, Texas, 77401, United States

Location

Research Site 98

Dallas, Texas, 75230, United States

Location

Research Site 99

Forney, Texas, 75126, United States

Location

Research Site 154

Houston, Texas, 77024, United States

Location

Research Site 162

Houston, Texas, 77084, United States

Location

Research Site 68

Katy, Texas, 77494, United States

Location

Research Site 29

Lewisville, Texas, 75057, United States

Location

Research Site 161

McAllen, Texas, 78503, United States

Location

Research Site 32

Pearland, Texas, 77584, United States

Location

Research Site 30

Red Oak, Texas, 75154, United States

Location

Research Site 22

San Antonio, Texas, 78209, United States

Location

Research Site 26

San Antonio, Texas, 78229, United States

Location

Research Site 21

San Antonio, Texas, 78249, United States

Location

Research Site 80

Tomball, Texas, 77375, United States

Location

Research Site 134

Waco, Texas, 76710, United States

Location

Research Site 105

Ogden, Utah, 84403, United States

Location

Research Site 57

Salt Lake City, Utah, 84107, United States

Location

Research Site 65

Sandy City, Utah, 84092, United States

Location

Research Site 16

South Ogden, Utah, 84405, United States

Location

Research Site 77

Chesapeake, Virginia, 23320, United States

Location

Research Site 136

Richmond, Virginia, 23236, United States

Location

Research Site 97

Morgantown, West Virginia, 26505, United States

Location

Study Officials

  • Leah Hollins

    Braintree Laboratories / Sebela Pharmaceuticals

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 17, 2022

First Posted

October 20, 2022

Study Start

October 30, 2022

Primary Completion

June 16, 2025

Study Completion

June 16, 2025

Last Updated

September 24, 2025

Record last verified: 2025-09

Data Sharing

IPD Sharing
Will not share

Locations