NCT05432167

Brief Summary

This study will evaluate the efficacy and safety of CIN-107 for the treatment of hypertension in patients with uncontrolled hypertension (uHTN) and Chronic Kidney Disease (CKD).

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
195

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Apr 2022

Geographic Reach
1 country

71 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

April 29, 2022

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

June 20, 2022

Completed
7 days until next milestone

First Posted

Study publicly available on registry

June 27, 2022

Completed
1.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 2, 2024

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 2, 2024

Completed
1 year until next milestone

Results Posted

Study results publicly available

May 20, 2025

Completed
Last Updated

May 20, 2025

Status Verified

April 1, 2025

Enrollment Period

2 years

First QC Date

June 20, 2022

Results QC Date

March 25, 2025

Last Update Submit

May 2, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Mean Seated Systolic Blood Pressure (SBP) of Pooled CIN-107 and Placebo

    Mean change in seated SBP from baseline to Week 26 of pooled CIN-107 and placebo was assessed.

    At Week 26

Secondary Outcomes (2)

  • Change From Baseline in SBP in CIN-107 Compared to Placebo in Participants Assigned to the High-dose Strategy Group

    At Week 26

  • Change From Baseline of SBP in CIN-107 Compared to Placebo in Participants Assigned to the Low-dose Strategy Group

    At Week 26

Other Outcomes (1)

  • Number of Participants With Treatment Emergent Adverse Events (TEAEs)

    From randomization (Day 1) until the end of Follow up period (approximately 8 months)

Study Arms (3)

Low dose CIN-107

EXPERIMENTAL

Patients will take oral tablets of CIN-107 for 26 weeks. The dose strength may be titrated within 6 weeks.

Drug: CIN-107

High dose CIN-107

EXPERIMENTAL

Patients will take oral tablets of CIN-107 for 26 weeks. The dose strength may be titrated within 6 weeks.

Drug: CIN-107

Placebo

PLACEBO COMPARATOR

Patients will take oral tablets of Placebo for 26 weeks. The dose strength may be titrated within 6 weeks.

Drug: Placebo

Interventions

Patients will take CIN-107 tablets by mouth once daily.

High dose CIN-107Low dose CIN-107

Patients will take placebo tablets by mouth once daily.

Placebo

Eligibility Criteria

Age18 Years - 130 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has a mean seated SBP ≥ 140 mmHg.
  • Has a prior diagnosis of mild-to-severe CKD.
  • Has an elevated UACR.
  • Is currently taking an angiotensin-converting enzyme inhibitor (ACEi) or angiotensin receptor blocker (ARB) at the maximum tolerated daily dose.

You may not qualify if:

  • Have a documented diagnosis of type 1 diabetes.
  • Are not willing or not able to discontinue a mineralocorticoid receptor antagonist (MRA) or a potassium sparing diuretic as part of an existing antihypertensive regimen.
  • Have a single occurrence of mean seated SBP \>180 mmHg or DBP \>110 mmHg during the Screening Period.
  • Has a body mass index (BMI) \>50 kg/m\^2.
  • Has documented bilateral clinically relevant renal artery stenosis of ≥70%.
  • Has had dialysis for acute kidney injury/acute renal failure within 12 weeks prior to the Screening Period or has a planned dialysis or kidney transplantation during the course of the study.
  • Has known documented chronic heart failure New York Heart Association Class III or Class IV and/or hospitalization for heart failure within 6 months of Screening.
  • Has had a stroke, transient ischemic attack, hypertensive encephalopathy, acute coronary syndrome, or hospitalization for heart failure within 6 months of Screening.
  • Has known current severe left ventricular outflow obstruction, such as obstructive hypertrophic cardiomyopathy and/or severe aortic valvular disease.
  • Has planned any major cardiac surgery during the study or had major cardiac surgery within 6 months of Screening.
  • Has had a prior solid organ transplant or cell transplant.
  • Has a known hypersensitivity to CIN-107 or drugs of the same class
  • Has received immunotherapy for treatment of CKD within 6 months of Screening.
  • Has any clinically relevant medical or surgical conditions including unstable conditions and/or conditions requiring regular transfusion or treatment with systemic immunosuppressants, including corticosteroids.
  • Serum potassium \<3.5 mEq/L or \>5.0 mEq/L
  • +6 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (71)

Research Site

Birmingham, Alabama, 35209, United States

Location

Research Site

Huntsville, Alabama, 35805, United States

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Research Site

Beverly Hills, California, 90211, United States

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Research Site

Chula Vista, California, 91910, United States

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Fountain Valley, California, 92708, United States

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Research Site

Granada Hills, California, 91344, United States

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Research Site

Lancaster, California, 93534, United States

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Research Site

Lincoln, California, 95648, United States

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Research Site

Los Angeles, California, 90010, United States

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Research Site

Lynwood, California, 90262, United States

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Northridge, California, 91324, United States

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Research Site

Panorama City, California, 91402, United States

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Research Site

Pomona, California, 91767, United States

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Research Site

Rancho Cucamonga, California, 91730, United States

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Research Site

Riverside, California, 92503, United States

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San Dimas, California, 91773, United States

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South Gate, California, 90280, United States

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Tarzana, California, 91356, United States

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Vacaville, California, 95687, United States

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Victorville, California, 92392, United States

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Arvada, Colorado, 80002, United States

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Littleton, Colorado, 80120, United States

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Hollywood, Florida, 33021, United States

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Orlando, Florida, 32807, United States

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Orlando, Florida, 32808, United States

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Tampa, Florida, 33612, United States

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West Palm Beach, Florida, 33401, United States

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Columbus, Georgia, 31904, United States

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Decatur, Georgia, 30030, United States

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Nampa, Idaho, 83687, United States

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Chicago, Illinois, 60643, United States

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Brownsburg, Indiana, 46112, United States

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Lexington, Kentucky, 40503, United States

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Metairie, Louisiana, 70006, United States

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Monroe, Louisiana, 71201, United States

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Silver Spring, Maryland, 20904, United States

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New Bedford, Massachusetts, 02740, United States

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Flint, Michigan, 48504, United States

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Research Site

Flint, Michigan, 48532, United States

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Research Site

Troy, Michigan, 48085, United States

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Olive Branch, Mississippi, 38654, United States

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Kansas City, Missouri, 64111, United States

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Trenton, New Jersey, 08611, United States

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The Bronx, New York, 10455, United States

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Durham, North Carolina, 27704, United States

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Greenville, North Carolina, 27834, United States

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Kinston, North Carolina, 28504, United States

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Morganton, North Carolina, 28655, United States

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Oxford, North Carolina, 27565, United States

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Wilmington, North Carolina, 28401, United States

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Cincinnati, Ohio, 45246, United States

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Bethany, Oklahoma, 73008, United States

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Scottdale, Pennsylvania, 15683, United States

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Smithfield, Pennsylvania, 15478, United States

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Providence, Rhode Island, 02903, United States

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Memphis, Tennessee, 38119, United States

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Houston, Texas, 77099, United States

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Research Site

Lampasas, Texas, 76550, United States

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Paris, Texas, 75462, United States

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Red Oak, Texas, 75154, United States

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San Antonio, Texas, 78212, United States

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Research Site

San Antonio, Texas, 78249, United States

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Salt Lake City, Utah, 84132, United States

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Burlington, Vermont, 05401, United States

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Research Site

Alexandria, Virginia, 22304, United States

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Research Site

Burke, Virginia, 22015, United States

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Research Site

Charlottesville, Virginia, 22908, United States

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Research Site

Manassas, Virginia, 20110, United States

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Research Site

Newport News, Virginia, 23606, United States

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Research Site

Salem, Virginia, 24153, United States

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Research Site

Kingwood, West Virginia, 26537, United States

Location

Related Publications (2)

  • Dwyer JP, Maklad N, Vedin O, Monyak J, Myte R, Chertow GM, Heerspink HJL, Little DJ. Efficacy and Safety of Baxdrostat in Participants with CKD and Uncontrolled Hypertension: A Randomized, Double-Blind, Placebo-Controlled Trial. J Am Soc Nephrol. 2025 Sep 6. doi: 10.1681/ASN.0000000849. Online ahead of print. No abstract available.

  • Townsend RR. Blocking Aldosterone Synthesis: Whose BrigHTN Idea Was That? Clin J Am Soc Nephrol. 2023 Dec 1;18(12):1631-1633. doi: 10.2215/CJN.0000000000000265. Epub 2023 Jul 24. No abstract available.

Related Links

MeSH Terms

Conditions

Renal Insufficiency, Chronic

Condition Hierarchy (Ancestors)

Renal InsufficiencyKidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Results Point of Contact

Title
Global Clinical Lead
Organization
AstraZeneca

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 20, 2022

First Posted

June 27, 2022

Study Start

April 29, 2022

Primary Completion

May 2, 2024

Study Completion

May 2, 2024

Last Updated

May 20, 2025

Results First Posted

May 20, 2025

Record last verified: 2025-04

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data from AstraZeneca group of companies sponsored clinical trials via the request portal Vivli.org. All requests will be evaluated as per the AZ disclosure commitment: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure. "Yes", indicates that AZ are accepting requests for IPD, but this does not mean all requests will be approved.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
AstraZeneca will meet or exceed data availability as per the commitments made to the EFPIA/PhRMA Data-Sharing Principles. For details of our timelines, please refer to our disclosure commitment at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
Access Criteria
When a request has been approved AstraZeneca will provide access to the anonymized individual patient-level data via secure research environment Vivli.org. A Signed Data Usage Agreement (non-negotiable contract for data accessors) must be in place before accessing requested information.
More information

Locations