NCT05063539

Brief Summary

The purpose of this study is to assess the safety, tolerability and effect of study drug LY3372689 in participants with early symptomatic Alzheimer's Disease

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
327

participants targeted

Target at P75+ for phase_2 alzheimer-disease

Timeline
Completed

Started Sep 2021

Typical duration for phase_2 alzheimer-disease

Geographic Reach
5 countries

69 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 14, 2021

Completed
2 days until next milestone

Study Start

First participant enrolled

September 16, 2021

Completed
15 days until next milestone

First Posted

Study publicly available on registry

October 1, 2021

Completed
2.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 9, 2024

Completed
11 months until next milestone

Study Completion

Last participant's last visit for all outcomes

May 22, 2025

Completed
2 months until next milestone

Results Posted

Study results publicly available

July 28, 2025

Completed
Last Updated

July 28, 2025

Status Verified

July 1, 2025

Enrollment Period

2.8 years

First QC Date

September 14, 2021

Results QC Date

July 9, 2025

Last Update Submit

July 9, 2025

Conditions

Keywords

DementiaMild Cognitive ImpairmentProdromal Alzheimer's DiseaseTauopathyTauOGA Inhibitor

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline to End Time Point in Integrated Alzheimer's Disease Rating Scale (iADRS) (Intermediate (Low-medium) Tau Population)

    iADRS is a simple linear combination of scores from 13-item alzheimer's disease assessment scale-cognitive subscale (ADAS-Cog13) and the Alzheimer's disease cooperative study-instrumental activities of daily living scale (ADCS-iADL). It is used to assess whether LY3372689 slows down the cognitive and functional decline associated with early symptomatic Alzheimer's Disease, compared to placebo. The iADRS score ranges from 0 to 144 with lower scores indicating worse performance and higher score better performance. Change from baseline was calculated using Bayesian disease progression model (DPM) adjusted for age at baseline, AChEI/Memantine use at baseline, pooled investigator. Data presented are posterior mean with 95% credible interval.

    Baseline, Week 100

Secondary Outcomes (14)

  • Change From Baseline to End Time Point in iADRS (Overall Population)

    Baseline, Week 100

  • Change From Baseline to End Time Point in Clinical Dementia Rating Scale - Sum of Boxes (CDR-SB) (Intermediate (Low-medium) Tau Population)

    Baseline, Week 76

  • Change From Baseline to End Time Point in Clinical Dementia Rating Scale - Sum of Boxes (CDR-SB) (Overall Population)

    Baseline, Week 76

  • Change From Baseline to End Time Point in Alzheimer's Disease Assessment Scale - Cognitive Subscale (ADAS-Cog13) (Intermediate (Low-medium) Tau Population)

    Baseline, Week 76

  • Change From Baseline to End Time Point in Alzheimer's Disease Assessment Scale - Cognitive Subscale (ADAS-Cog13) (Overall Population)

    Baseline, Week 76

  • +9 more secondary outcomes

Study Arms (3)

0.75 Milligram (mg) LY3372689

EXPERIMENTAL

Participants received 0.75 mg LY3372689 administered orally once daily for up to 124 weeks

Drug: LY3372689

3 mg LY3372689

EXPERIMENTAL

Participants received 3 mg LY3372689 administered orally once daily for up to 124 weeks.

Drug: LY3372689

Placebo

PLACEBO COMPARATOR

Participants received placebo administered orally once daily for up to 124 weeks.

Drug: Placebo

Interventions

given orally

0.75 Milligram (mg) LY3372689

given orally

Placebo

Eligibility Criteria

Age60 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Gradual and progressive change in memory function reported by participants or informants for ≥ 6 months
  • MMSE score of 22 to 30 (inclusive) at screening
  • CDR global score of 0.5 to 1.0 (inclusive), with a memory box score ≥0.5.
  • Meet 18F flortaucipir positron emission tomography (PET) scan (central analysis) criteria
  • Have a study partner who will provide written informed consent to participate

You may not qualify if:

  • Contraindication to MRI or PET scans
  • Have known allergies to LY3372689, related compounds, or any components of the formulations

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (69)

Hope Clinical Research, Inc.

Canoga Park, California, 91303, United States

Location

Neuro-Pain Medical Center

Fresno, California, 93710, United States

Location

Irvine Clinical Research

Irvine, California, 92614, United States

Location

Sharp Mesa Vista Hospital

San Diego, California, 92123, United States

Location

Institute for Neurodegenerative Disorders

New Haven, Connecticut, 06510, United States

Location

JEM Research Institute

Atlantis, Florida, 33462, United States

Location

VIN-Julie Schwartzbard

Aventura, Florida, 33180, United States

Location

Neurology Offices of South Florida

Boca Raton, Florida, 33428, United States

Location

Brain Matters Research

Delray Beach, Florida, 33445, United States

Location

Neuropsychiatric Research Center of Southwest Florida

Fort Myers, Florida, 33912, United States

Location

K2 Medical Research

Maitland, Florida, 32751, United States

Location

ClinCloud - Viera

Melbourne, Florida, 32940, United States

Location

Merritt Island Medical Research, LLC

Merritt Island, Florida, 32952, United States

Location

VIN-Andrew Lerman

Miami, Florida, 33133, United States

Location

IMIC, Inc.

Miami, Florida, 33176, United States

Location

VIN-Victor Faradji

Miami, Florida, 33176, United States

Location

Suncoast Clinical Research, Inc.

New Port Richey, Florida, 34652, United States

Location

Renstar Medical Research

Ocala, Florida, 34470, United States

Location

VIN- Margarita Almeida El-Ramey

Pembroke Pines, Florida, 33026, United States

Location

Brain Matters Research

Stuart, Florida, 34997, United States

Location

Charter Research - Lady Lake

The Villages, Florida, 32162, United States

Location

Josephson Wallack Munshower Neurology, PC

Indianapolis, Indiana, 46256, United States

Location

Boston Center for Memory

Newton, Massachusetts, 02459, United States

Location

Donald S. Marks M.D., P.C.

Plymouth, Massachusetts, 02360, United States

Location

MedVadis Research Corporation

Waltham, Massachusetts, 02451, United States

Location

Adams Clinical

Watertown, Massachusetts, 02472, United States

Location

The Cognitive and Research Center of New Jersey

Springfield, New Jersey, 07081, United States

Location

Advanced Memory Research Institute of New Jersey

Toms River, New Jersey, 08755, United States

Location

University at Buffalo - UBMD Neurology

Buffalo, New York, 14203, United States

Location

Abington Neurological Associates, Ltd.

Abington, Pennsylvania, 19001, United States

Location

Keystone Clinical Studies

Plymouth Meeting, Pennsylvania, 19462, United States

Location

Rhode Island Mood & Memory Research Institute

East Providence, Rhode Island, 02914, United States

Location

Kerwin Medical Center

Dallas, Texas, 75231, United States

Location

The University of Texas Health Science Center at Houston

Houston, Texas, 77054, United States

Location

The Memory Clinic

Bennington, Vermont, 05201-9810, United States

Location

Central Coast Neurosciences Research (Tumbi Umbi)

Central Coast, New South Wales, 2261, Australia

Location

St Vincent's Hospital

Sydney, New South Wales, 2010, Australia

Location

HammondCare Greenwich Hospital

Sydney, New South Wales, 2065, Australia

Location

Hornsby Ku-Ring-Gai Hospital

Sydney, New South Wales, 2077, Australia

Location

KARA Institute for Neurological Diseases

Sydney, New South Wales, 2113, Australia

Location

Private Practice - Dr PL Morris

Southport, Queensland, 4215, Australia

Location

The Queen Elizabeth Hospital

Woodville, South Australia, 5011, Australia

Location

Box Hill Hospital

Box Hill, Victoria, 3128, Australia

Location

NeuroCentrix

Carlton, Victoria, 3053, Australia

Location

Delmont Private Hospital

Glen Iris, Victoria, 3146, Australia

Location

HammondCare

Malvern, Victoria, 3144, Australia

Location

Bruyère Research Institute

Ottawa, Ontario, K1N 5C8, Canada

Location

Clinique de la Mémoire de l'Outaouais

Ottawa, Ontario, K1Z 1G3, Canada

Location

Ottawa Memory Clinic

Ottawa, Ontario, K1Z 1G3, Canada

Location

Toronto Memory Program

Toronto, Ontario, M3B 2S7, Canada

Location

Diex Recherche Sherbrooke Inc.

Sherbrooke, Quebec, J1L 0H8, Canada

Location

National Center for Geriatrics and Gerontology

Ōbu, Aichi-ken, 4748511, Japan

Location

Himeji Central Hospital Affiliated Clinic

Himeji, Hyōgo, 672-8043, Japan

Location

Kobe City Medical Center General Hospital

Kobe, Hyōgo, 650-0047, Japan

Location

Memory Clinic Toride

Toride, Ibaraki, 302-0004, Japan

Location

Oita University Hospital

Yufu, Oita Prefecture, 879-5593, Japan

Location

Katayama Medical Clinic

Kurashiki, Okayama-ken, 710-0813, Japan

Location

Nozomi Memory Clinic

Mitaka-shi, Tokyo, 181-0013, Japan

Location

Kikukawa Clinic

Nerima City, Tokyo, 179-0072, Japan

Location

Memory Clinic Ochanomizu

Tokyo, 113-0034, Japan

Location

Nzoz Neuro-Kard Ilkowski i Partnerzy SPL

Poznan, Greater Poland Voivodeship, 61-853, Poland

Location

Centrum Medyczne NEUROMED

Bydgoszcz, Kuyavian-Pomeranian Voivodeship, 85-163, Poland

Location

Diamond Clinic

Krakow, Lesser Poland Voivodeship, 31-559, Poland

Location

Wroclawskie Centrum Alzheimerowskie

Wroclaw, Lower Silesian Voivodeship, 53-203, Poland

Location

Centrum Medyczne NeuroProtect

Warsaw, Masovian Voivodeship, 01-684, Poland

Location

Podlaskie Centrum Psychogeriatrii

Bialystok, Podlaskie Voivodeship, 15-756, Poland

Location

Centrum Badan Klinicznych PI-House sp. z o.o.

Gdansk, Pomeranian Voivodeship, 80-546, Poland

Location

Centrum Medyczne SENIOR

Sopot, Pomeranian Voivodeship, 81-855, Poland

Location

Centrum Medyczne Euromedis

Szczecin, West Pomeranian Voivodeship, 70-111, Poland

Location

Related Links

MeSH Terms

Conditions

Alzheimer DiseaseDementiaCognitive DysfunctionTauopathiesPick Disease of the Brain

Condition Hierarchy (Ancestors)

Brain DiseasesCentral Nervous System DiseasesNervous System DiseasesNeurodegenerative DiseasesNeurocognitive DisordersMental DisordersCognition DisordersFrontotemporal DementiaFrontotemporal Lobar Degeneration

Results Point of Contact

Title
Chief Medical Officer
Organization
Eli Lilly and Company

Study Officials

  • Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

    Eli Lilly and Company

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
GT60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Based on a common closed study design. Participants final endpoint time will be between 76-124 weeks.
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 14, 2021

First Posted

October 1, 2021

Study Start

September 16, 2021

Primary Completion

July 9, 2024

Study Completion

May 22, 2025

Last Updated

July 28, 2025

Results First Posted

July 28, 2025

Record last verified: 2025-07

Data Sharing

IPD Sharing
Will share

Anonymized individual patient level data will be provided in a secure access environment upon approval of a research proposal and a signed data sharing agreement.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
Data are available 6 months after the primary publication and approval of the indication studied in the US and European Union (EU), whichever is later. Data will be indefinitely available for requesting.
Access Criteria
A research proposal must be approved by an independent review panel and researchers must sign a data sharing agreement.
More information

Locations