NCT04888728

Brief Summary

An open label, 2-part, one-sequence, 3-period study to evaluate drug-drug interactions between DWN12088 and nebivolol or Paroxetine in healthy volunteers

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
24

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started Jun 2021

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 28, 2021

Completed
19 days until next milestone

First Posted

Study publicly available on registry

May 17, 2021

Completed
1 month until next milestone

Study Start

First participant enrolled

June 30, 2021

Completed
12 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 12, 2021

Completed
15 days until next milestone

Study Completion

Last participant's last visit for all outcomes

July 27, 2021

Completed
Last Updated

August 4, 2021

Status Verified

August 1, 2021

Enrollment Period

12 days

First QC Date

April 28, 2021

Last Update Submit

August 3, 2021

Conditions

Outcome Measures

Primary Outcomes (4)

  • Cmax of Nebivolol

    Cmax of Nebivolol

    Day 1, Day 2, Day 3, Day 6, Day 7, and Day 8

  • AUCt of Nebivolol

    AUCt of Nebivolol

    Day 1, Day 2, Day 3, Day 6, Day 7, and Day 8

  • Cmax of DWN12088

    Cmax of DWN12088

    Day 1, Day 2, Day 3, Day 4, Day 9, Day 10, Day 11, and Day 12

  • AUCt of DWN12088

    AUCt of DWN12088

    Day 1, Day 2, Day 3, Day 4, Day 9, Day 10, Day 11, and Day 12

Study Arms (2)

DWN12088 and Nebivolol

EXPERIMENTAL

Period 1 - Nebivolol A mg, Tablet, oral, once daily, Period 2 - DWN12088 X mg, Tablet, oral, twice daily, Period 3 - 1) Nebivolol A mg, Tablet, oral, once daily \& DWN12088 X mg, Tablet, oral, twice daily, 2) DWN12088 X mg, Tablet, oral, once daily

Drug: DWN12088Drug: Nebivolol

DWN12088 and Paroxetine

EXPERIMENTAL

Period 1 - DWN12088 X mg, Tablet, oral, once daily , Period 2 - Paroxetine B mg, Tablet, oral, once daily, Period 3 - 1) DWN12088 X mg, Tablet, oral, once daily \& Paroxetine B mg, Tablet, oral, once daily, 2) Paroxetine B mg, Tablet, oral, once daily

Drug: DWN12088Drug: Paroxetine

Interventions

Prolyl-tRNA synthetase (PRS) inhibitor

DWN12088 and NebivololDWN12088 and Paroxetine

Nebivolol

DWN12088 and Nebivolol

Paroxetine

DWN12088 and Paroxetine

Eligibility Criteria

Age20 Years - 55 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy male adults aged ≥ 20 and ≤ 55 years at screening
  • Subjects who voluntarily decided to participate in the study and provided written consent to follow study compliance requirements after receiving a detailed explanation on this study and fully understanding the information

You may not qualify if:

  • Subjects unable to have the standard meal provided at the study site
  • Subjects who took (the day of taking the last dose) another investigational or bioequivalence study product within 180 days prior to the first dose

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Inje University Busan Paik Hospital

Busan, 47397, South Korea

Location

MeSH Terms

Conditions

Idiopathic Pulmonary Fibrosis

Interventions

NebivololParoxetine

Condition Hierarchy (Ancestors)

Pulmonary FibrosisLung Diseases, InterstitialLung DiseasesRespiratory Tract Diseases

Intervention Hierarchy (Ancestors)

EthanolaminesAmino AlcoholsAlcoholsOrganic ChemicalsAminesBenzopyransPyransHeterocyclic Compounds, 1-RingHeterocyclic CompoundsHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingPiperidines

Study Officials

  • Jong-Lyul Ghim

    Busan Paik Hospital

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 28, 2021

First Posted

May 17, 2021

Study Start

June 30, 2021

Primary Completion

July 12, 2021

Study Completion

July 27, 2021

Last Updated

August 4, 2021

Record last verified: 2021-08

Locations