NCT04803864

Brief Summary

Depite successful primary percutaneous coronary intervention (PCI) and standardized medical treatment, prognosis of acute ST-elevation myocardial infarction patents are still a poor, with high morality and various complications such as heart failure. Roxadustat is a new drug targeting hypoxia-inducible factor prolyl hydroxylase (HIF-PH) inhibition and has shown promising effect in reducing infarct size in pre-clinical studies. This study aims to evaluate the efficacy and safety of early and short-term administration of roxadustat in the treatment of acute ST-elevation myocardial infarction.

Trial Health

43
At Risk

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Trial has exceeded expected completion date
Enrollment
158

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Jun 2021

Geographic Reach
1 country

1 active site

Status
unknown

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 2, 2021

Completed
1 month until next milestone

First Posted

Study publicly available on registry

March 18, 2021

Completed
3 months until next milestone

Study Start

First participant enrolled

June 10, 2021

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 30, 2022

Completed
11 months until next milestone

Study Completion

Last participant's last visit for all outcomes

August 31, 2023

Completed
Last Updated

September 1, 2021

Status Verified

August 1, 2021

Enrollment Period

1.3 years

First QC Date

February 2, 2021

Last Update Submit

August 31, 2021

Conditions

Keywords

ST Elevation Myocardial InfarctionRoxadustatInfarct SizeCardiac MRI

Outcome Measures

Primary Outcomes (1)

  • Infarct Size

    Infarct size as a percentage of LV mass measured on delayed-enhanced CMR imaging 30 days post-MI compared to control

    30 days

Secondary Outcomes (4)

  • MACE

    0 - 1 year

  • Left Ventricular Function

    1 month, 6 months, 1 year

  • Cardiac enzymes - peak concentration

    0 - 3 days

  • Cardiac enzymes - Area under curve

    0 - 3 days

Other Outcomes (1)

  • Myocardial fibrosis

    30 days

Study Arms (2)

Roxadustat

EXPERIMENTAL

Early and short-term Roxadustat treatment

Drug: Roxadustat

Control

NO INTERVENTION

Patients only receive conventional therapies as recommended by guidelines.

Interventions

Orally 100mg, 3 times per week for 2 weeks First dose administered immediately after successful PCI.

Also known as: Evrenzo
Roxadustat

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Acute STEMI (ST segment elevation myocardial infarction) diagnosed by ST elevation
  • Coronary angiography within 12 hours of symptom onset, with TIMI flow grade 0 - 1 of culprit vessel
  • Primary PCI with TIMI flow grade 2 - 3 after successful intervention
  • Capable and willing to provide informed consent and capable of completing study visits

You may not qualify if:

  • Previous acute myocardial infarction history
  • Cardiogenic Shock at admission
  • Previously treated by roxadustat
  • Contraindications of roxadustat treatment
  • Contraindication of Cardiac MRI (e.g. eGFR \< 30 ml/min, pacemaker, metal prosthesis, etc.)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Ruijin Hospital

Shanghai, Shanghai Municipality, 200025, China

RECRUITING

Related Publications (6)

  • Howell NJ, Tennant DA. The role of HIFs in ischemia-reperfusion injury. Hypoxia (Auckl). 2014 Jul 30;2:107-115. doi: 10.2147/HP.S49720. eCollection 2014.

    PMID: 27774470BACKGROUND
  • Sousa Fialho MDL, Abd Jamil AH, Stannard GA, Heather LC. Hypoxia-inducible factor 1 signalling, metabolism and its therapeutic potential in cardiovascular disease. Biochim Biophys Acta Mol Basis Dis. 2019 Apr 1;1865(4):831-843. doi: 10.1016/j.bbadis.2018.09.024. Epub 2018 Sep 25.

    PMID: 30266651BACKGROUND
  • Schreiber T, Salhofer L, Quinting T, Fandrey J. Things get broken: the hypoxia-inducible factor prolyl hydroxylases in ischemic heart disease. Basic Res Cardiol. 2019 Mar 11;114(3):16. doi: 10.1007/s00395-019-0725-2.

    PMID: 30859331BACKGROUND
  • Chen N, Hao C, Peng X, Lin H, Yin A, Hao L, Tao Y, Liang X, Liu Z, Xing C, Chen J, Luo L, Zuo L, Liao Y, Liu BC, Leong R, Wang C, Liu C, Neff T, Szczech L, Yu KP. Roxadustat for Anemia in Patients with Kidney Disease Not Receiving Dialysis. N Engl J Med. 2019 Sep 12;381(11):1001-1010. doi: 10.1056/NEJMoa1813599. Epub 2019 Jul 24.

    PMID: 31340089BACKGROUND
  • Deguchi H, Ikeda M, Ide T, Tadokoro T, Ikeda S, Okabe K, Ishikita A, Saku K, Matsushima S, Tsutsui H. Roxadustat Markedly Reduces Myocardial Ischemia Reperfusion Injury in Mice. Circ J. 2020 May 25;84(6):1028-1033. doi: 10.1253/circj.CJ-19-1039. Epub 2020 Mar 24.

    PMID: 32213720BACKGROUND
  • Groenendaal-van de Meent D, den Adel M, Rijnders S, Krebs-Brown A, Kerbusch V, Golor G, Schaddelee M. The Hypoxia-inducible Factor Prolyl-Hydroxylase Inhibitor Roxadustat (FG-4592) and Warfarin in Healthy Volunteers: A Pharmacokinetic and Pharmacodynamic Drug-Drug Interaction Study. Clin Ther. 2016 Apr;38(4):918-28. doi: 10.1016/j.clinthera.2016.02.010. Epub 2016 Mar 4.

    PMID: 26947173BACKGROUND

MeSH Terms

Conditions

ST Elevation Myocardial Infarction

Interventions

roxadustat

Condition Hierarchy (Ancestors)

Myocardial InfarctionMyocardial IschemiaHeart DiseasesCardiovascular DiseasesVascular DiseasesInfarctionIschemiaPathologic ProcessesPathological Conditions, Signs and SymptomsNecrosis

Study Officials

  • Ruiyan Zhang, M.D., Ph.D.

    Ruijin Hospital

    PRINCIPAL INVESTIGATOR

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
SINGLE
Who Masked
OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Director of Cardiology Department, Chief Physician

Study Record Dates

First Submitted

February 2, 2021

First Posted

March 18, 2021

Study Start

June 10, 2021

Primary Completion

September 30, 2022

Study Completion

August 31, 2023

Last Updated

September 1, 2021

Record last verified: 2021-08

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data by contacting principle investigator of this study. Requests for IPD will be recieved, but this does not mean all requests will be shared by the investigators.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
1 year after the end of this study
Access Criteria
Please contact the investigators through email in the time frame.

Locations