NCT03985293

Brief Summary

This multicenter, randomized, double-blind, placebo controlled, parallel group study is being conducted to provide data on efficacy, safety, tolerability and pharmacokinetics (PK) of multiple dose levels of PF-06882961 in adults with type 2 diabetes mellitus (T2DM) inadequately controlled on metformin and/or diet and exercise. In addition, the study is intended to enable selection of efficacious doses for future clinical development of PF-06882961.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
412

participants targeted

Target at P75+ for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started Oct 2019

Typical duration for phase_2 diabetes-mellitus-type-2

Geographic Reach
8 countries

83 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 11, 2019

Completed
2 days until next milestone

First Posted

Study publicly available on registry

June 13, 2019

Completed
4 months until next milestone

Study Start

First participant enrolled

October 15, 2019

Completed
1.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 8, 2021

Completed
29 days until next milestone

Study Completion

Last participant's last visit for all outcomes

July 7, 2021

Completed
12 months until next milestone

Results Posted

Study results publicly available

June 30, 2022

Completed
Last Updated

June 30, 2022

Status Verified

June 1, 2022

Enrollment Period

1.6 years

First QC Date

June 11, 2019

Results QC Date

June 2, 2022

Last Update Submit

June 2, 2022

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Glycated Hemoglobin (HbA1c) at Week 16

    HbA1c can be used as a diagnostic test for diabetes. The target HbA1c level for people with diabetes is usually less than 7%.

    Baseline, Week 16

Secondary Outcomes (22)

  • Percentage of Participants Achieving Less Than (<) 7% Glycated Hemoglobin (HbA1c) Levels

    Baseline, Week 16

  • Change From Baseline in Glycated Hemoglobin (HbA1c) at Week 2

    Baseline, Week 2

  • Change From Baseline in Glycated Hemoglobin (HbA1c) at Week 4

    Baseline, Week 4

  • Change From Baseline in Glycated Hemoglobin (HbA1c) at Week 6

    Baseline, Week 6

  • Change From Baseline in Glycated Hemoglobin (HbA1c) at Week 8

    Baseline, Week 8

  • +17 more secondary outcomes

Study Arms (6)

Placebo

PLACEBO COMPARATOR
Drug: Placebo

PF-06882961 2.5 milligrams (mg)

EXPERIMENTAL
Drug: PF-06882961

PF-06882961 10 mg

EXPERIMENTAL
Drug: PF-06882961

PF-06882961 40 mg

EXPERIMENTAL

Participants will be titrated up to 2 weeks to reach desired dose level

Drug: PF-06882961

PF-06882961 80 mg

EXPERIMENTAL

Participants will be titrated up to 4 weeks to reach desired dose level

Drug: PF-06882961

PF-06882961 120 mg

EXPERIMENTAL

Participants will be titrated up to 6 weeks to reach desired dose level

Drug: PF-06882961

Interventions

4 matching placebo tablets taken twice a day (BID)

Placebo

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

PF-06882961 10 mgPF-06882961 120 mgPF-06882961 2.5 milligrams (mg)PF-06882961 40 mgPF-06882961 80 mg

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patients with T2DM who are treated with metformin and/or diet and exercise
  • HbA1c greater than or equal to 7% and less than or equal to 10.5%
  • Total body weight \>50 kg (110 lb) with BMI 24.5 to 45.4 kg/m\^2

You may not qualify if:

  • Any condition possibly affecting drug absorption
  • Diagnosis of Type 1 diabetes
  • History of myocardial infarction, unstable angina, arterial revascularization, stroke, heart failure, or transient ischemic attack within 6 months of screening
  • Any malignancy not considered cured
  • Personal or family history of MTC or MEN2, or participants with suspected MTC
  • Acute pancreatitis or history of chronic pancreatitis
  • Symptomatic gallbladder disease
  • Known medical history of active proliferative retinopathy and/or macular edema
  • Known medical history of active liver disease, including chronic active hepatitis B or C, or primary biliary cirrhosis
  • Known history of HIV
  • Supine blood pressure greater than or equal to 160 mmHg (systolic) or greater than or equal to 100 mmHg (diastolic)
  • Clinically relevant ECG abnormalities
  • Positive urine drug test

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (83)

Holy Trinity Medical Clinic

Harbor City, California, 90710, United States

Location

Innovative Clinical Research, Inc.

Harbor City, California, 90710, United States

Location

Long Beach Clinical Trials Services, Inc.

Long Beach, California, 90806, United States

Location

National Research Institute

Los Angeles, California, 90057, United States

Location

Catalina Research Institute, LLC

Montclair, California, 91763, United States

Location

Empire Clinical Research

Pomona, California, 91767, United States

Location

Rancho Cucamonga Clinical Research

Rancho Cucamonga, California, 91730, United States

Location

Encompass Clinical Research

Spring Valley, California, 91978, United States

Location

University Clinical Investigators, Incorporated

Tustin, California, 92780, United States

Location

San Fernando Valley Health Institute, LLC

Van Nuys, California, 91405, United States

Location

Diablo Clinical Research Incorporated

Walnut Creek, California, 94598, United States

Location

Accel Research Sites - DeLand Clinical Research Unit

DeLand, Florida, 32720, United States

Location

East Coast Institute for Research, LLC

Jacksonville, Florida, 32204, United States

Location

East Coast Institute for Research, LLC

Jacksonville, Florida, 32216, United States

Location

New Horizon Research Center

Miami, Florida, 33165, United States

Location

NewPhase Clinical Trials, Corp.

Miami Beach, Florida, 33140, United States

Location

Sunshine Research Center, Inc

Opa-locka, Florida, 33054, United States

Location

Andres Patron D.O. P.A.

Pembroke Pines, Florida, 33026, United States

Location

Ellipsis Group

Alpharetta, Georgia, 30022, United States

Location

East Coast Institute for Research, LLC

Macon, Georgia, 31210, United States

Location

Cedar Crosse Research Center

Chicago, Illinois, 60607, United States

Location

Buynak Clinical Research

Valparaiso, Indiana, 46383, United States

Location

Viable Research Management LLC

Henderson, Nevada, 89014, United States

Location

Premier Research

Trenton, New Jersey, 08611, United States

Location

PharmQuest

Greensboro, North Carolina, 27408, United States

Location

Lillestol Research LLC

Fargo, North Dakota, 58104, United States

Location

Velocity Clinical Research

Cincinnati, Ohio, 45242, United States

Location

Conrad Clinical Research

Edmond, Oklahoma, 73013, United States

Location

Family Medical Associates

Levittown, Pennsylvania, 19056, United States

Location

Preferred Primary Care Physicians, Inc.

Pittsburgh, Pennsylvania, 15236, United States

Location

Spartanburg Medical Research

Spartanburg, South Carolina, 29303, United States

Location

Palmetto Clinical Research

Summerville, South Carolina, 29485, United States

Location

Palmetto Primary Care Physicians (physicals only)

Summerville, South Carolina, 29485, United States

Location

Dallas Diabetes Research Center

Dallas, Texas, 75230, United States

Location

Endocrine Associates

Houston, Texas, 77004, United States

Location

PrimeCare Medical Group

Houston, Texas, 77024, United States

Location

Juno Research, LLC

Houston, Texas, 77074, United States

Location

Northeast Clinical Research of San Antonio

Live Oak, Texas, 78233, United States

Location

Sun Research Institute

San Antonio, Texas, 78215, United States

Location

DM Clinical Research

Tomball, Texas, 77375, United States

Location

Martin Diagnostic Clinic

Tomball, Texas, 77375, United States

Location

Rainier Clinical Research Center, Inc.

Renton, Washington, 98057, United States

Location

MHAT Dobrich AD

Dobrich, 9300, Bulgaria

Location

Medical Center ASKLEPII OOD

Dupnitsa, 2600, Bulgaria

Location

UMHAT Pulmed

Plovdiv, 4002, Bulgaria

Location

Fourth MHAT - Sofia EAD

Sofia, 1606, Bulgaria

Location

MHAT "Doverie" AD

Sofia, 1632, Bulgaria

Location

MC "New rehabilitation center" EOOD

Stara Zagora, 6000, Bulgaria

Location

GA Research Associates Ltd.

Moncton, New Brunswick, E1G 1A7, Canada

Location

Aggarwal and Associates Limited

Brampton, Ontario, L6T 0G1, Canada

Location

Manna Research (Toronto)

Toronto, Ontario, M9W4L6, Canada

Location

Manna Research (Quebec)

Lévis, Quebec, G6W 0M5, Canada

Location

Manna Research (Mirabel)

Mirabel, Quebec, J7J 2K8, Canada

Location

Diex Recherche Quebec Inc.

Québec, Quebec, G1N 4V3, Canada

Location

Alpha Recherche Clinique

Québec, Quebec, G3K2P8, Canada

Location

Diex Recherche Sherbrooke Inc.

Sherbrooke, Quebec, J1L 0H8, Canada

Location

Diex Recherche Victoriaville Inc.

Victoriaville, Quebec, G6P 6P6, Canada

Location

Centre de Recherche Saint-Louis

Québec, G1W 4R4, Canada

Location

Belinus Orvosi es Szamitastechnikai Bt

Debrecen, 4025, Hungary

Location

Debreceni Egyetem Klinikai Kozpont

Debrecen, 4032, Hungary

Location

CRU Hungary Kft.

Miskolc, 3529, Hungary

Location

Borbanya Praxis Egeszsegugyi KFT

Nyíregyháza, H-4405, Hungary

Location

Clinfan Kft.

Szekszárd, H-7100, Hungary

Location

Zdrowie Osteo-Medic s.c. Lidia i Artur Racewicz, Agnieszka i Jerzy Supronik

Bialystok, 15-351, Poland

Location

Medyczne Centrum Diabetologiczno-Endokrynologiczno-Metaboliczne DIAB-ENDO-MET Sp. z o. o.

Krakow, 31-261, Poland

Location

Prywatny Gabinet Lekarski i Wizyty Lekarskie Jan Ruxer

Lodz, 94-060, Poland

Location

MEDICOME Sp. z o.o.

Oświęcim, 32-600, Poland

Location

KO-MED CENTRA KLINICZNE Sp. z o.o. Ośrodek Badań Klinicznych w Puławach

Puławy, 24-100, Poland

Location

Centralny Szpital Kliniczny MSWiA

Warsaw, 02-507, Poland

Location

Metabol KLINIK s.r.o.

Bratislava, 811 08, Slovakia

Location

Medispektrum, s.r.o

Bratislava, 851 01, Slovakia

Location

HUMAN-CARE, s.r.o.

Košice, 040 01, Slovakia

Location

SchronerMED s.r.o.

Moldava nad Bodvou, 04501, Slovakia

Location

Funkystuff, s.r.o.

Nové Zámky, 940 01, Slovakia

Location

DIAB s.r.o.

Rožňava, 048 01, Slovakia

Location

MUDr. Jana Rociakova, s.r.o.

Žilina, 010 01, Slovakia

Location

Yonsei University-Wonju Severance Christian Hospital

Wŏnju, Gangwon-do, 26426, South Korea

Location

Hanyang University Guri Hospital

Guri-si, Gyeonggi-do, 11923, South Korea

Location

Ajou University Hospital

Suwon, Gyeonggi-do, 16499, South Korea

Location

Samsung Medical Center

Gangnam-Gu, Seoul, 06351, South Korea

Location

Far Eastern Memorial Hospital

New Taipei City, 220, Taiwan

Location

Taichung Veterans General Hospital

Taichung, 40705, Taiwan

Location

National Cheng Kung University Hospital

Tainan, 704, Taiwan

Location

Related Publications (1)

  • Saxena AR, Frias JP, Brown LS, Gorman DN, Vasas S, Tsamandouras N, Birnbaum MJ. Efficacy and Safety of Oral Small Molecule Glucagon-Like Peptide 1 Receptor Agonist Danuglipron for Glycemic Control Among Patients With Type 2 Diabetes: A Randomized Clinical Trial. JAMA Netw Open. 2023 May 1;6(5):e2314493. doi: 10.1001/jamanetworkopen.2023.14493.

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Interventions

danuglipron

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Results Point of Contact

Title
Pfizer ClinicalTrials.gov Call Center
Organization
Pfizer Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 11, 2019

First Posted

June 13, 2019

Study Start

October 15, 2019

Primary Completion

June 8, 2021

Study Completion

July 7, 2021

Last Updated

June 30, 2022

Results First Posted

June 30, 2022

Record last verified: 2022-06

Data Sharing

IPD Sharing
Will share

Pfizer will provide access to individual de-identified participant data and related study documents (e.g. protocol, Statistical Analysis Plan (SAP), Clinical Study Report (CSR)) upon request from qualified researchers, and subject to certain criteria, conditions, and exceptions. Further details on Pfizer's data sharing criteria and process for requesting access can be found at: https://www.pfizer.com/science/clinical\_trials/trial\_data\_and\_results/data\_requests.

More information

Locations