NCT03902080

Brief Summary

This study will assess the efficacy of vibegron compared with placebo in men with overactive bladder (OAB) symptoms on pharmacological therapy for benign prostatic hyperplasia (BPH) as defined by micturition and urgency episodes.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
1,105

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Mar 2019

Typical duration for phase_3

Geographic Reach
8 countries

140 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 26, 2019

Completed
6 days until next milestone

First Submitted

Initial submission to the registry

April 1, 2019

Completed
2 days until next milestone

First Posted

Study publicly available on registry

April 3, 2019

Completed
4.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 15, 2023

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 15, 2023

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

August 7, 2024

Completed
Last Updated

August 7, 2024

Status Verified

June 1, 2024

Enrollment Period

4.2 years

First QC Date

April 1, 2019

Results QC Date

June 11, 2024

Last Update Submit

July 15, 2024

Conditions

Keywords

Overactive BladderBenign Prostatic HyperplasiaVibegronBeta-3 adrenergic receptor (ß3-AR)ß3-AR agonist

Outcome Measures

Primary Outcomes (2)

  • Change From Baseline at Week 12 in the Average Number of Micturition Episodes Per Day

    Micturition was defined as the number of times a participant voided in the toilet as indicated on the Bladder Diary. Baseline was defined as the last non-missing result on or prior to the randomization date. Change from baseline was calculated as the post-baseline value minus the baseline value. Daily Averages were calculated as the sum of the event type on Complete Diary Days divided by the number of Complete Diary Days.

    Baseline; Week 12

  • Change From Baseline at Week 12 in the Average Number of Urgency Episodes (Need to Urinate Immediately) Per Day

    Urgency was defined as the number of times a participant checked that they had the need to urinate immediately as indicated on the Bladder Diary. Baseline was defined as the last non-missing result on or prior to the randomization date. Change from baseline was calculated as the post-baseline value minus the baseline value. Daily Averages were calculated as the sum of the event type on Complete Diary Days divided by the number of Complete Diary Days.

    Baseline; Week 12

Secondary Outcomes (4)

  • Change From Baseline at Week 12 in the Average Number of Nocturia Episodes Per Night

    Baseline; Week 12

  • Change From Baseline at Week 12 in the Average Number of Urge Urinary Incontinence (UUI) Episodes Per Day for Participants With Urinary Incontinence at Baseline

    Baseline; Week 12

  • Change From Baseline at Week 12 in the International Prostate Symptom Score (IPSS) Storage Score (1-week Recall)

    Baseline; Week 12

  • Change From Baseline at Week 12 in the Average Volume Voided Per Micturition

    Baseline; Week 12

Study Arms (2)

Vibegron 75 mg

EXPERIMENTAL

Participants will receive vibegron 75 milligrams (mg) orally once daily for 24 weeks.

Drug: Vibegron

Placebo

PLACEBO COMPARATOR

Participants will receive matching placebo orally once daily for 24 weeks.

Drug: Placebo

Interventions

oral administration

Also known as: RVT-901, MK-4618, KRP-114V, URO-901
Vibegron 75 mg

oral administration

Placebo

Eligibility Criteria

Age45 Years+
Sexmale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participant should have been on and agree to continue to stay on a stable dose of benign prostatic hyperplasia (BPH) treatment with either a) alpha blocker monotherapy or b) alpha blocker + 5 alpha reductase inhibitor.
  • Participant has an International Prostate Symptom Score total score of ≥ 8
  • Participant has a prostate-specific antigen level \< 4 nanograms per milliliter (ng/mL), or if ≥ 4 ng/mL but ≤ 10 ng/mL, prostate cancer has been ruled out to the satisfaction of the investigator
  • Participant must have both additional qualifications based on the 3-day Bladder Diary period: a) having an average of ≥ 8 but ≤ 20 micturition episodes per day over the 3-day diary period, and (b) having an average of ≥ 3 urgency episodes per day over the 3-day diary period
  • Participant must have a post void residual volume value of \< 100 mL
  • Having at least 2 average nocturia episodes per night based on 3-day Bladder Diary at baseline. Nocturia is defined as waking to pass urine during the main sleep period.

You may not qualify if:

  • Participant has a history of 24-hour urine volume greater than 3,000 mL
  • Has lower urinary tract pathology that could, in the opinion of the investigator, be responsible for urgency, frequency, or incontinence
  • Has a history of prostate surgery, including minimally invasive transurethral or transrectal procedures, procedural treatments for BPH within 6 months of Screening or has a planned prostate surgery
  • Has a history of urinary retention requiring an intervention (e.g., catheterization) for any reason
  • Has maximum urinary flow (Qmax) \< 5.0 mL/second with a minimum voided volume of 125 mL
  • Has a history of or current nocturnal polyuria
  • Has an active or recurrent (\> 3 episodes per year) urinary tract infection by clinical symptoms or laboratory criteria (≥ 5 white blood cells/high power field \[hpf\] with presence of red blood cell \[RBC\] and/or a positive urine culture, defined as ≥ 10\^5 colony forming units (CFU)/mL (i.e., 100 × 10\^3 CFU/mL in a single specimen)
  • Has uncontrolled hyperglycemia (defined as fasting blood glucose \> 150 milligrams per deciliter (mg/dL) or 8.33 millimoles per liter (mmol/L) or non-fasting blood glucose \> 200 mg/dL or 11.1 mmol/L) or, if in the opinion of the investigator, is uncontrolled
  • Has uncontrolled hypertension (systolic blood pressure of ≥ 180 millimeters of mercury (mmHg) and/or diastolic blood pressure of ≥ 100 mmHg) or has a resting heart rate (by pulse) \> 100 beats per minute (min)
  • Has a history of cerebral vascular accident, transient ischemic attack, unstable angina, myocardial infarction, coronary artery interventions (e.g., coronary artery bypass grafting or percutaneous coronary interventions \[e.g., angioplasty, stent insertion\]), or neurovascular interventions (e.g., carotid artery stenting) within 6 months prior to the Screening Visit
  • Has alanine aminotransferase or aspartate aminotransferase \> 2.0 times the upper limit of normal (ULN), or bilirubin (total bilirubin) \> 1.5 × ULN (or \> 2.0 × ULN if secondary to Gilbert syndrome or pattern consistent with Gilbert syndrome)
  • Has an estimated glomerular filtration rate \< 30 mL/min/1.73 meters squared (m\^2)
  • Has a history or current evidence of any condition, therapy, laboratory abnormality, or other circumstances that might, in the opinion of the investigator, confound the results of the study, interfere with the participant's ability to comply with the study procedure, or make participation in the study not in the participant's best interest

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (140)

Urology Centers of Alabama

Homewood, Alabama, 35209, United States

Location

Private Practice

Huntsville, Alabama, 35801, United States

Location

Coastal Clinical Research, Inc.

Mobile, Alabama, 36608, United States

Location

Gen1 Research- Arizona Urology Specialists

Glendale, Arizona, 85308, United States

Location

Urological Associates Of Southern Arizona

Tucson, Arizona, 85741, United States

Location

California Research Medical Group, Inc.

Fullerton, California, 92835, United States

Location

San Diego Clinical Trials

La Mesa, California, 91942, United States

Location

Clinical Trials Research

Lincoln, California, 95648, United States

Location

West Coast Urology

Los Alamitos, California, 90720, United States

Location

American Institute of Research

Los Angeles, California, 90017, United States

Location

Norris Comprehensive Cancer Center

Los Angeles, California, 90033, United States

Location

Tri Valley Urology Medical Group

Murrieta, California, 92562, United States

Location

Northern California Research Corp

Sacramento, California, 95821, United States

Location

Medical Center for Clinical Research

San Diego, California, 92108, United States

Location

Urology Specialists of Southern California (USSC)

Sherman Oaks, California, 91411, United States

Location

Skyline Urology

Torrance, California, 90505, United States

Location

Urology Associates - Urology

Denver, Colorado, 80220, United States

Location

Imagine Research of Palm Beach County - Urology

Boynton Beach, Florida, 33435, United States

Location

Tampa Bay Medical Research

Clearwater, Florida, 33761, United States

Location

Urological Research Network Corp

Hialeah, Florida, 33016, United States

Location

LCC Medical Research Institute

Miami, Florida, 33126, United States

Location

Quantum Clinical Trials

Miami, Florida, 33140, United States

Location

Private Practice

Orlando, Florida, 32808, United States

Location

Urology Center Of Florida

Pompano Beach, Florida, 33060, United States

Location

Pinellas Urology, Inc.

St. Petersburg, Florida, 33710, United States

Location

Precision Clinical Research

Sunrise, Florida, 33351, United States

Location

Florida Urology Partners, LLP

Tampa, Florida, 33615, United States

Location

Clinical Research of Central Florida

Winter Haven, Florida, 33880, United States

Location

Meridian Clinical Research - Urology

Savannah, Georgia, 31405, United States

Location

Idaho Urologic Institute

Meridian, Idaho, 83642, United States

Location

NorthShore University Health System

Glenview, Illinois, 60153, United States

Location

First Urology

Jeffersonville, Indiana, 47130, United States

Location

The Iowa Clinic

West Des Moines, Iowa, 50266, United States

Location

GU Research Network/Wichita Urology Group

Wichita, Kansas, 67226, United States

Location

DelRicht Research

New Orleans, Louisiana, 70115, United States

Location

Regional Urology, LLC

Shreveport, Louisiana, 71106, United States

Location

Chesapeake Urology Research Associates

Baltimore, Maryland, 21204, United States

Location

Boston Clinical Trials Inc - Urology

Boston, Massachusetts, 02131, United States

Location

Mens Health Boston - Urology

Chestnut Hill, Massachusetts, 02467, United States

Location

Bay State Clinical Trials, Inc.

Watertown, Massachusetts, 02472, United States

Location

Beaumont Hospital Royal Oak - Urology Research

Royal Oak, Michigan, 48703, United States

Location

CentraCare Clinic - Adult & Pediatric Urology

Sartell, Minnesota, 56377, United States

Location

Poplar Bluff Urology

Poplar Bluff, Missouri, 63901, United States

Location

Adult & Pediatric Urology P.C. - Urology

Omaha, Nebraska, 68114, United States

Location

Excel Clinical Research - Internal Medicine

Las Vegas, Nevada, 89109, United States

Location

Private Practice

Las Vegas, Nevada, 89148, United States

Location

Premier Urology Group, LLC

Edison, New Jersey, 08837, United States

Location

New Jersey Urology NJU

Englewood, New Jersey, 07631, United States

Location

New Jersey Urology, LLC

Mount Laurel, New Jersey, 08054, United States

Location

New Jersey Urology, LLC

Voorhees Township, New Jersey, 08043, United States

Location

Albany Medical College

Albany, New York, 12208, United States

Location

Western New York Urology Associates

Buffalo, New York, 14203, United States

Location

AccuMed research Asociates

Garden City, New York, 11530, United States

Location

Urological Surgeons of Long Island

Garden City, New York, 11530, United States

Location

Manhattan Research Associates

New York, New York, 10016, United States

Location

Columbia University Medical Center - Clinical Research

New York, New York, 10032, United States

Location

Weill Cornell Medicine

New York, New York, 10065, United States

Location

Advanced Urology Centers of NY, A Division of Integrated Medical Professionals (IMP)

Plainview, New York, 11803, United States

Location

Private Practice

Poughkeepsie, New York, 12603, United States

Location

Duke Medical Center - Urology

Durham, North Carolina, 27710, United States

Location

Carolina Institute for Clinical Research

Fayetteville, North Carolina, 27612, United States

Location

Alliance Urology Specialists - Greensboro

Greensboro, North Carolina, 27403, United States

Location

Triad Clinical Trials

Greensboro, North Carolina, 27410, United States

Location

Peters Medical Research

High Point, North Carolina, 27262, United States

Location

Associated Urologists of North Carolina - Urology

Raleigh, North Carolina, 27612, United States

Location

Clinical Research Solutions

Middleburg Heights, Ohio, 44130, United States

Location

Lowcountry Urology

North Charleston, South Carolina, 29406, United States

Location

Urology Clinics of North Texas

Dallas, Texas, 75231, United States

Location

Advances In Health, Inc.

Houston, Texas, 77030, United States

Location

Urology San Antonio

San Antonio, Texas, 78229, United States

Location

Discovery Clinical Trials

San Antonio, Texas, 78258, United States

Location

Baylor Scott & White Medical Center

Temple, Texas, 76508, United States

Location

Wasatch Clinical Research LLC

Salt Lake City, Utah, 84107, United States

Location

Urology of Virginia (UVA)

Virginia Beach, Virginia, 23462, United States

Location

Seattle Urology Research Center

Burien, Washington, 98166, United States

Location

Uz Antwerpen

Edegem, Antwerpen, 02650, Belgium

Location

Algemeen Stedelijk Ziekenhuis

Aalst, Oost-Vlaanderen, 09300, Belgium

Location

Onze-Lieve-Vrouwziekenhuis VZW - Campus Aalst

Aalst, Oost-Vlaanderen, 09300, Belgium

Location

AZ Maria Middelares - Campus Maria Middelares

Ghent, Oost-Vlaanderen, 09000, Belgium

Location

UZ Leuven - Campus Gasthuisberg

Leuven, Vlaams Brabant, 03000, Belgium

Location

AZ Delta - Campus Wilgenstraat

Roeselare, West-Vlaanderen, 08800, Belgium

Location

CHU de Liège - Domaine Universitaire du Sart Tilman - Urologie

Liège, 04000, Belgium

Location

Private Practice

Brampton, Ontario, L6T 4S5, Canada

Location

Bluewater Clinical Research Group Inc

Sarnia, Ontario, N7T 4X3, Canada

Location

Sunnybrook Health Sciences Center

Toronto, Ontario, M4N 3M5, Canada

Location

Toronto Western Hospital

Toronto, Ontario, M5T 2S8, Canada

Location

Diex Research Quebec Inc.

Québec, Quebec, G1N 4V3, Canada

Location

Centre Hospitalier Universitaire De Sherbrooke (CHUS)

Sherbrooke, Quebec, J1H 5N4, Canada

Location

Diex Research Sherbrooke Inc.

Sherbrooke, Quebec, J1L 0H8, Canada

Location

Diex Research Victoriaville Inc.

Victoriaville, Quebec, G6P 6P6, Canada

Location

University of Szeged

Szeged, Csongrád megye, 06725, Hungary

Location

DRC Kft.

Sopron, Győr-Moson-Sopron, H-9400, Hungary

Location

Semmelweis Egyetem

Budapest, 01082, Hungary

Location

Jahn Ferenc Dél-Pesti Kórház és Rendelointézet

Budapest, 01204, Hungary

Location

Szarka Ödön Egyesitett Egeszsegügyi es Szocialis Intezmeny

Csongrád, 06640, Hungary

Location

Szabolcs-Szatmár-Bereg Megyei Kórházak és Egyetemi Oktatókór

Nyíregyháza, 04400, Hungary

Location

Uro-Clin Kft.

Pècs, 07621, Hungary

Location

Szent Borbala Korhaz

Tatabánya, 02800, Hungary

Location

Kaunas Hospital of Lithuanian Universoity of Health Sciences

Kaunas, Kaunas County, LT-47144, Lithuania

Location

JSC Saules seimos medicinos centras

Kaunas, Kaunas County, LT-49449, Lithuania

Location

Uab "Vakk"

Kaunas, Kaunas County, LT-50128, Lithuania

Location

Hospital of University of Health Sciences Kauno Klinikos

Kaunas, Kaunas County, LT-50161, Lithuania

Location

Respublikine Klaipedos ligonine - Urology

Klaipėda, Klaipėda County, LT-92231, Lithuania

Location

Klaipedos Universitetine Ligonine (Klaipeda Hospital)

Klaipėda, Klaipėda County, LT-92288, Lithuania

Location

National Cancer Institute

Vilnius, Vilnius County, LT-08660, Lithuania

Location

Republican Vilnius University Hospital

Vilnius, Vilnius County, LT-08660, Lithuania

Location

Vilnius University Hospital Santariskiu Klinikos

Vilnius, Vilnius County, LT-08661, Lithuania

Location

Vilnius City Clinical Hospital

Vilnius, Vilnius County, LT-10207, Lithuania

Location

EuroMediCare Szpital Specjalistyczny z Przychodnia

Wroclaw, Dolnoslaskie Województwo, 54-144, Poland

Location

Clinical Research Center Sp. z o.o., Medic-R Sp. K.

Poznan, Greater Poland Voivodeship, 60-856, Poland

Location

Nasz Lekarz Osrodek Badan Klinicznych

Bydgoszcz, Kuyavian-Pomeranian Voivodeship, 85-650, Poland

Location

Wojewodzki Szpital Specjalist

Wroclaw, Lower Silesian Voivodeship, 51-124, Poland

Location

NZOZ Specjalista

Kutno, Lódzkie, 99-300, Poland

Location

ETG Lodz

Lodz, Lódzkie, 90-302, Poland

Location

Centrum Medyczne PROMED

Krakow, Malopolskie Województwo, 31-513, Poland

Location

Szpital Specjalistyczny Slupsk

Słupsk, Pomeranian Voivodeship, 76-200, Poland

Location

Centrum Urologiczne sp. z o.o.

Mysłowice, Silesian Voivodeship, 41-400, Poland

Location

Centrum Medyczne Linden

Krakow, 37-721, Poland

Location

Medicome Sp. z o.o.

Oświęcim, 32-600, Poland

Location

Nzoz Heureka

Piaseczno, 05-500, Poland

Location

Lexmedica Hanna Durbajlo-Gradziel

Wroclaw, 53-114, Poland

Location

Hospital Garcia de Orta

Almada, 2805-267, Portugal

Location

Centro Clínico Académico Braga, Hospital de Braga

Braga, 4710-243, Portugal

Location

Hospital Senhora de Oliveiro Guimaraes EPE

Guimarães, 4835-044, Portugal

Location

H. Egas Moniz. Centro Hospitalar Lisboa Ocidental

Lisbon, 1349-019, Portugal

Location

Hospital de Santa Maria

Lisbon, 1649-035, Portugal

Location

H. Santo António. Centro Hospitalar do Porto

Porto, 4099-001, Portugal

Location

Hospital Santiago Apostol

Miranda de Ebro, Burgos, 09200, Spain

Location

Hospital Universitario Fundación Alcorcón

Alcorcón, Madrid, 28922, Spain

Location

Hospital Universitario HM Monteprincipe

Boadilla del Monte, Madrid, 28660, Spain

Location

Hospital General Universitario Gregorio Marañón

Majadahonda, Madrid, 28007, Spain

Location

Hospital Universitario Puerta de Hierro Majadahonda

Majadahonda, Madrid, 28222, Spain

Location

Hospital Universitario Infanta Sofía

San Sebastián de los Reyes, Madrid, 28702, Spain

Location

Hospital del Mar

Barcelona, 08003, Spain

Location

Hospital Universitario Reina Sofia

Córdoba, 14004, Spain

Location

Clínica Universitaria de Navarra

Madrid, 28027, Spain

Location

Hospital Universitario 12 de Octubre

Madrid, 28041, Spain

Location

H.U. Virgen de la Victoria

Málaga, 29010, Spain

Location

Hospital Universitario de Salamanca

Salamanca, 37007, Spain

Location

Hospital Universitari i Politecnic La Fe

Valencia, 46026, Spain

Location

Related Publications (1)

  • Rovner ES, Owens-Grillo J, Thomas E, Herschorn S, Peters KM, Staskin D, Mujais S. Bladder Function and Safety of Vibegron in Men With Overactive Bladder Receiving Treatment for Benign Prostatic Hyperplasia: Outcomes From the Phase 3 Randomized Controlled COURAGE Trial. Neurourol Urodyn. 2025 Dec 9. doi: 10.1002/nau.70199. Online ahead of print.

MeSH Terms

Conditions

Urinary Bladder, OveractiveProstatic Hyperplasia

Interventions

N-(4-((5-(hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-4-oxo-4,6,7,8-tetrahydropyrrolo(1,2-a)pyrimidine-6-carboxamide

Condition Hierarchy (Ancestors)

Urinary Bladder DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesLower Urinary Tract SymptomsUrological ManifestationsSigns and SymptomsPathological Conditions, Signs and SymptomsProstatic DiseasesGenital Diseases, MaleGenital Diseases

Results Point of Contact

Title
Information, Clinical Trial Results
Organization
Urovant Sciences

Study Officials

  • Study Director

    Urovant Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 1, 2019

First Posted

April 3, 2019

Study Start

March 26, 2019

Primary Completion

June 15, 2023

Study Completion

June 15, 2023

Last Updated

August 7, 2024

Results First Posted

August 7, 2024

Record last verified: 2024-06

Data Sharing

IPD Sharing
Will share

Urovant is committed to sharing patient-level data and supporting clinical documents from eligible studies with qualified external researchers. Data requests will be reviewed and approved on the basis of scientific merit. All data provided will be anonymized according to applicable laws and regulations.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
The data will be made available within 24 months after study completion and will be accessible for a time frame appropriate for the approved proposal.
Access Criteria
Access to these clinical trial data can be requested by emailing medinfo@urovant.com and will be provided following Urovant review and approval of a research proposal and execution of a Data Sharing Agreement (DSA).

Locations