NCT03802565

Brief Summary

This is a double-blind, randomized, placebo-controlled, parallel group study of the efficacy and safety of tolperisone (a non-opioid) or placebo administered as multiple doses three times a day (TID) in approximately 400 male and female subjects experiencing back pain due to or associated with muscle spasm.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
415

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2019

Shorter than P25 for phase_2

Geographic Reach
1 country

43 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 10, 2019

Completed
4 days until next milestone

First Posted

Study publicly available on registry

January 14, 2019

Completed
18 days until next milestone

Study Start

First participant enrolled

February 1, 2019

Completed
5 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 28, 2019

Completed
14 days until next milestone

Study Completion

Last participant's last visit for all outcomes

July 12, 2019

Completed
1.3 years until next milestone

Results Posted

Study results publicly available

November 10, 2020

Completed
Last Updated

February 1, 2022

Status Verified

January 1, 2022

Enrollment Period

5 months

First QC Date

January 10, 2019

Results QC Date

October 19, 2020

Last Update Submit

January 28, 2022

Conditions

Outcome Measures

Primary Outcomes (1)

  • Mean Effect Size in Subjected-Rated Pain

    Mean effect size between Tolperisone and Placebo of subject-rated pain due to acute back spasm using a Numerical Rating Scale (NRS; 0-10 scale, from no pain to worst possible pain) on Day 14 "right now."

    Day 1 to Day 14

Study Arms (5)

Tolperisone 50 mg

EXPERIMENTAL

TID (150 mg/day)

Drug: Tolperisone

Tolperisone 100 mg

EXPERIMENTAL

TID (300 mg/day)

Drug: Tolperisone

Tolperisone 150 mg

EXPERIMENTAL

TID (450 mg/day)

Drug: Tolperisone

Tolperisone 200 mg

EXPERIMENTAL

TID (600 mg/day)

Drug: Tolperisone

Placebo

PLACEBO COMPARATOR

TID

Drug: Placebo

Interventions

TID

Tolperisone 100 mgTolperisone 150 mgTolperisone 200 mgTolperisone 50 mg

Placebo

Placebo

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Ambulatory
  • Current acute back pain and/or stiffness due to acute and painful muscle spasm starting within 7 days prior to study entry and more than 8 weeks after the last episode of acute back pain.
  • Pain of 4 or more on the subject "right now" rating of pain intensity Numeric Rating Scale (NRS) scale of 0-10.
  • Willing to discontinue all medication used for the treatment of pain or muscle spasm on study entry.
  • Pain localized below the neck and above the inferior gluteal folds.
  • Body mass index ranging between 18 and 35 kg/m².

You may not qualify if:

  • Unwillingness to stop taking pain or antispasmodic medication other than the study medication (specifically opioid use \[e.g., Vicodin\], barbiturates, and cannabis).
  • Chronic pain for the previous 3 months or longer, on more days than not.
  • Radicular pain in the lower extremity (i.e. pain radiating below the knee), sciatica pain down the leg, or pain below the knee (indicating a lumber radiculopathy); radicular pain in the upper extremity, radiating into the forearm or hand (indicating a cervical radiculopathy).
  • Concomitant severe pain in a region other than the back.
  • Spinal surgery within 1 year of study entry.
  • Back pain due to major trauma (e.g., motor vehicle accident, fracture of bone) unless resolved for more than 1 year.
  • Treatment of back pain ongoing with non-pharmacological therapy (e.g., acupuncture, chiropractic adjustment, massage, Transcutaneous Electrical Nerve Stimulation \[TENS\], physiotherapy).
  • Subjects who test positive for alcohol by breathalyzer test.
  • Unwilling to stop taking moderate to potent inhibitors of cytochrome P450 (CYP) isozymes CYP2D6 and CYP2C19, which are likely to cause drug interactions with tolperisone HCl (e.g., medications such as paroxetine and fluvoxamine).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (43)

Tennessee Valley Pain Consultants

Huntsville, Alabama, 35801, United States

Location

Fiel Family and Sports Medicine

Tempe, Arizona, 85283, United States

Location

Center of Applied Research

Little Rock, Arkansas, 72212, United States

Location

Research Center of Fresno

Fresno, California, 93702, United States

Location

Long Beach Clinical Trials Services, Inc.

Long Beach, California, 90806, United States

Location

Northern California Research

Sacramento, California, 95628, United States

Location

Pacific Research Network, LLC

San Diego, California, 92103, United States

Location

San Diego Sports Medicine

San Diego, California, 92120, United States

Location

CITrials

Santa Ana, California, 92705, United States

Location

Riverside Clinical Research

Edgewater, Florida, 32132, United States

Location

Empirical Research Group

Gainesville, Florida, 32653, United States

Location

LLC Medical Research

Miami, Florida, 33126, United States

Location

Savin Medical Group

Miami Lakes, Florida, 33014, United States

Location

Avail Clinical Research

Orange City, Florida, 32763, United States

Location

Private Practice

Plantation, Florida, 33313, United States

Location

NeuroTrials Research, Inc.

Atlanta, Georgia, 30342, United States

Location

Georgia Institute for Clinical Research

Marietta, Georgia, 30060, United States

Location

Georgia Clinical Research

Snellville, Georgia, 30078, United States

Location

MediSphere Medical Research Center

Evansville, Indiana, 47714, United States

Location

Otrimed Clinical Research

Edgewood, Kentucky, 41017, United States

Location

Centex Studies, Inc.

Lake Charles, Louisiana, 70601, United States

Location

Center for Rheumatology and Bone

Wheaton, Maryland, 20902, United States

Location

Michigan Head Pain and Neurological

Ann Arbor, Michigan, 48104, United States

Location

Sundance Clinical Research

St Louis, Missouri, 63141, United States

Location

Jubilee Clinical Research

Las Vegas, Nevada, 89106, United States

Location

Albuquerque Clinical Trials, Inc.

Albuquerque, New Mexico, 87102, United States

Location

Upstate Clinical Research Associates

Williamsville, New York, 14221, United States

Location

Clinical Trials of America

Winston-Salem, North Carolina, 27103, United States

Location

Sterling Research Group- Springdale

Cincinnati, Ohio, 45246, United States

Location

Cleveland Clinic

Cleveland, Ohio, 44195, United States

Location

Center for Providence Health Partners

Dayton, Ohio, 45439, United States

Location

IPS Research

Oklahoma City, Oklahoma, 73103, United States

Location

Williamette Valley Clinical Studies

Eugene, Oregon, 97404, United States

Location

Frontier Clinical Research, Inc.

Smithfield, Pennsylvania, 15478, United States

Location

Omega Medical Research

Warwick, Rhode Island, 02886, United States

Location

Health Concepts

Rapid City, South Dakota, 57702, United States

Location

Inquest Clinical Research

Baytown, Texas, 77521, United States

Location

DiscoveResearch, Inc.

Bryan, Texas, 77802, United States

Location

HD Research Corp

Houston, Texas, 77004, United States

Location

Centex Studies, Inc.

McAllen, Texas, 78504, United States

Location

ClinRX Research Joseph, Inc.

Plano, Texas, 75007, United States

Location

Highland Clinical Research

Salt Lake City, Utah, 84124, United States

Location

Health Research of Hampton Roads, Inc.

Newport News, Virginia, 23606, United States

Location

MeSH Terms

Conditions

Back PainAcute PainMuscle CrampSpasmLow Back Pain

Interventions

Tolperisone

Condition Hierarchy (Ancestors)

PainNeurologic ManifestationsSigns and SymptomsPathological Conditions, Signs and SymptomsMuscular DiseasesMusculoskeletal DiseasesNeuromuscular ManifestationsNervous System Diseases

Intervention Hierarchy (Ancestors)

PropiophenonesKetonesOrganic ChemicalsPyridinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Results Point of Contact

Title
Randall Kaye, MD - Chief Medical Officer
Organization
Neurana Pharmaceuticals, Inc.

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 10, 2019

First Posted

January 14, 2019

Study Start

February 1, 2019

Primary Completion

June 28, 2019

Study Completion

July 12, 2019

Last Updated

February 1, 2022

Results First Posted

November 10, 2020

Record last verified: 2022-01

Data Sharing

IPD Sharing
Will not share

Locations