NCT03471988

Brief Summary

The objective of this study is to investigate the safety and efficacy of administering 372.6 mg of AK1820 (isavuconazonium sulfate) intravenously or orally to adult Japanese patients with deep mycosis. The primary endpoint is safety (percentage of patients with adverse events after starting the study treatment).

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
103

participants targeted

Target at P25-P50 for phase_3

Timeline
Completed

Started Apr 2018

Typical duration for phase_3

Geographic Reach
1 country

33 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 26, 2018

Completed
23 days until next milestone

First Posted

Study publicly available on registry

March 21, 2018

Completed
26 days until next milestone

Study Start

First participant enrolled

April 16, 2018

Completed
3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 21, 2021

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 21, 2021

Completed
Last Updated

May 14, 2021

Status Verified

January 1, 2021

Enrollment Period

3 years

First QC Date

February 26, 2018

Last Update Submit

May 13, 2021

Conditions

Keywords

deep mycosisaspergillosismucormycosiscryptococcosisisavuconazonium sulfateisavuconazoleAK1820Cresemba

Outcome Measures

Primary Outcomes (1)

  • Percentage of patients with adverse events between the first administration of investigational product and the end of Follow-up.

    From the first study drug administration until 28 days after the last dose of study drug (up to approximately Day 112).

Secondary Outcomes (4)

  • Percentage of participants with an overall outcome of success evaluated by the data review committee (DRC).

    Day 42, Day 84 and End of Treatment* (maximum Day 84).*End of treatment (EOT) is defined as the last day of study drug treatment.

  • Percentage of participants with clinical, radiological and mycological response assessed by the DRC.

    Day 42, Day 84 and End of Treatment* (maximum Day 84).*End of treatment (EOT) is defined as the last day of study drug treatment.

  • Percentage of participants with overall outcome, clinical, radiological and mycological response evaluated by investigator.

    Day 42, Day 84 and End of Treatment* (maximum Day 84).*End of treatment (EOT) is defined as the last day of study drug treatment.

  • All-cause mortality.

    Through 28 days after the last dose of study drug (up to approximately Day 112).

Study Arms (2)

AK1820

EXPERIMENTAL

Participants will receive a loading dose of isavuconazole, 200 mg three times a day by intravenous infusion (IV) or orally for the first 2 days followed by a maintenance dose from Day 3 of 200 mg once daily either IV or orally until they will reach a treatment endpoint or for a maximum of 84 days.

Drug: AK1820

Voriconazole

ACTIVE COMPARATOR

Participants will receive a loading dose of voriconazole, 6 mg/kg every 12 hours IV or 300 mg every 12 hours orally for the first 24 hours, followed by a maintenance dose from Day 2 of 4 mg/kg every 12 hours by IV or 200 mg every 12 hours orally, until they will reach a treatment endpoint or for a maximum of 84 days.

Drug: Voriconazole

Interventions

AK1820DRUG

Only a switch from IV infusion (vial) to oral administration (capsule) will be permitted; a switch from oral administration to IV infusion will not be possible. 372.6 mg of AK1820 (isavuconazonium sulfate) is equivalent to 200 mg of isavuconazole. Other Names: Cresemba, BAL8557

AK1820

Only a switch from IV infusion (vial) to oral administration (tablet) will be permitted; a switch from oral administration to IV infusion will not be possible. Other Name : VFend

Voriconazole

Eligibility Criteria

Age20 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patients must have the below proven, probable or possible deep mycosis;
  • invasive aspergillosis
  • chronic pulmonary aspergillosis
  • mucormycosis
  • cryptococcosis
  • Female patients must be non-lactating and at no risk for pregnancy.

You may not qualify if:

  • Women who are pregnant or breastfeeding.
  • Patients with hypersensitivity to any of the components of the azole class of antifungals or the investigational product.
  • Patients at high risk for QT/QTc prolongation, or patients with risk factors for torsades de pointes, or taking concomitant medications known to prolong the QT/QTc interval.
  • Patients with a history of short QT syndrome.
  • Patients with liver dysfunction at enrollment.
  • Patients with moderate to severe kidney dysfunction at enrollment.
  • Patients who receive prohibited concomitant drugs.
  • Patients with any other fungal infection other than Aspergillus species, order Mucorales, or Cryptococcus species.
  • Patients who are not expected to survive study duration.
  • Patients with an underlying disease, complication or general condition that would complicate safety and efficacy evaluations.
  • Patients with a history of taking voriconazole for deep mycosis and showing no response to this treatment.
  • Patients taking systemic antifungals who are unable to stop taking these drugs during the study, or who are showing signs of improvement in their symptoms of deep mycosis as a result of these drugs.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (33)

Research site

Nagakute, Aichi-ken, Japan

Location

Research site

Nagoya, Aichi-ken, Japan

Location

Research site

Seto, Aichi-ken, Japan

Location

Research site

Higashiku, Fukuoka, Japan

Location

Research site

Minamiku, Fukuoka, Japan

Location

Research site

Nagara, Gifu, Japan

Location

Research site

Naka-Ku, Hiroshima, Japan

Location

Research site

Asahikawa, Hokkaido, Japan

Location

Research site

Kawasaki, Kanagawa, Japan

Location

Research site

Yokohama, Kanagawa, Japan

Location

Research site

Chuo-Ku, Kumamoto, Japan

Location

Research site

Tsu, Mie-ken, Japan

Location

Research site

Isahaya, Nagasaki, Japan

Location

Research site

Ōmura, Nagasaki, Japan

Location

Research site

Sasebo, Nagasaki, Japan

Location

Research site

Tenri, Nara, Japan

Location

Research site

Yufu, Oita Prefecture, Japan

Location

Research site

Kurashiki, Okayama-ken, Japan

Location

Research site

Nakagami, Okinawa, Japan

Location

Research site

Abeno-Ku, Osaka, Japan

Location

Research site

Sakai, Osaka, Japan

Location

Research site

Ōmiya, Saitama, Japan

Location

Research site

Hamamatsu, Shizuoka, Japan

Location

Research site

Shimotsuke, Tochigi, Japan

Location

Research site

Kiyose, Tokyo, Japan

Location

Research site

Minato-Ku, Tokyo, Japan

Location

Research site

Mitaka, Tokyo, Japan

Location

Research site

Ōta-ku, Tokyo, Japan

Location

Research site

Shinagawa-Ku, Tokyo, Japan

Location

Research site

Shinjuku-Ku, Tokyo, Japan

Location

Research site

Chiba, Japan

Location

Research site

Ibaraki, Japan

Location

Research site

Nagasaki, Japan

Location

Related Publications (2)

  • Kohno S, Izumikawa K, Takazono T, Miyazaki T, Yoshida M, Kamei K, Ogawa K, Taniguchi S, Akashi K, Tateda K, Mukae H, Miyazaki Y, Okada F, Kanda Y, Kakeya H, Suzuki J, Kimura SI, Kishida M, Matsuda M, Niki Y. Efficacy and safety of isavuconazole against deep-seated mycoses: A phase 3, randomized, open-label study in Japan. J Infect Chemother. 2023 Feb;29(2):163-170. doi: 10.1016/j.jiac.2022.10.010. Epub 2022 Oct 25.

  • Shirae S, Ose A, Kumagai Y. Pharmacokinetics, Safety, and Tolerability of Single and Multiple Doses of Isavuconazonium Sulfate in Healthy Adult Japanese Subjects. Clin Pharmacol Drug Dev. 2022 Jun;11(6):744-753. doi: 10.1002/cpdd.1079. Epub 2022 Feb 21.

MeSH Terms

Conditions

AspergillosisMucormycosisCryptococcosis

Interventions

isavuconazoleVoriconazole

Condition Hierarchy (Ancestors)

MycosesBacterial Infections and MycosesInfectionsZygomycosis

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 26, 2018

First Posted

March 21, 2018

Study Start

April 16, 2018

Primary Completion

April 21, 2021

Study Completion

April 21, 2021

Last Updated

May 14, 2021

Record last verified: 2021-01

Data Sharing

IPD Sharing
Will not share

Locations