NCT03412006

Brief Summary

The purpose of the trial is the analysis of safety and efficacy of the chymase inhibitor BAY1142524 at a dose of 25 mg BID in comparison to placebo using a 6 months treatment period in type II diabetic patients with a clinical diagnosis of diabetic kidney disease. BAY1142524 or placebo will be given on top of evidence-based standard of care for diabetic kidney disease. Primary objective is the analysis of first signs of efficacy as determined by favourable changes in urinary albumin creatinine ratio. Secondary objective is the analysis of safety and tolerability as evidenced by the incidence and severity of adverse events. 64 valid patients have to complete treatment with verum and 32 valid patients have to complete treatment with placebo.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
152

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2018

Geographic Reach
7 countries

27 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 22, 2018

Completed
4 days until next milestone

First Posted

Study publicly available on registry

January 26, 2018

Completed
7 days until next milestone

Study Start

First participant enrolled

February 2, 2018

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 2, 2019

Completed
8 days until next milestone

Study Completion

Last participant's last visit for all outcomes

October 10, 2019

Completed
Last Updated

March 3, 2022

Status Verified

February 1, 2022

Enrollment Period

1.7 years

First QC Date

January 22, 2018

Last Update Submit

February 16, 2022

Conditions

Keywords

type II diabetesdiabetic kidney disease

Outcome Measures

Primary Outcomes (1)

  • Change in urinary albumin to creatinine ratio (UACR)

    The ratio of albumin to creatinin will be determined in first morning void urine at baseline (before treatment start) and after 6 months of treatment

    Baseline and at 6 months

Secondary Outcomes (2)

  • Number of patients with treatment-emergent adverse event

    From first intake of study drug up to 3 days after last administration of study drug

  • Number of patients with serious adverse events

    From first intake of study drug up to 3 days after last administration of study drug

Study Arms (2)

Fulacimstat (BAY1142524)

EXPERIMENTAL

Patients have to have a clinical diagnosis of diabetic kidney disease and have to be treated with standard of care for this condition

Drug: Fulacimstat (BAY1142524)

Placebo

PLACEBO COMPARATOR

Patients have to have a clinical diagnosis of diabetic kidney disease and have to be treated with standard of care for this condition

Drug: Placebo

Interventions

25 mg BAY1142524 are given twice daily over a treatment period of 6 months

Fulacimstat (BAY1142524)

Matching placebo tablets are given twice daily over a treatment period of 6 months

Placebo

Eligibility Criteria

Age18 Years - 79 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patients with Type 2 Diabetes Mellitus and a clinical diagnosis of diabetic kidney disease (DKD) (as judged by the investigator) who have finished their up-titration with an angiotensin receptor blocker (ARB) or an ACEI (angiotensin-converting enzyme inhibitor) to their maximum tolerated dose at least 3 months prior to the screening visit, whereby the maximum tolerated dose has to be at least as high as the minimal recommended dose of an ARB or ACEI according to local and/or international guidelines. Patients have to be treated with an ARB or ACEI, but not with both simultaneously, without any adjustments to this therapy for at least 4 weeks prior to the screening visit.
  • UACR \>50 mg/g and \<3000 mg/g in 2 out of 3 consecutive morning void samples at the screening and the baseline visit
  • estimated glomerular filtration rate (eGFR) ≥30 mL/min/1.73 m\*2 and \<90 mL/min/1.73 m\*2 (Chronic Kidney Disease Epidemiology Collaboration \[CKD-EPI\]) at the screening visit and the baseline visit

You may not qualify if:

  • Non-DKD if it is the main diagnosis contributory to chronic kidney disease (CKD), as judged by the investigator
  • Known bilateral clinical relevant renal artery stenosis (\>75%)
  • New York Heart Association (NYHA) Class IV
  • Acute kidney injury or dialysis within the last 3 months before the screening visit
  • Renal replacement therapy during study conduct
  • Renal allograft in place or a scheduled kidney transplant during study conduct
  • Stroke, transient ischemic cerebral attack, acute coronary syndrome, or hospitalization for heart failure in the last 3 months prior to screening visit
  • Clinically relevant hepatic dysfunction
  • Uncontrolled hypertension as evidenced by systolic blood pressure \>160 mmHg, diastolic blood pressure \>100 mmHg (mean of triplicate values at the screening or baseline visit)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (27)

Med Centre Diamedical 2013

Dimitrovgrad, 6400, Bulgaria

Location

MCOMH Preventsia-2000

Stara Zagora, 6000, Bulgaria

Location

Med. Center Equita

Varna, 9000, Bulgaria

Location

Rigshospitalet

Copenhagen, 2100, Denmark

Location

Steno Diabetes Center Copenhagen

Gentofte Municipality, 2730, Denmark

Location

Nordsjællands Hospital

Hillerød, 3400, Denmark

Location

Pihlajalinna ITE Kuopio

Kuopio, 70100, Finland

Location

Terveystalo Oulu

Oulu, FI-90100, Finland

Location

TAYS TKI Keskus Tutkimusvastaanotto

Tampere, 33520, Finland

Location

Turun yliopistollinen keskussairaala, kantasairaala

Turku, FIN-20520, Finland

Location

Barzilai Medical Center

Ashkelon, 7830604, Israel

Location

Edith Wolfson Medical Center

Holon, 5822012, Israel

Location

Hadassah Hebrew University Hospital Ein Kerem

Jerusalem, 9112001, Israel

Location

The Nazareth Trust Hospital EMMS

Nazareth, 16100, Israel

Location

DMC - Diabetes Medical Center

Tel Aviv, 6937947, Israel

Location

Shamir Medical Center (Assaf Harofeh)

Ẕerifin, 7030000, Israel

Location

IRCCS Casa Sollievo della Sofferenza

Foggia, Apulia, 71013, Italy

Location

A.O.U. Policlinico Federico II Napoli

Napoli, Campania, 80131, Italy

Location

Univ. Alma Mater - Dip. Medicina Spec, Diagnostica e Sperim

Bologna, Emilia-Romagna, 40138, Italy

Location

A.O.U. di Padova

Padua, Veneto, 35128, Italy

Location

Complexo Hospitalario Universitario de Ferrol

Ferrol, A Coruña, 15405, Spain

Location

Hospital de Galdakao

Galdakao, Vizcaya, 48960, Spain

Location

Hospital Fundació Puigvert

Barcelona, 08025, Spain

Location

Centralsjukhuset Kristianstad

Kristianstad, 29185, Sweden

Location

Universitetssjukhuset Örebro

Örebro, 701 85, Sweden

Location

Akardo MedSite AB

Stockholm, 114 46, Sweden

Location

S3 Clinical Research Centers

Vällingby, 162 68, Sweden

Location

Related Links

MeSH Terms

Conditions

Diabetic NephropathiesDiabetes Mellitus, Type 2

Interventions

fulacimstat

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesDiabetes ComplicationsDiabetes MellitusEndocrine System DiseasesGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 22, 2018

First Posted

January 26, 2018

Study Start

February 2, 2018

Primary Completion

October 2, 2019

Study Completion

October 10, 2019

Last Updated

March 3, 2022

Record last verified: 2022-02

Locations