NCT03350386

Brief Summary

This is an open-label, 2-period add-on study to assess the drug-drug interaction between FYU-981 and oxaprozin. The purpose of this study is to investigate the pharmacokinetics of each period in a single administration of FYU-981 and concomitant administration of FYU-981 with oxaprozin at steady -state in healthy volunteers.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
12

participants targeted

Target at below P25 for phase_1 healthy

Timeline
Completed

Started Nov 2017

Shorter than P25 for phase_1 healthy

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 2, 2017

Completed
17 days until next milestone

First Submitted

Initial submission to the registry

November 19, 2017

Completed
3 days until next milestone

First Posted

Study publicly available on registry

November 22, 2017

Completed
13 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 5, 2017

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 5, 2017

Completed
Last Updated

September 14, 2022

Status Verified

September 1, 2022

Enrollment Period

1 month

First QC Date

November 19, 2017

Last Update Submit

September 9, 2022

Conditions

Outcome Measures

Primary Outcomes (9)

  • Pharmacokinetics (Cmax: Maximum plasma concentration)

    48 hours

  • Pharmacokinetics (Tmax: Time to reach the peak plasma concentration)

    48 hours

  • Pharmacokinetics (T1/2: Elimination half-life of plasma concentration)

    48 hours

  • Pharmacokinetics (AUC: Area under the plasma concentration-time curve)

    48 hours

  • Pharmacokinetics (CLtot/F: Total clearance / Fraction of dose absorbed)

    48 hours

  • Pharmacokinetics (kel: Elimination rate constant)

    48 hours

  • Pharmacokinetics (Vd/F: Distribution volume / Fraction of dose absorbed)

    48 hours

  • Pharmacokinetics (MRT: Mean residence time)

    48 hours

  • Safety (Incidence of treatment-emergent adverse event)

    20 days

Study Arms (2)

Single dose

EXPERIMENTAL

Single administration of FYU-981

Drug: FYU-981

Concomitant administration

EXPERIMENTAL

Concomitant administration of FYU-981 with oxaprozin at steady state

Drug: FYU-981Drug: Oxaprozin

Interventions

Single administration

Concomitant administrationSingle dose

Repeated administration

Concomitant administration

Eligibility Criteria

Age20 Years - 35 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Adult healthy subjects
  • Body mass index: \>=18.5 and \<25.0

You may not qualify if:

  • Subject with any disease or any history of disease that might be unsuitable for participation in the clinical study

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

P-One Clinic

Hachiōji, Tokyo, 192-0071, Japan

Location

Related Publications (1)

  • Furihata K, Nagasawa K, Hagino A, Kumagai Y. A drug-drug interaction study of a novel, selective urate reabsorption inhibitor dotinurad and the non-steroidal anti-inflammatory drug oxaprozin in healthy adult males. Clin Exp Nephrol. 2020 Mar;24(Suppl 1):36-43. doi: 10.1007/s10157-020-01855-2. Epub 2020 Feb 19.

MeSH Terms

Interventions

dotinuradOxaprozin

Intervention Hierarchy (Ancestors)

PropionatesAcids, AcyclicCarboxylic AcidsOrganic ChemicalsOxazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • Nagasawa Katsuaki

    Clinical Research Department

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 19, 2017

First Posted

November 22, 2017

Study Start

November 2, 2017

Primary Completion

December 5, 2017

Study Completion

December 5, 2017

Last Updated

September 14, 2022

Record last verified: 2022-09

Data Sharing

IPD Sharing
Will not share

Locations