NCT03335904

Brief Summary

Sleep disordered breathing (SDB) is characterized by regular periods of no breathing (apnea) or low levels of breathing (hypopnea) and leads to repeated periods of low oxygenation, termed intermittent hypoxia that causes fluctuations in blood oxygen levels. This leads to increased peripheral chemoreflex sensitivity that is thought to occur through the stimulation of angiotensin-II, type-I receptors (AT1R) that are expressed primarily on glomus cells within the peripheral chemoreflex and ultimately results in long lasting hypertension. The goal of this study is to determine if AT1R receptor blockade can prevent the increase in chemoreflex sensitivity following one night of hypoxia and improve the severity of SDB.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
14

participants targeted

Target at below P25 for phase_4

Timeline
Completed

Started Jan 2018

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

November 1, 2017

Completed
7 days until next milestone

First Posted

Study publicly available on registry

November 8, 2017

Completed
2 months until next milestone

Study Start

First participant enrolled

January 1, 2018

Completed
1.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2019

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2019

Completed
Last Updated

September 4, 2020

Status Verified

September 1, 2020

Enrollment Period

1.6 years

First QC Date

November 1, 2017

Last Update Submit

September 2, 2020

Conditions

Keywords

Angiotensin receptor blockadecontrol of breathingbreath-holding

Outcome Measures

Primary Outcomes (1)

  • apnea-hypopnea index

    the number of apnea and hypopneas per hour during sleep in hypoxia

    8 hours

Secondary Outcomes (6)

  • Average oxygen saturation

    8 hours

  • Hyperoxic Hypercapnic Ventilatory Response

    0 and 8 hours

  • Hypoxic Hypercapnic Ventilatory Response

    0 and 8 hours

  • Change in systolic and diastolic blood pressure during breath-hold

    0 and 8 hours

  • Hyperoxic Hypercapnic Cerebral Blood Flow Response

    0 and 8 hours

  • +1 more secondary outcomes

Study Arms (2)

Placebo

PLACEBO COMPARATOR

Participants will ingest microcrystalline cellulose by mouth on two consecutive days. The first tablet will be consumed on day 1 at 0700 hrs. The second tablet will be consumed at 1900 hrs and the final tablet will be consumed at 0700hrs on day 2. Participants will undergo a Hyperoxic Hypercapnic Ventilatory Response Test, a Hypoxic Hypercapnic Ventilatory Response Test, and Repeated Hypoxic Apneas before and after a Hypoxic Sleep Study.

Other: Hyperoxic Hypercapnic Ventilatory Response TestOther: Hypoxic Hypercapnic Ventilatory Response TestOther: Repeated Hypoxic ApneasOther: Hypoxic Sleep StudyDrug: Placebo

Losartan

EXPERIMENTAL

Participants will ingest 50 mg of losartan, an angiotensin receptor blocker, by mouth on two consecutive days. The first tablet will be consumed on day 1 at 0700 hrs. The second tablet will be consumed at 1900 hrs and the final tablet will be consumed at 0700hrs on day 2. Participants will undergo a Hyperoxic Hypercapnic Ventilatory Response Test, a Hypoxic Hypercapnic Ventilatory Response Test, and Repeated Hypoxic Apneas before and after a Hypoxic Sleep Study.

Other: Hyperoxic Hypercapnic Ventilatory Response TestOther: Hypoxic Hypercapnic Ventilatory Response TestOther: Repeated Hypoxic ApneasOther: Hypoxic Sleep StudyDrug: Losartan

Interventions

End-tidal PO2 will be clamped at 300 mmHg while end-tidal PCO2 will be increased in three minutes stages from baseline to +2, +4, and +6 mmHg.

LosartanPlacebo

End-tidal PO2 will be clamped at normoxic levels while end-tidal PCO2 will be increased in three minutes stages from baseline to +2, +4, and +6 mmHg.

LosartanPlacebo

Six hypoxic apnea cycles will be performed. One apneic cycle involves breathing 2-3 breaths of 100% Nitrogen and breath-holding for 20s followed by room air breathing.

LosartanPlacebo

Participants will be instrumented with a sleep monitoring system and will sleep in a normobaric hypoxic chamber with a fraction of inspired oxygen of 13.5%.

LosartanPlacebo

Losartan, 50mg, BID

Also known as: Cozaar
Losartan

Placebo, 50mg, BID

Also known as: microcrystalline cellulose
Placebo

Eligibility Criteria

Age18 Years - 45 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • normotensive
  • forced expiratory volume in 1s : forced vital capacity ratio \> 0.75
  • no medical history of cardiovascular and respiratory disease
  • not taking medications other than oral contraceptives
  • free from sleep apnea
  • body mass index less than 30 kg/m2

You may not qualify if:

  • history of hypertension
  • known impaired renal function
  • liver disease
  • heart failure
  • myocardial infarction
  • coronary artery disease
  • smoked within the past year
  • apnea hypopnea index \> 5 events per hour

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

University of British Columbia

Kelowna, British Columbia, V1V 1V7, Canada

Location

Related Publications (1)

  • Brown CV, Boulet LM, Vermeulen TD, Sands SA, Wilson RJA, Ayas NT, Floras JS, Foster GE. Angiotensin II-Type I Receptor Antagonism Does Not Influence the Chemoreceptor Reflex or Hypoxia-Induced Central Sleep Apnea in Men. Front Neurosci. 2020 Apr 28;14:382. doi: 10.3389/fnins.2020.00382. eCollection 2020.

MeSH Terms

Conditions

Sleep Apnea SyndromesHypoxiaRespiratory AspirationSleep Wake Disorders

Interventions

Losartanmicrocrystalline cellulose

Condition Hierarchy (Ancestors)

ApneaRespiration DisordersRespiratory Tract DiseasesSleep Disorders, IntrinsicDyssomniasNervous System DiseasesSigns and Symptoms, RespiratorySigns and SymptomsPathological Conditions, Signs and SymptomsPathologic ProcessesNeurologic ManifestationsMental Disorders

Intervention Hierarchy (Ancestors)

Biphenyl CompoundsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsImidazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsTetrazoles

Study Officials

  • Glen Foster, PhD

    University of British Columbia

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 4
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Assistant Professor

Study Record Dates

First Submitted

November 1, 2017

First Posted

November 8, 2017

Study Start

January 1, 2018

Primary Completion

August 1, 2019

Study Completion

August 1, 2019

Last Updated

September 4, 2020

Record last verified: 2020-09

Locations