NCT03195452

Brief Summary

Raltegravir (RAL) is a very effective antiretroviral drug with a favorable long term tolerability. RAL offers many advantages such as lack of drug-drug interactions, a good safety profile particularly on lipids, inflammation and bone parameters. Ral can be an very interesting for patient with comorbidities and comedications, intolerance or toxicities with their current ARV treatment. However its current formulation of one tablet of 400mg twice a day coul not suit many patients. A new once-a-day formulation of RAL has been developed, with two tablets of 600 mg QD. Pharmacokinetic study in healthy volunteers has shown that this dosing provides increased RAL exposure compared to the standard formulation of 400 mg given twice a day. The objective of this study is to evaluate the maintain of virologic suppression with raltegravir 600mg 2 tablets qd as part of a triple antiretroviral regimen in virologically controlled patients.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
100

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Nov 2017

Geographic Reach
1 country

17 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 29, 2017

Completed
24 days until next milestone

First Posted

Study publicly available on registry

June 22, 2017

Completed
5 months until next milestone

Study Start

First participant enrolled

November 8, 2017

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 30, 2019

Completed
6 months until next milestone

Study Completion

Last participant's last visit for all outcomes

May 6, 2020

Completed
Last Updated

May 19, 2020

Status Verified

May 1, 2020

Enrollment Period

2 years

First QC Date

May 29, 2017

Last Update Submit

May 15, 2020

Conditions

Keywords

HIVAntiretroviralsRaltegravir

Outcome Measures

Primary Outcomes (1)

  • Number of copie/ml plasma HIV - RNA

    48 weeks

Secondary Outcomes (8)

  • Score evaluation of patient satisfaction

    48 weeks

  • Score evaluation of patient quality of life with PROQOL-HIV questionnaires

    48 weeks

  • Score evaluation of adherence

    48 weeks

  • Number of incidence of Treatment-Emergent Adverse Events

    48 weeks

  • Number of patient who have a viral load < 50 copies/ml

    48 weeks

  • +3 more secondary outcomes

Study Arms (1)

Raltegravir

EXPERIMENTAL

antiretroviral tritherapy: Raltegravir 600 mg tablet orally (2 tablets QD) and 2 Nucleoside/Nucleotide reverse transcriptase inhibitor (NRTI)

Drug: Raltegravir and 2 Nucleoside/Nucleotide reverse transcriptase inhibitor (NRTI)

Interventions

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Adults of both gender ≥ 18 years
  • Signed informed consent form
  • Documented HIV-1 infection
  • Stable antiretroviral therapy for ≥ 6 months consisting of 2 NRTIs (TDF/FTC or ABC/3TC )+ a 3rd agent either as a once or twice daily regimen, unless there is intolerance requiring change of therapy. In this situation of intolerance, patient with less than 6 months of current antiretroviral therapy will be allowed in the study.
  • As soon as TAF/FTC will be available in France, patients receiving TAF/FTC + 3rd agent could be enrolled.
  • Switch of TDF/FTC to TAF/FTC will be authorized as long as the change has occurred for more than 3 months prior to the screening visit. Such switch will be also allowed during the study, and, unless urgently needed, after the W24 visit.
  • Patients on stable raltegravir 400 mg 1 tablet twice daily plus 2 NRTI can be enrolled; number of these patients will be limited to 33% of the total cohort.
  • Indication to current change antiretroviral therapy for at least one of the following reasons :
  • Intolerance or prevention of toxicity
  • Presence of a comorbid condition justifying change of the 3rd agent
  • Management of drug-drug-interaction
  • Patient's request, including switch to simplify or to improve convenience
  • No prior virological failure on integrase-containing antiretroviral therapy or NNRTI-containing antiretroviral therapy or NRTI only-therapy
  • HIV-1 RNA \< 50 c/mL for ≥ 6 months. However, a single HIV-1 RNA ≥ 50 copies/mL and \< 200 copies/mL with a subsequent HIV-1 RNA \< 50 c/mL in the past 6 months is allowed.
  • AST and ALT \< 5 times the upper limit of normal
  • +5 more criteria

You may not qualify if:

  • HIV-2 co-infection
  • Concomitant treatments contra-indicated with raltegravir
  • Patients receiving raltegravir 400mg, 2 tablets in one daily intake
  • Patients with prior virological failure on NRTI+PI/r based regimen can be enrolled as long as historical plasma genotype and/or screening DNA genotype demonstrate absence of resistance or possible resistance to any drug. Subjects with previous failure to any other antiretroviral regimen cannot be enrolled.
  • Presence of possible resistance or resistance to any nucleoside reverse transcriptase inhibitor or integrase inhibitor on a historical plasma genotype.
  • Presence of possible resistance or resistance to any non- nucleoside reverse transcriptase inhibitor on a historical plasma genotype, with the exception of polymorphic mutations E138A/G/K/Q/R/S and V179D in patients naïve to NNRTI.
  • Presence of resistance to any PI on a historical plasma genotype
  • For HCV co-infected patients, if specific treatment for hepatitis is required during the trial duration, such HCV therapy should be compatible with the ARV combination and only started after the W24 visit.
  • HBV infection, in the absence of treatment with TDF or TAF
  • Severe associated diseases requiring specific treatment, such as curative treatment of acute opportunistic infection
  • Treatment with interferon, interleukin or any immunotherapeutic agent or chemotherapy
  • Cancer diagnosis in the past 3 years with the exception of Kaposi sarcoma
  • Any condition which might compromise the safety of treatment and/or patient's adherence to trial procedures
  • Person under guardianship, trusteeship or deprived of freedom by a judicial or administrative decision
  • Difficulty in terms of follow-up (vacation, job transfer, geographical distance, lack of motivation)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (17)

CHU De Bordeaux

Bordeaux, France

Location

CH de la Roche Sur Yon

La Roche-sur-Yon, France

Location

CH du Mans

Le Mans, France

Location

CHU de Lyon

Lyon, France

Location

CHRU de Montpellier

Montpellier, France

Location

CHU of NANTES

Nantes, France

Location

CHU de Nice

Nice, France

Location

CHR orléans

Orléans, France

Location

CHU de Bichat

Paris, France

Location

CHu hotel dieu

Paris, France

Location

CHU la pitié

Paris, France

Location

Hopital Avicenne

Paris, France

Location

Hopital Necker

Paris, France

Location

Hopital St Louis

Paris, France

Location

CHU de Reims

Reims, France

Location

CH de Tourcoing

Tourcoing, France

Location

CHRU de Tours

Tours, France

Location

Related Publications (1)

  • Hall N, Allavena C, Katlama C, Jobert A, Molina JM, Cua E, Bani-Sadr F, Hocqueloux L, Duvivier C, Merrien D, Hikombo H, Andre-Garnier E, Gaultier A, Raffi F; QDISS Study Group. Raltegravir 1200 mg once daily as maintenance therapy in virologically suppressed HIV-1 infected adults: QDISS open-label trial. AIDS Res Ther. 2022 Jan 15;19(1):4. doi: 10.1186/s12981-022-00428-5.

MeSH Terms

Conditions

Acquired Immunodeficiency Syndrome

Interventions

Raltegravir Potassium

Condition Hierarchy (Ancestors)

HIV InfectionsBlood-Borne InfectionsCommunicable DiseasesInfectionsSexually Transmitted Diseases, ViralSexually Transmitted DiseasesLentivirus InfectionsRetroviridae InfectionsRNA Virus InfectionsVirus DiseasesSlow Virus DiseasesGenital DiseasesUrogenital DiseasesImmunologic Deficiency SyndromesImmune System Diseases

Intervention Hierarchy (Ancestors)

PyrrolidinonesPyrrolidinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NA
Masking
NONE
Masking Details
Open label
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
OTHER
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 29, 2017

First Posted

June 22, 2017

Study Start

November 8, 2017

Primary Completion

October 30, 2019

Study Completion

May 6, 2020

Last Updated

May 19, 2020

Record last verified: 2020-05

Locations