NCT02722304

Brief Summary

The purpose of this study is to conduct a pilot study to evaluate the safety and efficacy of weekly administration of Alpha1-Proteinase Inhibitor (A1PI) augmentation therapy in subjects with A1PI deficiency and emphysema/ chronic obstructive pulmonary disease (COPD).

Trial Health

60
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
7

participants targeted

Target at below P25 for phase_3 chronic-obstructive-pulmonary-disease

Timeline
Completed

Started Nov 2016

Typical duration for phase_3 chronic-obstructive-pulmonary-disease

Geographic Reach
3 countries

17 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 23, 2016

Completed
7 days until next milestone

First Posted

Study publicly available on registry

March 30, 2016

Completed
7 months until next milestone

Study Start

First participant enrolled

November 2, 2016

Completed
1.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 14, 2018

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 14, 2018

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

October 8, 2019

Completed
Last Updated

May 13, 2021

Status Verified

April 1, 2021

Enrollment Period

1.9 years

First QC Date

March 23, 2016

Results QC Date

September 18, 2019

Last Update Submit

April 17, 2021

Conditions

Outcome Measures

Primary Outcomes (1)

  • Rate of Change in Lung Density Based on Group 1 (ARALAST NP) Versus Placebo, Group 3 and Group 4 (GLASSIA) Versus Placebo

    Rate of change in lung density was assessed by computed tomography (CT) densitometry. Computed Tomography (CT) scans was used to measure lung density as a quantitative assessment of emphysema progression and treatment efficacy at each of the study visits. CT lung density at the 15th percentile (PD15) is the threshold below which 15% of the voxels have lower densities, and was used as the parameter for estimating the rate of lung density decline. Rate of change in lung density based on Group 1 (ARALAST NP) versus Placebo, Group 3 and Group 4 (GLASSIA) versus Placebo were reported. The safety analysis set used for all the efficacy parameter assessment.

    Baseline, Early termination of the study (approximately 22 months)

Secondary Outcomes (10)

  • Rate of Change in Lung Density for Each Treatment Group

    Baseline, Early termination of the study (approximately 22 months)

  • Mean Steady State Trough Concentration of Antigenic and Functional Alpha1-Proteinase Inhibitor (A1PI) for ARALAST NP and GLASSIA at Each Dose Level

    Baseline, Early termination of the study (approximately 22 months)

  • Number of Events With Related and Unrelated Serious and Non-Serious Treatment Emergent Adverse Event (TEAE)

    From start of study treatment up to early termination of the study (approximately 22 months)

  • Percentage of Participants With Related and Unrelated Serious and Non-Serious Treatment Emergent Adverse Events (TEAE's)

    From start of study treatment up to early termination of the study (approximately 22 months)

  • Number of Events With Temporally Related Serious and Non-Serious Treatment Emergent Adverse Events (AEs)

    From start of study treatment up to early termination of the study (approximately 22 months)

  • +5 more secondary outcomes

Study Arms (5)

ARALAST NP 60 mg/kg

EXPERIMENTAL

60 mg/kg body weight/week

Biological: ARALAST NP 60 mg/kg

ARALAST NP 120 mg/kg

EXPERIMENTAL

120 mg/kg body weight/week

Biological: ARALAST NP 120 mg/kg

GLASSIA 60 mg/kg

EXPERIMENTAL

60 mg/kg body weight/week

Biological: GLASSIA 60 mg/kg

GLASSIA 120 mg/kg

EXPERIMENTAL

120 mg/kg body weight/week

Biological: GLASSIA 120 mg/kg

Placebo

PLACEBO COMPARATOR

Human Albumin 2%

Biological: Human Albumin 2%

Interventions

ARALAST NP is an Alpha1-Proteinase Inhibitor (A1PI) augmentation therapy

Also known as: Alpha1-Proteinase Inhibitor (Human), A1PI, Alpha1-Proteinase Inhibitor
ARALAST NP 60 mg/kg

ARALAST NP is an Alpha1-Proteinase Inhibitor (A1PI) augmentation therapy

Also known as: Alpha1-Proteinase Inhibitor, Alpha1-Proteinase Inhibitor (Human), A1PI
ARALAST NP 120 mg/kg

GLASSIA is an Alpha1-Proteinase Inhibitor (A1PI) augmentation therapy

Also known as: Alpha1-Proteinase Inhibitor (Human), A1PI, Alpha1-Proteinase Inhibitor
GLASSIA 60 mg/kg

GLASSIA is an Alpha1-Proteinase Inhibitor (A1PI) augmentation therapy

Also known as: Alpha1-Proteinase Inhibitor, Alpha1-Proteinase Inhibitor (Human), A1PI
GLASSIA 120 mg/kg

Human albumin 2% (by appropriate dilution with normal saline solution)

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • ≥18 years of age at the time of screening
  • Participant has documented A1PI genotype of Pi\*Z/Z, Pi\*Z/Null, Pi\*Malton/Z, Pi\*Null/Null, or other rare genotypes (except PI\*MS, PI\*MZ, or PI\*SZ).
  • Clinically evident mild-moderate chronic obstructive pulmonary disease (COPD) (according to GOLD criteria for diagnosis) at the time of screening.
  • If the participant is treated with any respiratory medications including inhaled bronchodilators, inhaled corticosteroids, or systemic corticosteroids (e.g. prednisone ≤ 10 mg/day or its equivalent), the doses of the participant's medications have remained stable for at least 28 days prior to screening.
  • No clinically significant abnormalities (other than emphysema, bronchitis or bronchiectasis) detected via a chest computed tomography (CT) or chest X-ray at the time of screening.
  • If female of childbearing potential, participant must have a negative pregnancy test at screening and agree to employ adequate birth control measures for the duration of the study.
  • Participant is willing and able to comply with the requirements of the protocol.

You may not qualify if:

  • Known ongoing or history of clinically significant pulmonary impairment other than emphysema/ COPD.
  • The participant is experiencing lower respiratory infection (LRTI)/acute pulmonary exacerbation (APE) at the time of enrollment (signing Informed consent form (ICF)). Participant may be rescreened after both clinical resolution of LRTI/APE and having also remained stable for at least 4 weeks after the end of LRTI/APE).
  • Known ongoing or history of cor pulmonale.
  • Known resting partial pressure of carbon dioxide (PaCO2) levels of \> 45 mmHg.
  • Clinically significant congestive heart failure with New York Heart Association (NYHA) Class III/IV symptoms.
  • The participant has received an organ transplant, has undergone major lung surgery, or is currently on a transplant list.
  • Known history of ongoing malignancy (other than adequately treated basal cell or squamous cell carcinoma of the skin or carcinoma in situ of the cervix).
  • Smoker or participant that has ceased smoking for less than one year prior to screening whose levels of cotinine are outside of the normal range of a nonsmoker.
  • All participants must agree to refrain from smoking throughout the course of the study.
  • The participant is receiving long-term therapy (\> 28 days) of parenteral corticosteroids or oral corticosteroids at doses greater than 10 mg/day of prednisone or its equivalent).
  • The participant is receiving long-term round-the-clock oxygen supplementation (other than temporary for acute COPD exacerbation, or supplemental oxygen (O2) with continuous positive airway pressure \[CPAP\], or bi-level positive airway pressure \[BiPAP\] during the day).
  • Participant has contraindications for CT (e.g. body weight and/or body size exceeding the weight and gantry size limits specified by the manufacturer of the CT scanner, inability to lie flat in the CT scanner, claustrophobia, metal prosthesis or pacemaker in the chest wall or upper extremity that would impact lung density assessment).
  • Participant is unwilling or unable to modify bronchodilator medications for 6 hours for short acting β2 agonists, 24 hours for long-acting β2 agonists, and 48 hours for long acting anticholinergics prior to the scheduled quantitative CT scan.
  • Known severe immunoglobulin A (IgA) deficiency (ie, IgA level \< 8 mg/dL at screening).
  • Known history of hypersensitivity following infusions of human blood or blood components (eg, human immunoglobulins or human albumin).
  • +5 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (17)

Phoenix Medical Research Institute, LLC

Peoria, Arizona, 85381, United States

Location

Newport Native MD, Inc

Newport Beach, California, 92663, United States

Location

Pulmonary Disease Specialists, P.A., / PDS Research

Kissimmee, Florida, 34741, United States

Location

L&C Professional Medical Research Institute

Miami, Florida, 33144, United States

Location

Loyola University Health System

Maywood, Illinois, 60153, United States

Location

Indiana University Health

Indianapolis, Indiana, 46202, United States

Location

La Porte County Institute for Clinical Research, Inc.

Michigan City, Indiana, 46360, United States

Location

Pulmonary Health Physicians

Fayetteville, New York, 13066, United States

Location

Clinical Research of Gastonia

Gastonia, North Carolina, 28054, United States

Location

Southeastern Research Center LLC

Winston-Salem, North Carolina, 27103, United States

Location

Metroplex Pulmonary and Sleep Center

Allen, Texas, 75013, United States

Location

Houston Pulmonary and Sleep Associates

Houston, Texas, 77065, United States

Location

Element Research Group

San Antonio, Texas, 78258, United States

Location

Renovatio Clinical-Respiratory & Sleep Disorders Specialists

The Woodlands, Texas, 77005, United States

Location

St Vincent's Hospital Melbourne

Fitzroy, Victoria, 34741, Australia

Location

LHSC - Victoria Hospital

London, Ontario, N6A 5W9, Canada

Location

Inspiration Research Limited

Toronto, Ontario, M5T 3A9, Canada

Location

MeSH Terms

Conditions

Pulmonary Disease, Chronic Obstructivealpha 1-Antitrypsin Deficiency

Interventions

alpha 1-Antitrypsin

Condition Hierarchy (Ancestors)

Lung Diseases, ObstructiveLung DiseasesRespiratory Tract DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and SymptomsLiver DiseasesDigestive System DiseasesGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and AbnormalitiesSubcutaneous EmphysemaEmphysema

Intervention Hierarchy (Ancestors)

GlycoproteinsGlycoconjugatesCarbohydratesSerpinsPeptidesAmino Acids, Peptides, and ProteinsAcute-Phase ProteinsBlood ProteinsProteinsAlpha-GlobulinsSerum GlobulinsGlobulins

Limitations and Caveats

The Data Monitoring Committee (DMC) reviewed the available efficacy and safety data and unanimously recommended to terminate the study. The decision was based on the very low number of enrollees, and the slow rate of participant enrollment.

Results Point of Contact

Title
Study Director
Organization
Shire

Study Officials

  • Study Director

    Takeda

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 23, 2016

First Posted

March 30, 2016

Study Start

November 2, 2016

Primary Completion

September 14, 2018

Study Completion

September 14, 2018

Last Updated

May 13, 2021

Results First Posted

October 8, 2019

Record last verified: 2021-04

Data Sharing

IPD Sharing
Will not share

De-identified individual participant data from this particular study will not be shared as there is a reasonable likelihood that individual patients could be re-identified (due to the limited number of study participants).

Locations