NCT02526524

Brief Summary

The purpose of the study is to compare the glycemic effects of delayed-release metformin (Met DR) to placebo in subjects with type 2 diabetes mellitus (T2DM) over 16 weeks. The study is designed to evaluate several doses of Met DR (600 to 1500 mg once daily in the morning \[qAM\]) compared to placebo. A single-blind reference treatment of 2000 mg metformin immediate-release (Met IR) per day administered as equal divided doses (1000 mg Met IR BID) will also be included.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
571

participants targeted

Target at P75+ for phase_2 type-2-diabetes-mellitus

Timeline
Completed

Started Sep 2015

Geographic Reach
2 countries

137 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

August 16, 2015

Completed
2 days until next milestone

First Posted

Study publicly available on registry

August 18, 2015

Completed
14 days until next milestone

Study Start

First participant enrolled

September 1, 2015

Completed
1 year until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 1, 2016

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2016

Completed
1.7 years until next milestone

Results Posted

Study results publicly available

April 27, 2018

Completed
Last Updated

April 27, 2018

Status Verified

March 1, 2018

Enrollment Period

1 year

First QC Date

August 16, 2015

Results QC Date

March 27, 2018

Last Update Submit

March 27, 2018

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change in HbA1c (%) at 16 Weeks

    Baseline and 16 weeks after the first dose of study medication

Study Arms (7)

600 mg Met DR qAM

EXPERIMENTAL

600 mg metformin delayed-release once daily in the morning

Drug: Met DR

900 mg Met DR qAM

EXPERIMENTAL

900 mg metformin delayed-release once daily in the morning

Drug: Met DR

1200 mg Met DR qAM

EXPERIMENTAL

1200 mg metformin delayed-release once daily in the morning

Drug: Met DR

1500 mg Met DR qAM

EXPERIMENTAL

1500 mg metformin delayed-release once daily in the morning

Drug: Met DR

Placebo-1

PLACEBO COMPARATOR

placebo match for 600 and 1200 mg Met DR qAM treatment groups

Drug: Placebo

Placebo-2

PLACEBO COMPARATOR

placebo match for 900 and 1500 mg Met DR qAM treatment groups

Drug: Placebo

2000 mg Met IR

ACTIVE COMPARATOR

1000 mg metformin immediate-release twice daily

Drug: Met IR

Interventions

Met DRDRUG

metformin delayed-release tablets

1200 mg Met DR qAM1500 mg Met DR qAM600 mg Met DR qAM900 mg Met DR qAM
Met IRDRUG

metformin immediate-release tablets

2000 mg Met IR
Placebo-1Placebo-2

Eligibility Criteria

Age25 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Is at least 25 years old at Visit 1 (Screening).
  • Is male, or is female and meets all of the following criteria:
  • Not breastfeeding
  • Negative pregnancy test result at Visit 1 (not applicable to post-menopausal or surgically sterile females)
  • Surgically sterile, postmenopausal, or if of childbearing potential, must practice and be willing to continue to practice appropriate birth control during the entire duration of the study.
  • Body mass index (BMI) 20.0 to 45.0 kg/m² (inclusive) at Visit 1 (Screening).
  • Has a physical examination with no clinically significant abnormalities as judged by the investigator.
  • Has T2DM and an HbA1c of 7.5% to 10.5%, inclusive, at Visit 1.
  • Has an estimated glomerular filtration rate (eGFR) value of ≥60 mL/min/1.73 m² based on the Modification of Diet in Renal Disease (MDRD) equation.
  • Either is not treated with or has been on a stable treatment regimen with any of the following medications for a minimum of 3 months prior to Visit 1:
  • Thiazolidinedione, sulfonylurea, dipeptidyl peptidase-4 inhibitors, and alpha-glucosidase inhibitors
  • Hormone replacement therapy (female subjects) and testosterone (male subjects)
  • Oral contraceptives (female subjects)
  • Antihypertensive agents
  • Lipid-lowering agents
  • +3 more criteria

You may not qualify if:

  • Has a clinically significant medical condition as judged by the investigator that could potentially affect study participation and/or personal well-being, including but not limited to the following conditions:
  • Hepatic disease
  • Gastrointestinal disease
  • Endocrine disorder (T2DM is allowed)
  • Cardiovascular disease
  • Central nervous system diseases
  • Psychiatric or neurological disorders
  • Organ transplantation
  • Chronic or acute infection
  • Orthostatic hypotension, fainting spells or blackouts
  • Allergy or hypersensitivity.
  • A history of diabetic ketoacidosis or hyperosmolar non-ketotic hyperglycemia within the past year.
  • Prior major surgery of any kind within 6 months of Visit 1.
  • A history of \>3% weight change within 3 months of Visit 1.
  • A clinical laboratory test (clinical chemistry, hematology, or urinalysis) abnormality, other than that related to T2DM, judged by the investigator to be clinically significant at Visit 1.
  • +17 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (137)

Pinnacle Research Group, LLC

Anniston, Alabama, 36207, United States

Location

Central Alabama Research

Birmingham, Alabama, 35209, United States

Location

Achieve Clinical Research, LLC

Birmingham, Alabama, 35216, United States

Location

University of Alabama at Birmingham

Birmingham, Alabama, 35294, United States

Location

Terence T. Hart, MD

Tuscumbia, Alabama, 35674, United States

Location

Radiant Research - Phoenix

Chandler, Arizona, 85224, United States

Location

Arrowhead Health Centers

Glendale, Arizona, 85306, United States

Location

Holland Center for Family Health, LTD

Peoria, Arizona, 85381, United States

Location

Elite Clinical Studies

Phoenix, Arizona, 85018, United States

Location

Thunderbird Internal Medicine - Indian School Rd.

Phoenix, Arizona, 85037, United States

Location

Clinical Research Institute of Arizona, LLC

Surprise, Arizona, 85374, United States

Location

Summit Clinical Trials Center

Fayetteville, Arkansas, 72703, United States

Location

Searcy Medical Center

Searcy, Arkansas, 72143, United States

Location

Advanced Metabolic Care & Research Institute (AMCR)

Escondido, California, 92025, United States

Location

MD Studies, Inc.

Fountain Valley, California, 92708, United States

Location

National Research Institute

Huntington Park, California, 90255, United States

Location

Scripps Whittier Diabetes Institute

La Jolla, California, 92037, United States

Location

Clinical Trials Research

Lincoln, California, 95648, United States

Location

Collaborative Neuroscience Network, LLC

Long Beach, California, 90806, United States

Location

National Research Institute

Los Angeles, California, 90057, United States

Location

Catalina Research Institute

Montclair, California, 91763, United States

Location

SRSD, Inc. dba Synergy San Diego

National City, California, 91950, United States

Location

Providence Clinical Research

North Hollywood, California, 91606, United States

Location

Pacific Research Partners, LLC

Oakland, California, 94607, United States

Location

SDS Clinical Trials, Inc.

Orange, California, 92868, United States

Location

Center for Clinical Trials of Sacramento

Sacramento, California, 95823, United States

Location

Center for Clinical Trials of Scaramento

Sacramento, California, 95823, United States

Location

Superior Research LLC

Sacramento, California, 95825, United States

Location

Syrentis Clinical Research (formerly Research Across America)

Santa Ana, California, 92705, United States

Location

Encompass Clinical Research

Spring Valley, California, 91978, United States

Location

Clinical Trial Investigators

Tustin, California, 92780, United States

Location

Infosphere Clinical Research

Van Nuys, California, 91405, United States

Location

Colorado Springs Health Partners

Colorado Springs, Colorado, 80906, United States

Location

Creekside Endocrine Associates

Denver, Colorado, 80209, United States

Location

Meridien Research - Brooksville

Brooksville, Florida, 34601, United States

Location

ALL Medical Research, LLC

Cooper City, Florida, 33024, United States

Location

Neostart Corporation dba AGA Clinical Trials

Hialeah, Florida, 33012, United States

Location

Care Partners Clinical Research

Jacksonville, Florida, 32277, United States

Location

Health Awareness, Inc.

Jupiter, Florida, 33458, United States

Location

Family Health Care Clinical Studies

Kissimmee, Florida, 34741, United States

Location

Clinical Research of Central Florida-Lakeland

Lakeland, Florida, 33810, United States

Location

Clinical Pharmacology of Miami, Inc.

Miami, Florida, 33014, United States

Location

Tellus Clinical Research, Inc.

Miami, Florida, 33173, United States

Location

Internal Research Associates LLC - Breton

Miami, Florida, 33183, United States

Location

Clinical Neuroscience Solutions, Inc. Healthcare Orlando

Orlando, Florida, 32801, United States

Location

Ormond Medical Arts Pharmaceutical Research Center

Ormond Beach, Florida, 32174, United States

Location

Private Practice - Andres Patron, DO

Pembroke Pines, Florida, 33026, United States

Location

Progressive Medical Research

Port Orange, Florida, 32127, United States

Location

Meridien Reserach - St. Petersburg

St. Petersburg, Florida, 33709, United States

Location

Clinical Reserch Trials of Florida

Tampa, Florida, 33607, United States

Location

Meridien Research - Tampa

Tampa, Florida, 33634, United States

Location

Metabolic Research Institute, Inc.

West Palm Beach, Florida, 33401, United States

Location

Biofortis, Inc.

Addison, Illinois, 60101, United States

Location

AMR Sakeena Research

Aurora, Illinois, 60506, United States

Location

Cedar-Crosse Research Center

Chicago, Illinois, 60607, United States

Location

Evanston Premier Healthcare Research LLC

Evanston, Illinois, 60201, United States

Location

Buynak Clinical Research, PC

Valparaiso, Indiana, 46383, United States

Location

The Iowa Clinic; Cardiovascular Services

West Des Moines, Iowa, 50266, United States

Location

Heartland Research Associates, LLC - Augusta

Augusta, Kansas, 67010, United States

Location

Cotton-O'Neil Clinical Research Center

Topeka, Kansas, 66606, United States

Location

Otrimed

Edgewood, Kentucky, 41017, United States

Location

Kentucky Diabetes Endocrinology Center

Lexington, Kentucky, 40503, United States

Location

Louisville Metabolic and Atherosclerosis Research Center (L-MARC)

Louisville, Kentucky, 40213, United States

Location

Four Rivers Clinical Research

Paducah, Kentucky, 42003, United States

Location

Avant Research Associates

Crowley, Louisiana, 70526, United States

Location

Centex Studies, Inc. - lake Charles

Lake Charles, Louisiana, 70601, United States

Location

Columbia Medical Practice

Columbia, Maryland, 21045, United States

Location

Medstar Health Research Institute

Hyattsville, Maryland, 20782, United States

Location

MD Medical Research

Oxon Hill, Maryland, 20745, United States

Location

Beacon Clinical Research

Quincy, Massachusetts, 02169, United States

Location

Radiant Research - Edina

Edina, Minnesota, 55435, United States

Location

Planters Clinic

Port Gibson, Mississippi, 39150, United States

Location

Mercury Street Medical Group, PLLC

Butte, Montana, 59701, United States

Location

Quality Clinical Research, Inc.

Omaha, Nebraska, 68114, United States

Location

Heartland Clinical Research

Omaha, Nebraska, 68134, United States

Location

Alliance Against Diabetes

Las Vegas, Nevada, 89101, United States

Location

AB Clinical Trials

Las Vegas, Nevada, 89119, United States

Location

Palm Medical Research

Las Vegas, Nevada, 89128, United States

Location

Ingham Neuroscience Group, LLC

Las Vegas, Nevada, 89146, United States

Location

Comprehensive Clinical Research

Berlin, New Jersey, 08009, United States

Location

Albuquerque Clinical Trials

Albuquerque, New Mexico, 87102, United States

Location

Albuquerque Neuroscience, Inc.

Albuquerque, New Mexico, 87109, United States

Location

NY Scientific

Brooklyn, New York, 11235, United States

Location

Long Island Gastrointestinal Research Group

Great Neck, New York, 11023, United States

Location

Mid-Hudson Medical Research, PLLC

Hopewell Junction, New York, 12533, United States

Location

Great Lakes Medical Research

Westfield, New York, 14787, United States

Location

PharmQuest

Greensboro, North Carolina, 27408, United States

Location

Triad Clinical Trials LLC

Greensboro, North Carolina, 27410, United States

Location

PMG Research of Rocky Mount

Rocky Mount, North Carolina, 27804, United States

Location

PMG Research of Salisbury, LLC

Salisbury, North Carolina, 28144, United States

Location

PMG Research of Wilmington, LLC

Wilmington, North Carolina, 28401, United States

Location

Sterling Research Group, Ltd

Cincinnati, Ohio, 45219, United States

Location

Metabolic Atherosclerosis Research Center

Cincinnati, Ohio, 45227, United States

Location

New Horizons Clinical Research

Cincinnati, Ohio, 45242, United States

Location

Urgent Care Specialists, LLC DBA Hometown Urgent Care and Occupational Health

Columbus, Ohio, 43214, United States

Location

Prestige Clinical Research

Franklin, Ohio, 45005, United States

Location

Hometown Urgent Care and Research - Huber Heights

Huber Heights, Ohio, 45424, United States

Location

RAS Health LTD

Marion, Ohio, 43302, United States

Location

Summit Reserach Group, LLC

Stow, Ohio, 44224, United States

Location

COR Clinical Research, LLC

Oklahoma City, Oklahoma, 73103, United States

Location

Willamette Valley Clinical Studies

Eugene, Oregon, 97404, United States

Location

Brandywine Clinical Research

Downingtown, Pennsylvania, 19335, United States

Location

Medical Research South, LLC

Charleston, South Carolina, 29407, United States

Location

Mountain View Clinical Research - Greer

Greer, South Carolina, 29651, United States

Location

PMG of Charleston, LLC

Mt. Pleasant, South Carolina, 29464, United States

Location

Family Medicine of SayeBrook, LLC

Myrtle Beach, South Carolina, 29588, United States

Location

Hillcrest Clinical Research, LLC

Simpsonville, South Carolina, 29681, United States

Location

Palmetto Proactive Healthcare, LLC

Spartanburg, South Carolina, 29301, United States

Location

Spartanburg Medical Research

Spartanburg, South Carolina, 29303, United States

Location

Palmetto Clinical Research

Summerville, South Carolina, 29485, United States

Location

PMG Research of Bristol, LC - State

Bristol, Tennessee, 37620, United States

Location

PMG Research of Knoxville

Knoxville, Tennessee, 37912, United States

Location

Clinical Neuroscience Solutions, Inc. - Memphis

Memphis, Tennessee, 38119, United States

Location

Trinity Clinical Research

Tullahoma, Tennessee, 37388, United States

Location

Central Texas Clinical Research

Austin, Texas, 78705, United States

Location

Trinity Universal Research Associates, Inc.

Carrollton, Texas, 75007, United States

Location

Dallas Diabetes and Endocrine Center

Dallas, Texas, 75230, United States

Location

Research Institute of Dallas

Dallas, Texas, 75231, United States

Location

Galenos Research

Dallas, Texas, 75251, United States

Location

Pioneer Research Solutions, Inc.

Houston, Texas, 77036, United States

Location

Centex Studies, Inc.

Houston, Texas, 77058, United States

Location

Clinical Trial Network - Houston

Houston, Texas, 77074, United States

Location

Juno Research, LLC-Houston

Houston, Texas, 77074, United States

Location

Juno Research, LLC-Katy

Katy, Texas, 77450, United States

Location

Texas Diabetes Institute Research Center

San Antonio, Texas, 78207, United States

Location

Sun Research Institute

San Antonio, Texas, 78215, United States

Location

Victorium Clinical Research

San Antonio, Texas, 78231, United States

Location

Consano Clinical Research

Shavano Park, Texas, 78231, United States

Location

Southwest Health Associates, P.A.

Sugar Land, Texas, 77478, United States

Location

Chrysalis Clinical Research

St. George, Utah, 84790, United States

Location

Burke Internal Medicine & Research

Burke, Virginia, 22015, United States

Location

Manassas Clinical Research Center

Manassas, Virginia, 20110, United States

Location

Clinical Research Partners, LLC

Richmond, Virginia, 23235, United States

Location

Universal Research Group, LLC

Tacoma, Washington, 98405, United States

Location

Puerto Rico Renal and Health Research, Inc.

Carolina, 00987, Puerto Rico

Location

Advanced Medical Concepts

Cidra, 00736, Puerto Rico

Location

Manati Center for Clinical Reserach Doctor's Center Hospital

Manatí, 00674, Puerto Rico

Location

Related Publications (1)

  • Henry RR, Frias JP, Walsh B, Skare S, Hemming J, Burns C, Bicsak TA, Baron A, Fineman M. Improved glycemic control with minimal systemic metformin exposure: Effects of Metformin Delayed-Release (Metformin DR) targeting the lower bowel over 16 weeks in a randomized trial in subjects with type 2 diabetes. PLoS One. 2018 Sep 25;13(9):e0203946. doi: 10.1371/journal.pone.0203946. eCollection 2018.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Results Point of Contact

Title
Chief Scientific Officer
Organization
Elcelyx Therapeutics, Inc

Study Officials

  • Juan P Frias, MD

    National Research Institute - Wilshire

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 16, 2015

First Posted

August 18, 2015

Study Start

September 1, 2015

Primary Completion

September 1, 2016

Study Completion

September 1, 2016

Last Updated

April 27, 2018

Results First Posted

April 27, 2018

Record last verified: 2018-03

Locations