NCT02487433

Brief Summary

This study will evaluate the drug behavior and safety of a single dose of the 22 milligram tofacitinib (CP-690,550) modified-release formulation in 18 healthy volunteers when taken after eating a high fat meal (the effect of food). This will be compared to the drug behavior and safety of a single dose of the 22 milligram tofacitinib (CP-690,550) modified-release formulation when taken after a 10 hour fast.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
18

participants targeted

Target at below P25 for phase_1 healthy

Timeline
Completed

Started Jun 2015

Shorter than P25 for phase_1 healthy

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

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Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 23, 2015

Completed
1 month until next milestone

Study Start

First participant enrolled

June 1, 2015

Completed
1 month until next milestone

First Posted

Study publicly available on registry

July 1, 2015

Completed
Same day until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2015

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2015

Completed
Last Updated

August 19, 2015

Status Verified

August 1, 2015

Enrollment Period

1 month

First QC Date

April 23, 2015

Last Update Submit

August 17, 2015

Conditions

Keywords

food effectpharmacokineticshealthy volunteers

Outcome Measures

Primary Outcomes (3)

  • AUC inf

    Area under the plasma concentration-time profile from time zero to infinity (AUCinf).

    48 hours post dose

  • AUC last

    Area under the plasma concentration-time profile from time zero to time of last identifiable quantitation (AUC last).

    48 hours post dose

  • Cmax

    Maximum observed plasma concentration (Cmax).

    48 hours post dose

Secondary Outcomes (2)

  • Time to Reach Maximum Observed Plasma Concentration (Tmax)

    48 hours post dose

  • Plasma Decay Half-Life (t 1/2)

    48 hours post dose

Study Arms (2)

Tofacitinib MR 22 mg Fed

EXPERIMENTAL

Single dose of tofacitinib MR 22 mg administered under fed conditions

Drug: Tofacitinib MR 22 mg (Fed)

Tofacitinib MR 22 mg Fasted

EXPERIMENTAL

Single dose of tofacitinib MR 22 mg administered under fasted conditions

Drug: Tofacitinib MR 22 mg (Fasted)

Interventions

A single dose of tofacitinib modified release 22 mg tablet after receiving the standard FDA high-fat/high-calorie meal

Tofacitinib MR 22 mg Fed

A single dose of tofacitinib modified release 22 mg tablet after an overnight fast of 10 hours

Tofacitinib MR 22 mg Fasted

Eligibility Criteria

Age18 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy male volunteers and/or healthy female volunteers of non-childbearing potential who are 18 to 55 years of age;
  • Healthy volunteers with no evidence of active or latent or inadequately treated tuberculosis.

You may not qualify if:

  • Evidence or history of clinically significant hematological, renal, endocrine, pulmonary, gastrointestinal, cardiovascular, hepatic, psychiatric, neurologic, or allergic disease;
  • Clinically significant infections within the past 3 months

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Pfizer Clinical Research Unit

Brussels, B-1070, Belgium

Location

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 23, 2015

First Posted

July 1, 2015

Study Start

June 1, 2015

Primary Completion

July 1, 2015

Study Completion

July 1, 2015

Last Updated

August 19, 2015

Record last verified: 2015-08

Locations