NCT02344862

Brief Summary

The purpose of this study is exploratory investigation of safety and efficacy (dose response and optimal dose according to the percent reduction from baseline in serum urate level at the final visit) of FYU-981 administered orally to hyperuricemic patients with and without gout for 8 weeks (dose-escalating initial period: 4 weeks followed by maintenance period: 4 weeks) by the method of randomized (dynamic allocation), placebo-controlled, double-blind, parallel group comparison.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
80

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Jan 2014

Shorter than P25 for phase_2

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

January 1, 2014

Completed
6 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2014

Completed
2 months until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2014

Completed
5 months until next milestone

First Submitted

Initial submission to the registry

January 18, 2015

Completed
8 days until next milestone

First Posted

Study publicly available on registry

January 26, 2015

Completed
Last Updated

January 26, 2015

Status Verified

January 1, 2015

Enrollment Period

6 months

First QC Date

January 18, 2015

Last Update Submit

January 22, 2015

Conditions

Outcome Measures

Primary Outcomes (1)

  • Percent reduction from baseline in serum urate level at the final visit

    8 weeks

Study Arms (4)

FYU-981 High dose

ACTIVE COMPARATOR
Drug: FYU-981 High dose, (Oral daily dosing for 8 weeks)

FYU-981 Middle dose

ACTIVE COMPARATOR
Drug: FYU-981 Middle dose, (Oral daily dosing for 8 weeks)

FYU-981 Low dose

ACTIVE COMPARATOR
Drug: FYU-981 Low dose, (Oral daily dosing for 8 weeks)

Placebo

PLACEBO COMPARATOR
Drug: Placebo, (Oral daily dosing for 8 weeks)

Interventions

Subjects randomized to the FYU-981 High dose arm receive active drug, FYU-981 High dose.

FYU-981 High dose

Subjects randomized to the FYU-981 Middle dose arm receive active drug, FYU-981 Middle dose.

FYU-981 Middle dose

Subjects randomized to the FYU-981 Low dose arm receive active drug, FYU-981 Low dose.

FYU-981 Low dose

Subjects randomized to the placebo arm receive placebo.

Placebo

Eligibility Criteria

Age20 Years - 64 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64)

You may qualify if:

  • Hyperuricemic or gout patients
  • Serum urate level:
  • \>= 7.0mg/dL in patients with history of gout, or \>= 8.0mg/dL in patients with hypertension, diabetes or metabolic syndrome, or \>= 9.0mg/dL

You may not qualify if:

  • Gouty arthritis within two weeks before start of study treatment
  • Secondary hyperuricemia
  • HbA1c: \>= 8.4%
  • Uric acid-overproduction type in the classification of hyperuricemia
  • History of, clinically significant cardiac, hematologic and hepatic disease
  • Kidney calculi or clinically significant urinary calculi
  • eGFR: \< 60mL/min/1.73m\^2
  • Systolic blood pressure: \>= 180 mmHg
  • Diastolic blood pressure: \>= 110 mmHg

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Japan

Tokyo, Japan

Location

Related Publications (1)

  • Hosoya T, Sano T, Sasaki T, Fushimi M, Ohashi T. Clinical efficacy and safety of dotinurad, a novel selective urate reabsorption inhibitor, in Japanese hyperuricemic patients with or without gout: an exploratory, randomized, multicenter, double-blind, placebo-controlled, parallel-group early phase 2 study. Clin Exp Nephrol. 2020 Mar;24(Suppl 1):44-52. doi: 10.1007/s10157-019-01802-w. Epub 2019 Nov 21.

MeSH Terms

Conditions

Hyperuricemia

Interventions

dotinurad

Condition Hierarchy (Ancestors)

Pathologic ProcessesPathological Conditions, Signs and Symptoms

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 18, 2015

First Posted

January 26, 2015

Study Start

January 1, 2014

Primary Completion

July 1, 2014

Study Completion

September 1, 2014

Last Updated

January 26, 2015

Record last verified: 2015-01

Locations