NCT02332174

Brief Summary

The purpose of this study was to determine the pharmacokinetic (PK) and safety profile of single and multiple doses of rufinamide. The effects of food and sex on the PK properties of rufinamide in these Chinese volunteers were also evaluated.

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
40

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Mar 2014

Shorter than P25 for phase_1

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2014

Completed
3 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2014

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2014

Completed
7 months until next milestone

First Submitted

Initial submission to the registry

January 3, 2015

Completed
3 days until next milestone

First Posted

Study publicly available on registry

January 6, 2015

Completed
Last Updated

January 6, 2015

Status Verified

January 1, 2015

Enrollment Period

3 months

First QC Date

January 3, 2015

Last Update Submit

January 3, 2015

Conditions

Keywords

pharmacokineticsfood effectsex effecttolerability

Outcome Measures

Primary Outcomes (1)

  • AUC

    the area under the concentration-time curve

    three days

Study Arms (4)

200-mg group

EXPERIMENTAL

Ten healthy subjects were administered a single oral dose of 200 mg rufinamide tablets in fasted and fed state at day 1 and then received repeated oral doses of rufinamide (200 mg) once daily for 6 days.

Drug: rufinamide

400-mg group

EXPERIMENTAL

Ten healthy subjects were administered a single oral dose of 400 mg rufinamide tablets in fasted state.

Drug: rufinamide

800-mg group

EXPERIMENTAL

Ten healthy subjects were administered a single oral dose of 800 mg rufinamide tablets in fasted state.

Drug: rufinamide

1200-mg group

EXPERIMENTAL

Ten healthy subjects were administered a single oral dose of 1200 mg rufinamide tablets in fasted state.

Drug: rufinamide

Interventions

comparison of different doses, sex and medication conditions

Also known as: 106308-44-5
1200-mg group200-mg group400-mg group800-mg group

Eligibility Criteria

Age18 Years - 40 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • body mass index between19 and 24 kg/m2
  • negative for HIV and hepatitis B
  • had no clinicallyimportant findings on health tests
  • thorax radiography and ECG with no abnormalities
  • normal blood pressure values
  • heart rate

You may not qualify if:

  • any drug treatment within 2 weeks before starting the study
  • participation in another clinical study within the previous 3 months
  • alcoholism and smoking
  • pregnancy
  • breast-feeding
  • hypocalcemia
  • blood donation or participation in other clinical trials within 3 months before enrollment in the study
  • sitting blood pressure \<80/50 mm Hg or \>140/100 mm Hg
  • A ventricular rate \<60 beats/min or \>100 beats/min at rest

Contact the study team to confirm eligibility.

Sponsors & Collaborators

MeSH Terms

Conditions

Seizures

Interventions

rufinamide

Condition Hierarchy (Ancestors)

Neurologic ManifestationsNervous System DiseasesSigns and SymptomsPathological Conditions, Signs and Symptoms

Study Officials

  • Weiyong Li, PhD

    Tongji Medical College, Huazhong University of Science and Technology

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
PARALLEL
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Institute of Clinical Pharmacy

Study Record Dates

First Submitted

January 3, 2015

First Posted

January 6, 2015

Study Start

March 1, 2014

Primary Completion

June 1, 2014

Study Completion

June 1, 2014

Last Updated

January 6, 2015

Record last verified: 2015-01