NCT02064426

Brief Summary

Evaluate efficacy and safety up to 36 months of titrated dose treatment with BAY85-3934 versus epoetin alfa/beta. Titration will be based on the subject's hemoglobin (Hb) response and tolerability of the prior dose. Planned doses include 15, 25, 50, 75, 100,and 150 mg once daily.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
88

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Mar 2014

Geographic Reach
2 countries

26 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

February 14, 2014

Completed
3 days until next milestone

First Posted

Study publicly available on registry

February 17, 2014

Completed
24 days until next milestone

Study Start

First participant enrolled

March 13, 2014

Completed
2.6 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 19, 2016

Completed
28 days until next milestone

Study Completion

Last participant's last visit for all outcomes

November 16, 2016

Completed
Last Updated

September 20, 2019

Status Verified

September 1, 2019

Enrollment Period

2.6 years

First QC Date

February 14, 2014

Last Update Submit

September 17, 2019

Conditions

Keywords

Anemia of CKD on dialysis

Outcome Measures

Primary Outcomes (2)

  • Change in local laboratory hemoglobin level from baseline

    Baseline up to 36 months

  • Number of participants with serious adverse events as a measure of safety and tolerability

    Up to 36 months

Secondary Outcomes (12)

  • Maintenance in hemoglobin target range (10.0 to 11.0 g/dL)

    Up to 36 months

  • Maintenance in hemoglobin target range (9.5 to 11.5 g/dL)

    Up to 36 months

  • Duration of treatment exposure

    Up to 36 months

  • Number of subjects requiring titration of dose

    Up to 36 months

  • Change of reticulocyte count from baseline of this study

    Baseline up to 36 months

  • +7 more secondary outcomes

Study Arms (2)

Molidustat (BAY85-3934)

EXPERIMENTAL
Drug: Molidustat (BAY85-3934)

Epoetin alfa/beta

ACTIVE COMPARATOR
Biological: Epoetin alfa/beta

Interventions

Subjects will continue with the same treatment they were receiving in the parent study (16208). BAY85-3934 will be administered daily as oral tablets. Dose assessments will be made every 4 (± 1) weeks. At the scheduled visits, the dose may be titrated on an individualized basis taking into account the subject's Hb response and the tolerability of the previous dose. Total treatment time is up to 36 months. Planned doses include 15, 25, 50, 75, 100, and 150 mg once daily.

Molidustat (BAY85-3934)

Subjects will continue with the same treatment they were receiving in the parent study (16208). Epoetin alfa / beta will be administered as intravenous (IV) or subcutaneous (SC) injections per individual subject regimen according to the local label. Dose assessments will be made every 4 (± 1) weeks. At the scheduled visits,dose may be titrated on an individualized basis taking into account the subject's Hb response and the tolerability of the previous dose.Total treatment time is up to 36 months.

Epoetin alfa/beta

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Eligible male or female subjects were previously enrolled in Study 16208, have a diagnosis of anemia associated with CKD, and are on hemodialysis.
  • Men who agree to use adequate contraception when sexually active or women without childbearing potential
  • Participation and completion of treatment in Study 16208; subjects must have received 16 weeks of study medication and completed the end of treatment visit (Day 113) in the parent study
  • Mean Hb concentration of 9.5 to 11.5 g/dL, inclusive, during the evaluation period (i.e., the last 4 weeks of the parent study) when the subject completed 16 weeks of treatment with BAY85-3934, epoetin alfa, or epoetin beta in Study 16208

You may not qualify if:

  • A scheduled kidney transplant or any other organ transplant within the next 6 months (being on a waiting list does not exclude the subject)
  • Subjects treated with immunosuppressive therapy and the breast cancer resistant protein (BCRP) substrates, irinotecan, topotecan, methotrexate, imatinib, and lapatinib
  • Sustained, poorly controlled arterial hypertension or hypotension at baseline, defined as mean BP ≥ 180/110 mmHg or systolic BP \< 95 mmHg, respectively
  • Severe rhythm or conduction disorder (e.g., HR \< 50 or \> 110 bpm, atrial fibrillation or flutter, prolonged QT \> 500 msec, second or third degree atrioventricular \[AV\] block)
  • New York Heart Association Class III or IV congestive heart failure
  • Severe hepatic insufficiency (defined as alanine aminotransferase \[ALT\], aspartate aminotransferase \[AST\], or gamma-glutamyl transferase \> 3 x the upper limit of norma \[ULN\], total bilirubin \> 2 mg/dL, or Child-Pugh B or C) or active hepatitis in the investigator's opinion
  • An ongoing SAE from Study 16208 that is assessed as related to study drug
  • Alcohol or drug abuse

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (26)

Unknown Facility

Azusa, California, 91702, United States

Location

Unknown Facility

Long Beach, California, 90813, United States

Location

Unknown Facility

Lynwood, California, 90262, United States

Location

Unknown Facility

Northridge, California, 91324, United States

Location

Unknown Facility

San Dimas, California, 91773, United States

Location

Unknown Facility

Whittier, California, 90602, United States

Location

Unknown Facility

Whittier, California, 90606, United States

Location

Unknown Facility

New Port Richey, Florida, 34652, United States

Location

Unknown Facility

Pembroke Pines, Florida, 33028, United States

Location

Unknown Facility

Detroit, Michigan, 48202, United States

Location

Unknown Facility

Creve Coeur, Missouri, 63141, United States

Location

Unknown Facility

Buffalo, New York, 14215, United States

Location

Unknown Facility

Cincinnati, Ohio, 45206, United States

Location

Unknown Facility

Toledo, Ohio, 43615, United States

Location

Unknown Facility

Oklahoma City, Oklahoma, 73116, United States

Location

Unknown Facility

Nashville, Tennessee, 37212-8150, United States

Location

Unknown Facility

Fort Worth, Texas, 76104, United States

Location

Unknown Facility

Fort Worth, Texas, 76105, United States

Location

Unknown Facility

Fort Worth, Texas, 76164, United States

Location

Unknown Facility

Grand Prairie, Texas, 75050, United States

Location

Unknown Facility

Houston, Texas, 77004, United States

Location

Unknown Facility

Houston, Texas, 77091, United States

Location

Unknown Facility

Mansfield, Texas, 76063, United States

Location

Unknown Facility

Muroran, Hokkaido, 050-0083, Japan

Location

Unknown Facility

Kuwana, Mie-ken, 511-0061, Japan

Location

Unknown Facility

Kyoto, 607-8116, Japan

Location

Related Links

MeSH Terms

Conditions

AnemiaRenal Insufficiency, Chronic

Interventions

molidustat

Condition Hierarchy (Ancestors)

Hematologic DiseasesHemic and Lymphatic DiseasesRenal InsufficiencyKidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Study Officials

  • Bayer Study Director

    Bayer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 14, 2014

First Posted

February 17, 2014

Study Start

March 13, 2014

Primary Completion

October 19, 2016

Study Completion

November 16, 2016

Last Updated

September 20, 2019

Record last verified: 2019-09

Locations