NCT01970215

Brief Summary

The primary objective of this study is to evaluate the efficacy of different doses of TA-8995, a cholesteryl ester transfer protein (CETP) inhibitor, on the elevation of high-density lipoprotein cholesterol (HDL-C) and reduction of low-density lipoprotein cholesterol (LDL-C), alone and in combination with statin therapy. The secondary objectives of this study are to determine the safety and tolerability of TA-8995 in patients with mild dyslipidaemia.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
364

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Aug 2013

Shorter than P25 for phase_2

Geographic Reach
2 countries

17 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2013

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

October 21, 2013

Completed
7 days until next milestone

First Posted

Study publicly available on registry

October 28, 2013

Completed
8 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2014

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2014

Completed
Last Updated

August 21, 2014

Status Verified

August 1, 2014

Enrollment Period

11 months

First QC Date

October 21, 2013

Last Update Submit

August 20, 2014

Conditions

Outcome Measures

Primary Outcomes (1)

  • The co-primary efficacy endpoints are the percentage changes in both HDL-C and LDL-C levels at Week 12 compared to baseline.

    12 weeks

Study Arms (9)

Group 1

PLACEBO COMPARATOR

TA-8995 0mg (placebo) \& placebo statin

Drug: TA-8995 0mg (placebo)Drug: Placebo Statin

Group 2

EXPERIMENTAL

TA-8995 1mg \& placebo statin

Drug: TA-8995Drug: Placebo Statin

Group 3

EXPERIMENTAL

TA-8995 2.5mg \& placebo statin

Drug: TA-8995Drug: Placebo Statin

Group 4

EXPERIMENTAL

TA-8995 5mg \& placebo statin

Drug: TA-8995Drug: Placebo Statin

Group 5

EXPERIMENTAL

TA-8995 10mg \& placebo statin

Drug: TA-8995Drug: Placebo Statin

Group 6

ACTIVE COMPARATOR

TA-8995 0mg (placebo) \& atorvastatin 20mg

Drug: AtorvastatinDrug: TA-8995 0mg (placebo)

Group 7

ACTIVE COMPARATOR

TA-8995 10mg \& atorvastatin 20mg

Drug: TA-8995Drug: Atorvastatin

Group 8

ACTIVE COMPARATOR

TA-8995 0mg (placebo) \& rosuvastatin 10mg

Drug: RosuvastatinDrug: TA-8995 0mg (placebo)

Group 9

ACTIVE COMPARATOR

TA-8995 10mg \& rosuvastatin 10mg

Drug: TA-8995Drug: Rosuvastatin

Interventions

Group 2Group 3Group 4Group 5Group 7Group 9
Group 6Group 7
Group 8Group 9
Group 1Group 6Group 8
Group 1Group 2Group 3Group 4Group 5

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Fasting LDL-C levels \>2.5 mmol/L and \<4.5 mmol/L, HDL-C levels \<1.8 mmol/L and \>0.8 mmol/L, and TG levels \<4.5 mmol/L after run in or washout of existing therapies
  • Not on lipid-altering therapy at screening or on lipid-altering treatment regimens at screening

You may not qualify if:

  • Body mass index \>32 kg/m2;
  • Participation in another clinical study involving an investigational or marketed drug within 30 days prior to enrolment (Visit 2);
  • Any clinical manifestation of atherosclerotic vascular disease;
  • Diagnosis of type 1 diabetes;
  • Uncontrolled type 2 diabetes: haemoglobin A1c \>8%;
  • Uncontrolled hypertension: sitting systolic blood pressure \>160 mmHg and/or sitting diastolic blood pressure \>90 mmHg;
  • History of hyperaldosteronism;
  • Active muscle disease or persistent creatine kinase concentration \>3 Ă— the upper limit of normal (ULN). One retest will be allowed after 1 week to verify the result;

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (17)

H:S Amager Hospital

Copenhagen, Denmark

Location

Sydvestjysk Sygehus

Esbjerg, Denmark

Location

Herlev University Hospital

Herlev, Denmark

Location

Hvidovre Hospital

Hvidovre, Denmark

Location

Regionshopitalet - Silkeborg

Silkeborg, Denmark

Location

EB FlevoResearch B.V

Almere Stad, Netherlands

Location

Andromed Amsterdam

Amsterdam, Netherlands

Location

Andromed Leiden

Amsterdam, Netherlands

Location

Academic Medical Centre

Amsterdam-Zuidoost, Netherlands

Location

Andromed Breda B.V

Breda, Netherlands

Location

Andromed Eindhoven

Eindhoven, Netherlands

Location

Andromed Noord B.V

Groningen, Netherlands

Location

Andromed Zoetermeer

Leiderdorp, Netherlands

Location

Andromed Rotterdam BV

Rotterdam, Netherlands

Location

Albert Schweitzer Ziekenhuis

Sliedrecht, Netherlands

Location

Andromed Oost

Velp, Netherlands

Location

Praktijk Zwijndrecht

Zwijndrecht, Netherlands

Location

Related Publications (3)

  • Martin SS, Ditmarsch M, Simmons M, Alp N, Turner T, Davidson MH, Kastelein JJP. Comparison of low-density lipoprotein cholesterol equations in patients with dyslipidaemia receiving cholesterol ester transfer protein inhibition. Eur Heart J Cardiovasc Pharmacother. 2023 Feb 2;9(2):148-155. doi: 10.1093/ehjcvp/pvac056.

  • van Capelleveen JC, Kastelein JJ, Zwinderman AH, van Deventer SJ, Collins HL, Adelman SJ, Round P, Ford J, Rader DJ, Hovingh GK. Effects of the cholesteryl ester transfer protein inhibitor, TA-8995, on cholesterol efflux capacity and high-density lipoprotein particle subclasses. J Clin Lipidol. 2016 Sep-Oct;10(5):1137-1144.e3. doi: 10.1016/j.jacl.2016.06.006. Epub 2016 Jun 25.

  • Hovingh GK, Kastelein JJ, van Deventer SJ, Round P, Ford J, Saleheen D, Rader DJ, Brewer HB, Barter PJ. Cholesterol ester transfer protein inhibition by TA-8995 in patients with mild dyslipidaemia (TULIP): a randomised, double-blind, placebo-controlled phase 2 trial. Lancet. 2015 Aug 1;386(9992):452-60. doi: 10.1016/S0140-6736(15)60158-1. Epub 2015 Jun 2.

MeSH Terms

Conditions

Dyslipidemias

Interventions

TA-8995AtorvastatinRosuvastatin Calcium

Condition Hierarchy (Ancestors)

Lipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Intervention Hierarchy (Ancestors)

PyrrolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsHeptanoic AcidsFatty AcidsLipidsSulfonamidesAmidesOrganic ChemicalsFluorobenzenesHydrocarbons, FluorinatedHydrocarbons, HalogenatedHydrocarbonsSulfonesSulfur CompoundsPyrimidines

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 21, 2013

First Posted

October 28, 2013

Study Start

August 1, 2013

Primary Completion

July 1, 2014

Study Completion

July 1, 2014

Last Updated

August 21, 2014

Record last verified: 2014-08

Locations