NCT01702194

Brief Summary

The purpose of this study is to determine TD-1211 is processed by the body.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
10

participants targeted

Target at below P25 for phase_1

Timeline
Completed

Started Nov 2012

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 2, 2012

Completed
3 days until next milestone

First Posted

Study publicly available on registry

October 5, 2012

Completed
27 days until next milestone

Study Start

First participant enrolled

November 1, 2012

Completed
3 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2013

Completed
28 days until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2013

Completed
Last Updated

January 20, 2021

Status Verified

January 1, 2021

Enrollment Period

3 months

First QC Date

October 2, 2012

Last Update Submit

January 15, 2021

Conditions

Keywords

OICOpioid Induced ConstipationConstipation

Outcome Measures

Primary Outcomes (5)

  • Area under the plasma concentration versus time curve (AUC)

    0 to 168 hours postdose

  • Peak plasma concentration (Cmax)

    0 to 168 hours postdose

  • Time to peak plasma concentration (Tmax)

    0 to 168 hours postdose

  • Half-life (T 1/2)

    0 to 168 hours postdose

  • Percent total recovery of radioactivity in blood, urine, and feces

    0 to 312 hours postdose

Secondary Outcomes (1)

  • Number of participants with adverse events

    Baseline to 14 days

Study Arms (2)

TD-1211 IV [C14]

EXPERIMENTAL

TD-1211 IV \[C14\]

Drug: TD-1211 IV [C14]

TD-1211 PO [C14]

EXPERIMENTAL

TD-1211 PO \[C14\]

Drug: TD-1211 PO [C14]

Interventions

Also known as: TD-1211
TD-1211 IV [C14]
Also known as: TD-1211
TD-1211 PO [C14]

Eligibility Criteria

Age18 Years - 50 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy, nonsmoking male, 18 to 50 years old, inclusive.
  • Agrees to use a highly effective method of birth control.
  • Body mass index (BMI) 19 to 30 kg/m2, inclusive, and weighs at least 55 kg.
  • Willing and able to give written informed consent.

You may not qualify if:

  • Evidence or history of clinically significant allergic (except for untreated, asymptomatic, seasonal allergies at time of dosing), hematological, endocrine, pulmonary, gastrointestinal, cardiovascular, hepatic, psychiatric, or neurological disease.
  • Hemoglobin \<14.1 g/dL or hematocrit \< 40.6% at Screening.
  • History of hypersensitivity to drugs, or a history of or any current clinically significant hypersensitivities.
  • Any condition possibly affecting drug absorption (e.g., previous surgery on the gastrointestinal tract \[including removal of parts of the stomach, bowel, liver, gall bladder, or pancreas\]).
  • Participated in another clinical trial of an investigational drug (or medical device) within 60 days (or 5 half-lives of the investigational drug, whichever is longer) prior to Screening, or is currently participating in another trial of an investigational drug (or medical device).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Covance

Madison, Wisconsin, 53704, United States

Location

MeSH Terms

Conditions

Opioid-Induced ConstipationConstipation

Interventions

Carbon-143-(8-(2-(cyclohexylmethyl(2,3-dihydroxypropionyl)amino)ethyl)-8-azabicyclo(3.2.1)oct-3-yl)benzamide

Condition Hierarchy (Ancestors)

Signs and Symptoms, DigestiveSigns and SymptomsPathological Conditions, Signs and SymptomsNarcotic-Related DisordersSubstance-Related DisordersChemically-Induced DisordersMental Disorders

Study Officials

  • Medical Monitor

    Theravance Biopharma

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 2, 2012

First Posted

October 5, 2012

Study Start

November 1, 2012

Primary Completion

February 1, 2013

Study Completion

March 1, 2013

Last Updated

January 20, 2021

Record last verified: 2021-01

Locations