NCT01440166

Brief Summary

  • To evaluate the safety and tolerability of escalating single doses of CAT-1004 relative to placebo in healthy adult volunteers.
  • To evaluate the pharmacokinetics (PK) of escalating single doses of CAT-1004 in healthy adult volunteers.
  • To evaluate the effect of a high-fat meal on single doses of CAT-1004 in healthy adult volunteers.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
52

participants targeted

Target at P50-P75 for phase_1 healthy

Timeline
Completed

Started Sep 2011

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2011

Completed
7 days until next milestone

First Submitted

Initial submission to the registry

September 8, 2011

Completed
18 days until next milestone

First Posted

Study publicly available on registry

September 26, 2011

Completed
3 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2012

Completed
Last Updated

February 6, 2012

Status Verified

February 1, 2012

Enrollment Period

4 months

First QC Date

September 8, 2011

Last Update Submit

February 2, 2012

Conditions

Keywords

Human healthy volunteers

Outcome Measures

Primary Outcomes (1)

  • Safety

    Safety Endpoints: Laboratory evaluations including hematology, chemistry, coagulation and urinalysis, physical examinations, AEs, serious AEs (SAEs), ECGs, and vital signs.

    Change from Baseline versus Day-1 though 72 hrs post dose and EOT/FU

Secondary Outcomes (1)

  • Pharmacokinetic Profile

    Plasma blood samples through 72 hrs, urine collections through 48 hrs

Study Arms (9)

Cohort 1 / Dose level 1

EXPERIMENTAL

Single dose orally: CAT-1004 Dose level 1 or placebo

Drug: DrugOther: Placebo

Cohort 2 / Dose level 2

EXPERIMENTAL

Single dose orally: CAT-1004 Dose level 2 or placebo

Drug: DrugOther: Placebo

Cohort 3 /Dose level 3

EXPERIMENTAL

Single dose orally: CAT-1004 Dose level 3 or placebo

Drug: DrugOther: Placebo

Cohort 4/ Dose level 4

EXPERIMENTAL

Single dose orally: CAT-1004 Dose level 4 or placebo

Drug: DrugOther: Placebo

Cohort 5/ Dose level 5

EXPERIMENTAL

Single dose orally: CAT-1004 Dose level 5 or placebo

Drug: DrugOther: Placebo

Cohort 2/ Dose level 2 ( FE)

EXPERIMENTAL

Single dose orally (Under fed conditions): CAT-1004 Dose level 2 or placebo

Drug: DrugOther: Placebo

Cohort 3/ Dose level 3 (FE)

EXPERIMENTAL

Single dose orally (Under fed conditions): CAT-1004 Dose level 3 or placebo

Drug: DrugOther: Placebo

Cohort 6 / Dose level 6 (FE)

EXPERIMENTAL

Single dose orally (Under fed conditions) CAT-1004 Dose level 4 or placebo Subjects may be reenrolled from Cohort 4.

Drug: DrugOther: Placebo

Cohort 7 / Dose level 7 (FE)

EXPERIMENTAL

Single dose orally (Under fed conditions)CAT-1004 Dose level 5 or placebo Subjects may be reenrolled from Cohort 5.

Drug: DrugOther: Placebo

Interventions

DrugDRUG

Single dose oral administration of CAT1004 or placebo-6 to 8 subjects will be treated with CAT-1004 per cohort.

Also known as: CAT-1004
Cohort 1 / Dose level 1Cohort 2 / Dose level 2Cohort 2/ Dose level 2 ( FE)Cohort 3 /Dose level 3Cohort 3/ Dose level 3 (FE)Cohort 4/ Dose level 4Cohort 5/ Dose level 5Cohort 6 / Dose level 6 (FE)Cohort 7 / Dose level 7 (FE)
PlaceboOTHER

Single dose oral administration of CAT1004 or placebo- 2 subjects treated with placebo per cohort.

Cohort 1 / Dose level 1Cohort 2 / Dose level 2Cohort 2/ Dose level 2 ( FE)Cohort 3 /Dose level 3Cohort 3/ Dose level 3 (FE)Cohort 4/ Dose level 4Cohort 5/ Dose level 5Cohort 6 / Dose level 6 (FE)Cohort 7 / Dose level 7 (FE)

Eligibility Criteria

Age19 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • In good health.
  • Age: 19 to 55 years inclusive at Screening.
  • Satisfies one of the following
  • Females not of childbearing potential: non-pregnant and non-lactating; surgically sterile or postmenopausal, OR
  • Males: surgically sterile, abstinent, or subject or partner is utilizing an acceptable contraceptive method during and 3 months after the last study dose.
  • BMI: 18 to 30 kg/m2 at Screening.

You may not qualify if:

  • Clinically significant abnormalities in physical examination or vital signs.
  • Clinically significant electrocardiogram (ECG) abnormalities as assessed by the investigator.
  • Clinically significant screening laboratory result as assessed by the Investigator.
  • The subject has a history of clinically significant allergies (except for untreated, asymptomatic seasonal allergies at the time of dosing), or hematological, endocrine, pulmonary, gastrointestinal, cardiovascular, hepatic, psychiatric, or neurological disease.
  • History or presence of malignancy with the past 5 years.
  • History of alcohol or substance abuse or eating disorder within 2 years, OR regular use of alcohol within 6 months (\>14 units of alcohol per week; 1 unit = 150 mL of wine, 360 mL of beer, or 45 mL of 40% alcohol).
  • Use of any investigational drug or participation in any investigational study within 30 days prior to screening. For dose levels 6 and 7 fed cohorts, subjects may participate who have taken part in the dose levels 4 and 5 fasted cohort.
  • Any significant blood loss within 60 days prior to screening, e.g. blood donation, participation in study with multiple blood draws, etc.
  • Any condition, disease, disorder or clinically relevant laboratory abnormality that, in the opinion of the Investigator, would jeopardize the subject's appropriate participation in this study or obscure the effects of treatment.
  • A suspected allergy or sensitivity to CAT-1004 or excipients based upon known allergies to excipients or compounds of a similar class.
  • Any clinically significant systemic infection within 3 weeks prior to screening.
  • Use of prescription medications within 30 days of screening.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Celerion Clinical Research Unit

Lincoln, Nebraska, 68502, United States

Location

MeSH Terms

Interventions

Pharmaceutical Preparationsedasalonexent

Study Officials

  • Scott Rasmussen, MD

    Celerion

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 8, 2011

First Posted

September 26, 2011

Study Start

September 1, 2011

Primary Completion

January 1, 2012

Study Completion

January 1, 2012

Last Updated

February 6, 2012

Record last verified: 2012-02

Locations