NCT01410383

Brief Summary

Eprotirome is a liver selective thyroid hormone that can reduce several independent risk factors for cardiovascular disease, while an euthyroid state is preserved in the extrahepatic tissue. The purpose of this Phase III study is to assess the long-term efficacy and safety of Eprotirome in Patients with heterozygous Familial Hypercholesterolaemia who are on optimal standard of care.

Trial Health

55
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
236

participants targeted

Target at P25-P50 for phase_3

Timeline
Completed

Started Oct 2011

Typical duration for phase_3

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

July 13, 2011

Completed
23 days until next milestone

First Posted

Study publicly available on registry

August 5, 2011

Completed
2 months until next milestone

Study Start

First participant enrolled

October 1, 2011

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2013

Completed
1 year until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2014

Completed
Last Updated

September 3, 2012

Status Verified

August 1, 2012

Enrollment Period

2 years

First QC Date

July 13, 2011

Last Update Submit

August 31, 2012

Conditions

Keywords

hypercholesterolemia,dyslipidemia,thyroid,safety,Heterozygous Familial Hypercholesterolaemiacoronary artery disease

Outcome Measures

Primary Outcomes (1)

  • Percent reduction in low-density lipoprotein cholesterol (LDL-C) from baseline

    12 weeks treatment

Study Arms (3)

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Eprotirome I

EXPERIMENTAL
Drug: Eprotirome

Eprotirome II

EXPERIMENTAL
Drug: Eprotirome

Interventions

Tablets taken daily

Placebo

Tablets taken daily

Also known as: KB2115
Eprotirome I

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Patients with confirmed HeFH and 18 years of age at screening
  • Presence of clinical atherosclerotic disease that confers high risk for CAD events together with an LDL-C more than 2 mmol/L (more than 80 mg/dL)
  • Presence of risk factors for CVD (other than the HeFH diagnosis) together with an LDL-C more than 2.5 mmol/L (more than 100 mg/dL)
  • On an optimal standard of care, defined as being on a stable dose of statin (rosuvastatin, atorvastatin, or simvastatin) with or without ezetimibe for 8 weeks prior to randomisation

You may not qualify if:

  • Significant health problems in recent past including heart failure,cardiac electrophysiologic instability, rheumatoid arthritis, thyroid dysfunction, liver disease, cancer, secondary dyslipidaemia

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Related Publications (1)

  • Sjouke B, Langslet G, Ceska R, Nicholls SJ, Nissen SE, Ohlander M, Ladenson PW, Olsson AG, Hovingh GK, Kastelein JJ. Eprotirome in patients with familial hypercholesterolaemia (the AKKA trial): a randomised, double-blind, placebo-controlled phase 3 study. Lancet Diabetes Endocrinol. 2014 Jun;2(6):455-63. doi: 10.1016/S2213-8587(14)70006-3. Epub 2014 Feb 18.

MeSH Terms

Conditions

HypercholesterolemiaDyslipidemiasThyroid DiseasesCoronary Artery Disease

Interventions

3-((3,5-dibromo-4-(4-hydroxy-3-(1-methylethyl)phenoxy)phenyl)amino)-3-oxopropanoic acid

Condition Hierarchy (Ancestors)

HyperlipidemiasLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesCoronary DiseaseMyocardial IschemiaHeart DiseasesCardiovascular DiseasesArteriosclerosisArterial Occlusive DiseasesVascular Diseases

Study Officials

  • John Kastelein, Professor

    Academic Medical Center (AMC) of the University of Amsterdam

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

July 13, 2011

First Posted

August 5, 2011

Study Start

October 1, 2011

Primary Completion

October 1, 2013

Study Completion

October 1, 2014

Last Updated

September 3, 2012

Record last verified: 2012-08