NCT01328821

Brief Summary

The purpose of this study is to assess the safety, tolerability and pharmacokinetics of CTP-499 following single dose administration.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
38

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Mar 2011

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2011

Completed
29 days until next milestone

First Submitted

Initial submission to the registry

March 30, 2011

Completed
2 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2011

Completed
4 days until next milestone

First Posted

Study publicly available on registry

April 5, 2011

Completed
2 months until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2011

Completed
Last Updated

October 26, 2011

Status Verified

June 1, 2011

Enrollment Period

1 month

First QC Date

March 30, 2011

Last Update Submit

October 25, 2011

Conditions

Keywords

SafetyTolerabilityPharmacokineticsHealthy volunteers

Outcome Measures

Primary Outcomes (1)

  • To assess safety and tolerability of CTP-499

    Assessments will include monitoring of adverse events, vital signs (blood pressure, pulse rate, respiratory rate and oral temperature), clinical laboratory findings, 12 lead ECGs, and physical examination findings. Safety data will be summarized using descriptive statistics for all subjects who receive at least 1 dose. Adverse events will be summarized by frequency. Abnormal laboratory and physical exam findings will be summarized by dose and treatment.

    5 days

Secondary Outcomes (1)

  • To assess Pharmacokinetics, Pharmacodynamics and relative bioavailability

    2 days

Study Arms (2)

Part A

PLACEBO COMPARATOR

Single ascending dose administration of four doses of CTP-499 as tablets under fasting condition. 8 subjects per dose group will be enrolled with a 3:1 randomization of active drug to placebo. Dose levels: 600mg -\> 1200mg -\> 1800mg -\> 2400mg

Drug: CTP-499

Part B

ACTIVE COMPARATOR

Part B will consist of a single 400 mg dose of an immediate release capsule of CTP-499 administered under fasting conditions. In Part B 6 subjects will be enrolled.

Drug: CTP-499

Interventions

600 mg, 1200 mg, 1800 mg and 2400 mg

Part A

Eligibility Criteria

Age18 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • healthy volunteers
  • ages 18 to 55 years old
  • nonsmokers
  • BMI of 18 to 30 kg/m2

You may not qualify if:

  • Significant history of gastrointestinal, cardiovascular, musculoskeletal, endocrine, hematologic, psychiatric, renal, hepatic, bronchopulmonary, neurologic, immunologic, lipid metabolism disorders of drug hypersensitivity
  • Systolic Blood pressure \< 90 or \> 140, diastolic bp \> 90

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Frontage

Hackensack, New Jersey, 07601, United States

Location

MeSH Terms

Conditions

Diabetic Nephropathies

Interventions

1-(5-hydroxyhexyl)-3,7-dimethylxanthine

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesDiabetes ComplicationsDiabetes MellitusEndocrine System Diseases

Study Officials

  • Gregory Tracey, MD

    Frontage Clinical Services

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 30, 2011

First Posted

April 5, 2011

Study Start

March 1, 2011

Primary Completion

April 1, 2011

Study Completion

June 1, 2011

Last Updated

October 26, 2011

Record last verified: 2011-06

Locations